AP4E1

UniProt ID: Q9UPM8
Organism: Homo sapiens
Review Status: COMPLETE
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Gene Description

AP4E1 encodes the epsilon large subunit of the heterotetrameric AP-4 adaptor complex. AP-4 forms a nonclathrin coat on the cytoplasmic face of the trans-Golgi network and sorts membrane proteins into transport carriers. The epsilon N-terminal trunk contributes to the complex core and binds activated ARF1 for membrane recruitment, while its C-terminal ear binds the accessory protein tepsin. These interactions support coat assembly and cargo transport in coordination with the mu4 cargo-recognition subunit.

Existing Annotations Review

GO Term Evidence Action Reason
GO:0005515 protein binding
IPI
PMID:26496610
A human interactome in three quantitative dimensions organiz...
UNDECIDED
Summary: The original TEPSIN screen experiment remains unadjudicated.
Reason: The exact pair-specific supplementary entry, constructs and controls in this source were not independently inspected. Separate human epsilon–tepsin binding and recruitment experiments establish the partnership but do not adjudicate this particular screen record. Preserve the original assertion as uncertain without denying the interaction or transferring a different paper’s mechanistic evidence into its source fields.
GO:0005515 protein binding
IPI
PMID:26542808
Bivalent Motif-Ear Interactions Mediate the Association of t...
MODIFY
Summary: The epsilon appendage recruits tepsin to the AP-4 machinery.
Reason: Human epsilon ear binding to a defined tepsin peptide is supported by ITC, motif perturbation and reduced cellular recruitment. Epsilon incorporation into AP-4 supplies the second side of the bridge, so accessory-factor recruitment supports protein-macromolecule adaptor activity. AP-4 crosslinking is a proposed model. This refinement does not assign direct cargo-motif recognition or HOOK binding to epsilon. The parent adaptor term here describes epsilon-mediated accessory recruitment tested in this paper, whereas the inherited cargo-adaptor term describes the assembled heterotetramer with mu4 cargo recognition. These are distinct interfaces; no new ancestor annotation is added.
Supporting Evidence:
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:10066790
beta4 is a component of a multisubunit complex (AP-4) that also contains the sigma4 polypeptide and two additional adaptor subunit homologs named mu4 (mu-ARP2) and epsilon.
file:human/AP4E1/AP4E1-notes.md
GO:0005515 protein binding
IPI
PMID:32073997
The FTS-Hook-FHIP (FHF) complex interacts with AP-4 to media...
KEEP AS NON CORE
Summary: The human epsilon–tepsin Y2H positive control supports the partner interaction.
Reason: The original Results and Figure 3 include an inspected human epsilon–tepsin Y2H positive control. Retain that observed partner interaction as non-core. This pair assay does not itself demonstrate an adaptor bridge, and the separate recruitment experiments in PMID:26542808 are not substituted for it. Genericity alone does not establish that an experimentally observed interaction is incorrect. Direct HOOK binding elsewhere in the study belongs to mu4 and is not assigned to epsilon. The original-body result and public locator are recorded in notes; the normal cache remains abstract-only.
Supporting Evidence:
file:human/AP4E1/AP4E1-notes.md
Control experiments showed interactions of tepsin with AP-4 Ξ΅ and AP-4 Ξ²4
GO:0005515 protein binding
IPI
PMID:33961781
Dual proteome-scale networks reveal cell-specific remodeling...
UNDECIDED
Summary: The original TEPSIN screen experiment remains unadjudicated.
Reason: The exact pair-specific supplementary entry, constructs and controls in this source were not independently inspected. Separate human epsilon–tepsin binding and recruitment experiments establish the partnership but do not adjudicate this particular screen record. Preserve the original assertion as uncertain without denying the interaction or transferring a different paper’s mechanistic evidence into its source fields.
GO:0005768 endosome
IEA
GO_REF:0000117
UNDECIDED
Summary: A distinct endosomal pool is not resolved by the available target evidence.
Reason: AP-4 is enriched on the cytoplasmic face of the TGN. This does not exclude a transient endosomal pool. The actual ARBA00028568 inference chain has not been inspected, and delivery of APP cargo to endosomes does not by itself establish adaptor residence there. The broad endosome assertion therefore remains uncertain; the enclosed-lumen topology objection is a separate issue.
Supporting Evidence:
PMID:11707398
localizes to the cytoplasmic face of the trans-Golgi network (TGN).
file:human/AP4E1/AP4E1-notes.md
GO:0005794 Golgi apparatus
IEA
GO_REF:0000044
MODIFY
Summary: Refine the broad Golgi/TGN compartment to its membrane-associated AP-4 pool.
Reason: Human biochemical evidence places AP-4 on the cytoplasmic face of the TGN, where ARF1 recruits the epsilon-containing complex. The peripheral membrane pool is more precise than the broad compartment; this does not imply epsilon spans the bilayer.
Proposed replacements: trans-Golgi network membrane
Supporting Evidence:
PMID:11707398
localizes to the cytoplasmic face of the trans-Golgi network (TGN).
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0005802 trans-Golgi network
IEA
GO_REF:0000117
MODIFY
Summary: Refine the broad Golgi/TGN compartment to its membrane-associated AP-4 pool.
Reason: Human biochemical evidence places AP-4 on the cytoplasmic face of the TGN, where ARF1 recruits the epsilon-containing complex. The peripheral membrane pool is more precise than the broad compartment; this does not imply epsilon spans the bilayer.
Proposed replacements: trans-Golgi network membrane
Supporting Evidence:
PMID:11707398
localizes to the cytoplasmic face of the trans-Golgi network (TGN).
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0005802 trans-Golgi network
NAS
PMID:10436028
Characterization of a fourth adaptor-related protein complex...
MODIFY
Summary: Refine the broad Golgi/TGN compartment to its membrane-associated AP-4 pool.
Reason: Human biochemical evidence places AP-4 on the cytoplasmic face of the TGN, where ARF1 recruits the epsilon-containing complex. The peripheral membrane pool is more precise than the broad compartment; this does not imply epsilon spans the bilayer.
Proposed replacements: trans-Golgi network membrane
Supporting Evidence:
PMID:11707398
localizes to the cytoplasmic face of the trans-Golgi network (TGN).
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0006605 protein targeting
IC
PMID:10066790
AP-4, a novel protein complex related to clathrin adaptors.
ACCEPT
Summary: AP-4 coat assembly and cargo sorting support this protein-transport or localization assertion.
Reason: Epsilon is part of the AP-4 machinery that sorts membrane-protein cargo into carriers at the TGN. This supports the existing protein-specific targeting, localization or transport term. The original annotation remains valid even though vesicle-mediated transport describes a complementary mechanistic aspect. Replacing it with that already-present term would discard protein-cargo information and add no coverage. No downstream cargo chemistry is assigned to epsilon.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
GO:0006886 intracellular protein transport
IEA
GO_REF:0000002
ACCEPT
Summary: AP-4 coat assembly and cargo sorting support this protein-transport or localization assertion.
Reason: Epsilon is part of the AP-4 machinery that sorts membrane-protein cargo into carriers at the TGN. This supports the existing protein-specific targeting, localization or transport term. The original annotation remains valid even though vesicle-mediated transport describes a complementary mechanistic aspect. Replacing it with that already-present term would discard protein-cargo information and add no coverage. No downstream cargo chemistry is assigned to epsilon.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
GO:0008104 intracellular protein localization
IC
PMID:10066790
AP-4, a novel protein complex related to clathrin adaptors.
ACCEPT
Summary: AP-4 coat assembly and cargo sorting support this protein-transport or localization assertion.
Reason: Epsilon is part of the AP-4 machinery that sorts membrane-protein cargo into carriers at the TGN. This supports the existing protein-specific targeting, localization or transport term. The original annotation remains valid even though vesicle-mediated transport describes a complementary mechanistic aspect. Replacing it with that already-present term would discard protein-cargo information and add no coverage. No downstream cargo chemistry is assigned to epsilon.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
GO:0008104 intracellular protein localization
IEA
GO_REF:0000117
ACCEPT
Summary: AP-4 coat assembly and cargo sorting support this protein-transport or localization assertion.
Reason: Epsilon is part of the AP-4 machinery that sorts membrane-protein cargo into carriers at the TGN. This supports the existing protein-specific targeting, localization or transport term. The original annotation remains valid even though vesicle-mediated transport describes a complementary mechanistic aspect. Replacing it with that already-present term would discard protein-cargo information and add no coverage. No downstream cargo chemistry is assigned to epsilon.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
GO:0015031 protein transport
IEA
GO_REF:0000002
ACCEPT
Summary: AP-4 coat assembly and cargo sorting support this protein-transport or localization assertion.
Reason: Epsilon is part of the AP-4 machinery that sorts membrane-protein cargo into carriers at the TGN. This supports the existing protein-specific targeting, localization or transport term. The original annotation remains valid even though vesicle-mediated transport describes a complementary mechanistic aspect. Replacing it with that already-present term would discard protein-cargo information and add no coverage. No downstream cargo chemistry is assigned to epsilon.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
GO:0016192 vesicle-mediated transport
IEA
GO_REF:0000002
ACCEPT
Summary: AP4E1 participates in vesicle-mediated transport as an AP-4 coat subunit.
Reason: AP-4 is a nonclathrin carrier coat. Epsilon contributes the structural core, ARF1-dependent membrane recruitment and an accessory-protein-binding ear. These are direct roles in transport machinery, rather than an inference from a downstream cargo phenotype.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
GO:0016192 vesicle-mediated transport
NAS
PMID:10436028
Characterization of a fourth adaptor-related protein complex...
ACCEPT
Summary: AP4E1 participates in vesicle-mediated transport as an AP-4 coat subunit.
Reason: AP-4 is a nonclathrin carrier coat. Epsilon contributes the structural core, ARF1-dependent membrane recruitment and an accessory-protein-binding ear. These are direct roles in transport machinery, rather than an inference from a downstream cargo phenotype.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
GO:0030117 membrane coat
IEA
GO_REF:0000002
MODIFY
Summary: The membrane-coat assignment can be specified as AP-4.
Reason: Epsilon is an experimentally established component of the heterotetrameric AP-4 coat. Use this specific complex instead of the broad coat parent; clathrin binding is not assigned.
Proposed replacements: AP-4 adaptor complex
Supporting Evidence:
PMID:10066790
beta4 is a component of a multisubunit complex (AP-4) that also contains the sigma4 polypeptide and two additional adaptor subunit homologs named mu4 (mu-ARP2) and epsilon.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0030124 AP-4 adaptor complex
IBA
GO_REF:0000033
ACCEPT
Summary: Epsilon is a structural subunit of the AP-4 heterotetramer.
Reason: Human-cell biochemical complex characterization and purified human AP-4 structural work support epsilon membership with beta4, mu4 and sigma4. The PAINT node and all donors are retained. Target self-inclusion is legitimate descendant evidence, not circularity; the exact ancestral placement has not been independently reconstructed.
Supporting Evidence:
PMID:10066790
beta4 is a component of a multisubunit complex (AP-4) that also contains the sigma4 polypeptide and two additional adaptor subunit homologs named mu4 (mu-ARP2) and epsilon.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0030124 AP-4 adaptor complex
IDA
PMID:10066790
AP-4, a novel protein complex related to clathrin adaptors.
ACCEPT
Summary: Epsilon is a structural subunit of the AP-4 heterotetramer.
Reason: Human-cell biochemical complex characterization and purified human AP-4 structural work support epsilon membership with beta4, mu4 and sigma4.
Supporting Evidence:
PMID:10066790
beta4 is a component of a multisubunit complex (AP-4) that also contains the sigma4 polypeptide and two additional adaptor subunit homologs named mu4 (mu-ARP2) and epsilon.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0030124 AP-4 adaptor complex
IEA
GO_REF:0000002
ACCEPT
Summary: Epsilon is a structural subunit of the AP-4 heterotetramer.
Reason: Human-cell biochemical complex characterization and purified human AP-4 structural work support epsilon membership with beta4, mu4 and sigma4.
Supporting Evidence:
PMID:10066790
beta4 is a component of a multisubunit complex (AP-4) that also contains the sigma4 polypeptide and two additional adaptor subunit homologs named mu4 (mu-ARP2) and epsilon.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0030124 AP-4 adaptor complex
NAS
PMID:10436028
Characterization of a fourth adaptor-related protein complex...
ACCEPT
Summary: Epsilon is a structural subunit of the AP-4 heterotetramer.
Reason: Human-cell biochemical complex characterization and purified human AP-4 structural work support epsilon membership with beta4, mu4 and sigma4.
Supporting Evidence:
PMID:10066790
beta4 is a component of a multisubunit complex (AP-4) that also contains the sigma4 polypeptide and two additional adaptor subunit homologs named mu4 (mu-ARP2) and epsilon.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-5229111
REMOVE
Summary: The cargo destination in the Reactome event does not place epsilon inside the endosome lumen.
Reason: The cited event describes APP delivery and recognition of its cytoplasmic tail by mu4. GO0031904 is the enclosed endosomal volume. AP-4 instead forms a cytoplasm-facing coat recruited through epsilon–ARF1 contacts. Assigning that coat subunit to the cargo destination lumen conflicts with this topology. This is a source-specific TAS compartment correction; it does not claim a wrong experimental paper or exclude every endosome-associated pool.
Supporting Evidence:
PMID:11707398
localizes to the cytoplasmic face of the trans-Golgi network (TGN).
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
file:human/AP4E1/AP4E1-notes.md
Reactome:R-HSA-5229111
GO:0032588 trans-Golgi network membrane
TAS
Reactome:R-HSA-5229111
ACCEPT
Summary: AP-4 assembles at the trans-Golgi network membrane.
Reason: Both Reactome APP events place the initial AP-4 cargo-recognition machinery at the TGN. Human biochemical and structural studies independently support a cytoplasmic peripheral-membrane coat, with epsilon directly engaging ARF1.
Supporting Evidence:
PMID:11707398
localizes to the cytoplasmic face of the trans-Golgi network (TGN).
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
Reactome:R-HSA-5229111
GO:0032588 trans-Golgi network membrane
TAS
Reactome:R-HSA-5229132
ACCEPT
Summary: AP-4 assembles at the trans-Golgi network membrane.
Reason: Both Reactome APP events place the initial AP-4 cargo-recognition machinery at the TGN. Human biochemical and structural studies independently support a cytoplasmic peripheral-membrane coat, with epsilon directly engaging ARF1.
Supporting Evidence:
PMID:11707398
localizes to the cytoplasmic face of the trans-Golgi network (TGN).
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
Reactome:R-HSA-5229132
GO:0045184 establishment of protein localization
IEA
GO_REF:0000117
ACCEPT
Summary: AP-4 coat assembly and cargo sorting support this protein-transport or localization assertion.
Reason: Epsilon is part of the AP-4 machinery that sorts membrane-protein cargo into carriers at the TGN. This supports the existing protein-specific targeting, localization or transport term. The original annotation remains valid even though vesicle-mediated transport describes a complementary mechanistic aspect. Replacing it with that already-present term would discard protein-cargo information and add no coverage. No downstream cargo chemistry is assigned to epsilon.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
GO:0140312 cargo adaptor activity
IBA
GO_REF:0000033
ACCEPT
Summary: Epsilon contributes to AP-4 cargo-adaptor activity.
Reason: The inherited adaptor-family function agrees with the demonstrated human AP-4 coat. Epsilon helps assemble and recruit the complex and its accessory factor; mu4 supplies the characterized cargo-motif binding site. The source enables qualifier and PAINT node are preserved, while the core synthesis describes the activity as contributed within the heterotetramer. Donor count alone is not a confidence test, and no new ancestral placement is asserted.
Supporting Evidence:
PMID:10436028
Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.
PMID:26542808
Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
GO:0031267 small GTPase binding
IPI
PMID:11707398
Functional and physical interactions of the adaptor protein ...
NEW
Summary: Human epsilon directly binds activated ARF1 through its N-terminal trunk.
Reason: The original human-epsilon experiments compare GTP-locked and GDP-preferring ARF1, epsilon truncations and switch-I/II mutants in Y2H and in-vitro-translated binding assays. A negative short epsilon fragment still binds sigma4, providing a functional control. Independent recombinant human AP-4 experiments map the ARF1 interface to epsilon and test interface mutations. This is a specific ARF1-effector interaction, separate from the TEPSIN partnerships in the existing generic-binding rows. It does not assign GTP hydrolysis, exchange activity or mu4 cargo recognition to epsilon.
Supporting Evidence:
PMID:11707398
epsilon binds only to ARF1-GTP and requires residues in the switch I and switch II regions of ARF1.
PMID:11707398
ARF1Ξ”17-Q71L-myc but not ARF1Ξ”17-T31N-myc was found to co-precipitate with Ξ΅ 1–727
PMID:11707398
The cDNA for the Ξ΅ subunit of AP-4 was obtained by RT–PCR using gene-specific primers and total HeLa cell RNA.
PMID:41565640
Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.

Core Functions

Within AP-4, epsilon contributes the structural and membrane-recruitment side of a cargo-adaptor mechanism. Its trunk assembles into the heterotetramer and directly engages activated ARF1; its ear recruits tepsin. Together these contacts support formation of cytoplasmic carriers at the TGN. Cargo-motif recognition is supplied by mu4, so the cargo-adaptor activity is contributed in the complex rather than attributed to isolated epsilon.

Supporting Evidence:
  • PMID:10066790
    beta4 is a component of a multisubunit complex (AP-4) that also contains the sigma4 polypeptide and two additional adaptor subunit homologs named mu4 (mu-ARP2) and epsilon.
  • PMID:26542808
    Both peptide-ear interactions are required for efficient association of tepsin with AP-4, and for recruitment of tepsin to the TGN.
  • PMID:41565640
    Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.
  • PMID:11707398
    localizes to the cytoplasmic face of the trans-Golgi network (TGN).
  • PMID:10436028
    Immunogold electron microscopy indicates that AP-4 is associated with nonclathrin-coated vesicles in the region of the trans-Golgi network.

The epsilon trunk binds activated ARF1 and provides a regulated membrane-recruitment contact for AP-4. Epsilon is an ARF effector rather than a GTPase, exchange factor or activating protein.

Molecular Function:
small GTPase binding
Cellular Locations:
Supporting Evidence:
  • PMID:11707398
    epsilon binds only to ARF1-GTP and requires residues in the switch I and switch II regions of ARF1.
  • PMID:11707398
    ARF1Ξ”17-Q71L-myc but not ARF1Ξ”17-T31N-myc was found to co-precipitate with Ξ΅ 1–727
  • PMID:11707398
    The cDNA for the Ξ΅ subunit of AP-4 was obtained by RT–PCR using gene-specific primers and total HeLa cell RNA.
  • PMID:41565640
    Collectively, our structural and biochemical data demonstrated direct interaction between the N-terminal region of Ξ΅ and ARF1 in the AP-4/ARF1 complex.

References

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Suggested Questions for Experts

Q: Does endogenous human AP4E1 occupy a measurable endosomal membrane pool distinct from its TGN pool, and what evidence drives ARBA00028568?

Q: How does bivalent tepsin recruitment organize the AP-4 coat; does it bridge AP-4 complexes in a reconstituted human system?

Q: What contribution does epsilon ARF1 binding make to cargo selection beyond the mu4 recognition interface?

Suggested Experiments

Experiment: Quantify endogenous epsilon localization using a validated knock-in tag, TGN and endosomal markers, and correlative imaging to distinguish transient membrane residence from cargo destination.

Experiment: Reconstitute full-length human AP-4 with ARF1, membrane cargo and tepsin, comparing epsilon ear and ARF1-interface mutants to test recruitment and coat organization directly.

πŸ“š Additional Documentation

Notes

(AP4E1-notes.md)

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