APP

UniProt ID: P05067
Organism: Homo sapiens
Review Status: COMPLETE
πŸ“ Provide Detailed Feedback

Gene Description

Amyloid-beta precursor protein (APP) is a type I transmembrane glycoprotein that undergoes regulated proteolytic processing to generate soluble ectodomains, membrane-tethered C-terminal fragments, amyloid-beta peptides, and the APP intracellular domain. Full-length APP acts at the neuronal cell surface and in secretory/endocytic compartments, where it contributes to cell adhesion, synaptogenesis, neurite outgrowth, axonogenesis, and interactions with extracellular matrix ligands. Alternative splice isoforms differ in inclusion of the Kunitz protease inhibitor domain, giving APP751/770 protease-inhibitor activity that is absent from neuronal APP695. APP and amyloid-beta fragments bind transition metals, especially copper and zinc, linking the ectodomain and cleavage products to metal homeostasis and redox biology. In Alzheimer disease, familial APP variants and APP dosage alter amyloidogenic processing and the production or aggregation of amyloid-beta species.

Functional Isoforms

Curated functional classes representing distinct biological activities. These may be splice variants, cleavage products, or other forms with different functions.

APP695 (Neuronal) SPLICE CLASS
ID: APP_695_NEURONAL
UNIPROT ISOFORM: P05067-4
Brain-predominant isoform lacking the KPI (Kunitz protease inhibitor) domain encoded by exon 7. APP695 is the major isoform in neurons and is the primary substrate for amyloidogenic processing in the brain. Does NOT have serine protease inhibitor activity. The ratio of APP695 to KPI-containing isoforms decreases with aging and in Alzheimer's disease.
Isoform-specific terms: neuron projection development
APP751/770 (KPI-containing) SPLICE CLASS
ID: APP_KPI_CONTAINING
UNIPROT ISOFORM: P05067-1, P05067-8
Peripheral isoforms containing the KPI (Kunitz protease inhibitor) domain. APP770 (P05067-1) also has the OX-2 domain. These isoforms have serine protease inhibitor activity that APP695 lacks. Predominantly expressed in non-neuronal tissues. May regulate coagulation and inflammation.
Isoform-specific terms: serine-type endopeptidase inhibitor activity
sAPPalpha (Soluble APP-alpha) CLEAVAGE PRODUCT
ID: APP_SAPP_ALPHA
UNIPROT CHAIN:PRO_0000000088 (residues 18-687)
NEUROPROTECTIVE ectodomain released by alpha-secretase (ADAM10/17) cleavage. sAPPalpha promotes neurite outgrowth, synaptogenesis, and neuronal survival. Has 10-100x higher neurotrophic activity than sAPPbeta. The alpha-secretase pathway PRECLUDES Abeta generation - thus sAPPalpha represents the "non-amyloidogenic" pathway. Enhancing alpha-secretase is a therapeutic strategy for Alzheimer's disease.
Isoform-specific terms: negative regulation of neuron apoptotic process neuron projection development
sAPPbeta (Soluble APP-beta) CLEAVAGE PRODUCT
ID: APP_SAPP_BETA
UNIPROT CHAIN:PRO_0000000089 (residues 18-671)
Ectodomain released by beta-secretase (BACE1) cleavage. Unlike sAPPalpha, sAPPbeta has REDUCED neurotrophic activity and may promote apoptosis by binding to DR6 (death receptor 6). This is the first step of the AMYLOIDOGENIC pathway that leads to Abeta generation.
Amyloid-beta 42 (Abeta42) CLEAVAGE PRODUCT
ID: APP_ABETA42
UNIPROT CHAIN:PRO_0000000092 (residues 672-713)
NEUROTOXIC peptide - the pathogenic form in Alzheimer's disease. Abeta42 is more aggregation-prone than Abeta40 due to two additional hydrophobic C-terminal residues. Forms oligomers and fibrils that cause synaptic dysfunction, oxidative stress, and neuron death. The Abeta42/Abeta40 ratio is critical - increased ratio (even with normal total Abeta) causes familial AD. ANTAGONISTIC to sAPPalpha function - same gene produces both neuroprotective AND neurotoxic products depending on processing pathway.
Isoform-specific terms: positive regulation of neuron apoptotic process amyloid fibril formation
Amyloid-beta 40 (Abeta40) CLEAVAGE PRODUCT
ID: APP_ABETA40
UNIPROT CHAIN:PRO_0000000091 (residues 672-711)
Major Abeta species (90% of Abeta). Less aggregation-prone than Abeta42. May actually be protective by competing with Abeta42 for aggregation sites. The Abeta42/Abeta40 ratio is more predictive of AD than total Abeta levels.
Isoform-specific terms: amyloid fibril formation
AICD (APP Intracellular Domain) CLEAVAGE PRODUCT
ID: APP_AICD
UNIPROT CHAIN:PRO_0000000093, PRO_0000000094, PRO_0000000095 (residues 712-770 / 714-770 / 721-770)
Intracellular fragment released by gamma-secretase cleavage. AICD translocates to nucleus with Fe65 and Tip60, where it may act as a transcriptional regulator. Proposed targets include EGFR, p53, KAI1/CD82, GSK3B, and neprilysin. However, the transcription factor function of AICD remains CONTROVERSIAL - some studies suggest nuclear AICD is an artifact of overexpression. AICD is rapidly degraded by IDE (insulin-degrading enzyme).
N-APP (N-terminal fragment) CLEAVAGE PRODUCT
ID: APP_N_APP
UNIPROT CHAIN:PRO_0000381966 (residues 18-286)
N-terminal fragment that binds DR6 (death receptor 6, TNFRSF21) to trigger axon degeneration via caspase-6. Important for developmental axon pruning. May contribute to neurodegeneration in disease. Contains the growth factor and copper-binding domains.

Existing Annotations Review

GO Term Evidence Action Reason
GO:0007409 axonogenesis
IBA
GO_REF:0000033
ACCEPT
Summary: IBA annotation. Full-length APP regulates axon development. APP knockout mice show defects in axonogenesis. sAPPalpha promotes neurite outgrowth while full-length APP with Fe65/Mena inhibits branching to ensure directional growth.
Reason: Core biological process. Well-supported by knockout studies and mechanistic understanding.
GO:0007417 central nervous system development
IBA
GO_REF:0000033
ACCEPT
Summary: Phylogenetic inference (IBA) from GO_REF:0000033. IBA annotations undergo extensive phylogenetic review and are generally reliable.
Reason: IBA annotation supported by phylogenetic analysis.
GO:0005769 early endosome
IBA
GO_REF:0000033
ACCEPT
Summary: Cellular component annotation supported by APP trafficking and localization studies. APP is found in multiple cellular compartments consistent with its complex processing pathway (UniProt P05067).
Reason: Well-documented localization consistent with APP biology.
GO:0005102 signaling receptor binding
IBA
GO_REF:0000033
ACCEPT
Summary: Phylogenetic inference (IBA) from GO_REF:0000033. IBA annotations undergo extensive phylogenetic review and are generally reliable.
Reason: IBA annotation supported by phylogenetic analysis.
GO:0005886 plasma membrane
IBA
GO_REF:0000033
ACCEPT
Summary: Cellular component annotation supported by APP trafficking and localization studies. APP is found in multiple cellular compartments consistent with its complex processing pathway (UniProt P05067).
Reason: Well-documented localization consistent with APP biology.
GO:0030546 signaling receptor activator activity
IBA
GO_REF:0000033
ACCEPT
Summary: Abeta42 activates FPR2 (formyl peptide receptor 2), inducing chemotaxis and oxidant stress in phagocytes (PMID:11316806). Note: this is primarily an Abeta cleavage product function.
Reason: Supported by literature, though applies to Abeta rather than full-length APP.
GO:0005794 Golgi apparatus
IBA
GO_REF:0000033
ACCEPT
Summary: Cellular component annotation supported by APP trafficking and localization studies. APP is found in multiple cellular compartments consistent with its complex processing pathway (UniProt P05067).
Reason: Well-documented localization consistent with APP biology.
GO:0045121 membrane raft
IBA
GO_REF:0000033
ACCEPT
Summary: Cellular component annotation supported by APP trafficking and localization studies. APP is found in multiple cellular compartments consistent with its complex processing pathway (UniProt P05067).
Reason: Well-documented localization consistent with APP biology.
GO:0009986 cell surface
IBA
GO_REF:0000033
ACCEPT
Summary: Cellular component annotation supported by APP trafficking and localization studies. APP is found in multiple cellular compartments consistent with its complex processing pathway (UniProt P05067).
Reason: Well-documented localization consistent with APP biology.
GO:0004867 serine-type endopeptidase inhibitor activity
IEA
GO_REF:0000120
ACCEPT
Summary: ISOFORM-SPECIFIC: KPI-containing isoforms (APP751/770) only. The Kunitz protease inhibitor domain is absent from the neuronal APP695 isoform.
Reason: IEA annotation consistent with known APP biology. Note isoform specificity.
GO:0005576 extracellular region
IEA
GO_REF:0000044
ACCEPT
Summary: IEA annotation. Secreted sAPPalpha/beta and Abeta are found in extracellular region.
Reason: IEA annotation consistent with known APP functions.
GO:0005634 nucleus
IEA
GO_REF:0000044
ACCEPT
Summary: AICD translocates to nucleus with Fe65 and Tip60 for transcriptional regulation. However, this remains controversial.
Reason: IEA annotation consistent with known APP functions.
GO:0005737 cytoplasm
IEA
GO_REF:0000120
ACCEPT
Summary: IEA annotation. APP cytoplasmic domain interacts with multiple adaptor proteins.
Reason: IEA annotation consistent with known APP functions.
GO:0005769 early endosome
IEA
GO_REF:0000044
ACCEPT
Summary: IEA annotation. APP is processed in endosomes where BACE1 cleavage occurs.
Reason: IEA annotation consistent with known APP trafficking.
GO:0005783 endoplasmic reticulum
IEA
GO_REF:0000044
ACCEPT
Summary: IEA annotation. APP is synthesized and processed through ER.
Reason: IEA annotation consistent with known APP trafficking.
GO:0005794 Golgi apparatus
IEA
GO_REF:0000044
ACCEPT
Summary: IEA annotation. APP transits through Golgi during maturation.
Reason: IEA annotation consistent with known APP trafficking.
GO:0005886 plasma membrane
IEA
GO_REF:0000044
ACCEPT
Summary: IEA annotation. Full-length APP is a type I transmembrane protein at plasma membrane.
Reason: IEA annotation consistent with known APP functions.
GO:0005905 clathrin-coated pit
IEA
GO_REF:0000120
ACCEPT
Summary: IEA annotation. APP is internalized via clathrin-mediated endocytosis.
Reason: IEA annotation consistent with known APP trafficking.
GO:0006897 endocytosis
IEA
GO_REF:0000043
ACCEPT
Summary: IEA annotation. APP undergoes internalization via endocytosis.
Reason: IEA annotation consistent with known APP functions.
GO:0006915 apoptotic process
IEA
GO_REF:0000043
ACCEPT
Summary: CLEAVAGE PRODUCT DEPENDENT: Abeta induces apoptosis (neurotoxic), while sAPPalpha is neuroprotective. Full-length APP itself has dual roles depending on processing pathway.
Reason: IEA annotation consistent with APP biology but note cleavage product specificity.
GO:0007155 cell adhesion
IEA
GO_REF:0000043
ACCEPT
Summary: IEA annotation. Full-length APP functions as a cell adhesion molecule via trans-dimerization.
Reason: Core function of full-length APP.
GO:0007219 Notch signaling pathway
IEA
GO_REF:0000043
REMOVE
Summary: APP is not a component of the Notch signaling pathway. This IEA annotation likely arises because APP and Notch are both substrates of gamma-secretase (presenilin), but sharing an enzyme does not make APP part of the Notch pathway. APP has its own distinct signaling pathway via AICD.
Reason: APP is a substrate of gamma-secretase but is NOT a participant in Notch signaling. The connection is only that they share the same protease. This is an incorrect annotation that should be removed.
GO:0008201 heparin binding
IEA
GO_REF:0000120
ACCEPT
Summary: IEA annotation. APP ectodomain binds heparin and heparan sulfate proteoglycans.
Reason: IEA annotation consistent with known APP functions.
GO:0009986 cell surface
IEA
GO_REF:0000120
ACCEPT
Summary: IEA annotation. Full-length APP is a type I transmembrane protein at cell surface.
Reason: IEA annotation consistent with known APP localization.
GO:0010604 positive regulation of macromolecule metabolic process
IEA
GO_REF:0000117
MARK AS OVER ANNOTATED
Summary: IEA annotation for positive regulation of macromolecule metabolic process. This is extremely broad and does not provide useful functional information about APP.
Reason: Too broad to be informative. Over-annotation.
GO:0016020 membrane
IEA
GO_REF:0000120
ACCEPT
Summary: IEA annotation. Full-length APP is a type I transmembrane protein.
Reason: IEA annotation consistent with known APP localization.
GO:0030414 peptidase inhibitor activity
IEA
GO_REF:0000043
ACCEPT
Summary: ISOFORM-SPECIFIC: KPI-containing isoforms (APP751/770) only. The Kunitz protease inhibitor domain is absent from neuronal APP695.
Reason: IEA annotation consistent with known APP biology. Note isoform specificity.
GO:0030426 growth cone
IEA
GO_REF:0000120
ACCEPT
Summary: IEA annotation. APP is localized to growth cones and regulates axon guidance.
Reason: IEA annotation consistent with known APP localization and function.
GO:0031091 platelet alpha granule
IEA
GO_REF:0000117
ACCEPT
Summary: IEA annotation. APP is expressed in platelets and stored in alpha granules.
Reason: IEA annotation consistent with known APP expression.
GO:0031410 cytoplasmic vesicle
IEA
GO_REF:0000120
ACCEPT
Summary: IEA annotation. APP is transported in vesicles along axons.
Reason: IEA annotation consistent with known APP trafficking.
GO:0043005 neuron projection
IEA
GO_REF:0000117
ACCEPT
Summary: IEA annotation. APP is transported to and localized in neuron projections.
Reason: IEA annotation consistent with known APP localization.
GO:0043204 perikaryon
IEA
GO_REF:0000044
ACCEPT
Summary: IEA annotation. APP is found in neuronal cell bodies.
Reason: IEA annotation consistent with known APP localization.
GO:0046872 metal ion binding
IEA
GO_REF:0000043
ACCEPT
Summary: IEA annotation. APP binds copper and zinc via its ectodomain and regulates metal homeostasis.
Reason: Core function of APP. Well documented.
GO:0046914 transition metal ion binding
IEA
GO_REF:0000002
ACCEPT
Summary: IEA annotation. APP binds copper and zinc (transition metals) via its ectodomain.
Reason: Core function of APP. Well documented.
GO:0051246 regulation of protein metabolic process
IEA
GO_REF:0000117
MARK AS OVER ANNOTATED
Summary: IEA annotation for regulation of protein metabolic process. This is very broad and does not provide useful functional information about APP.
Reason: Too broad to be informative. Over-annotation.
GO:0140677 molecular function activator activity
IEA
GO_REF:0000117
MARK AS OVER ANNOTATED
Summary: IEA annotation for molecular function activator activity. This is extremely broad and does not specify what molecular function APP activates. Not informative.
Reason: Too broad to be informative. Over-annotation.
GO:0005515 protein binding
IPI
PMID:10677483
Human aspartic protease memapsin 2 cleaves the beta-secretas...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. BACE1 (memapsin 2) cleaves APP at the beta-secretase site. Functional interaction for APP processing.
Reason: Generic protein binding uninformative - the specific interaction is with BACE1.
Supporting Evidence:
PMID:10677483
Human aspartic protease memapsin 2 cleaves the beta-secretase site of beta-amyloid precursor protein.
GO:0005515 protein binding
IPI
PMID:10681545
beta-Amyloid(1-42) binds to alpha7 nicotinic acetylcholine r...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:10681545
beta-Amyloid(1-42) binds to alpha7 nicotinic acetylcholine receptor with high affinity.
GO:0005515 protein binding
IPI
PMID:11278849
beta -Amyloid peptide-induced apoptosis regulated by a novel...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:11278849
2001 Feb 20. beta -Amyloid peptide-induced apoptosis regulated by a novel protein containing a g protein activation module.
GO:0005515 protein binding
IPI
PMID:11297421
Apolipoprotein A-I directly interacts with amyloid precursor...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:11297421
Apolipoprotein A-I directly interacts with amyloid precursor protein and inhibits A beta aggregation and toxicity.
GO:0005515 protein binding
IPI
PMID:11724784
Jun NH2-terminal kinase (JNK) interacting protein 1 (JIP1) b...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:11724784
Nov 27. Jun NH2-terminal kinase (JNK) interacting protein 1 (JIP1) binds the cytoplasmic domain of the Alzheimer's beta-amyloid precursor protein (APP).
GO:0005515 protein binding
IPI
PMID:11877420
Tyrosine phosphorylation of the beta-amyloid precursor prote...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:11877420
2002 Mar 4. Tyrosine phosphorylation of the beta-amyloid precursor protein cytoplasmic tail promotes interaction with Shc.
GO:0005515 protein binding
IPI
PMID:12485888
Signal transduction through tyrosine-phosphorylated carboxy-...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:12485888
Signal transduction through tyrosine-phosphorylated carboxy-terminal fragments of APP via an enhanced interaction with Shc/Grb2 adaptor proteins in reactive astrocytes of Alzheimer's disease brain.
GO:0005515 protein binding
IPI
PMID:12901838
Presenilin-1 interacts directly with the beta-site amyloid p...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:12901838
Presenilin-1 interacts directly with the beta-site amyloid protein precursor cleaving enzyme (BACE1).
GO:0005515 protein binding
IPI
PMID:15896298
In cerebrospinal fluid ER chaperones ERp57 and calreticulin ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:15896298
In cerebrospinal fluid ER chaperones ERp57 and calreticulin bind beta-amyloid.
GO:0005515 protein binding
IPI
PMID:16027166
BRI2 interacts with amyloid precursor protein (APP) and regu...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16027166
2005 Jul 18. BRI2 interacts with amyloid precursor protein (APP) and regulates amyloid beta (Abeta) production.
GO:0005515 protein binding
IPI
PMID:16049941
A pilot proteomic study of amyloid precursor interactors in ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16049941
A pilot proteomic study of amyloid precursor interactors in Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:16174740
Neuronal sorting protein-related receptor sorLA/LR11 regulat...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16174740
Neuronal sorting protein-related receptor sorLA/LR11 regulates processing of the amyloid precursor protein.
GO:0005515 protein binding
IPI
PMID:16286452
Gerstmann-StrΓ€ussler-Scheinker disease amyloid protein polym...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16286452
Nov 10. Gerstmann-StrΓ€ussler-Scheinker disease amyloid protein polymerizes according to the "dock-and-lock" model.
GO:0005515 protein binding
IPI
PMID:16374483
Neurofibromatosis type 1 protein and amyloid precursor prote...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16374483
Neurofibromatosis type 1 protein and amyloid precursor protein interact in normal human melanocytes and colocalize with melanosomes.
GO:0005515 protein binding
IPI
PMID:16446437
Abeta and tau form soluble complexes that may promote self a...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16446437
Abeta and tau form soluble complexes that may promote self aggregation of both into the insoluble forms observed in Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:16480949
The intracellular domain of amyloid precursor protein intera...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16480949
The intracellular domain of amyloid precursor protein interacts with flotillin-1, a lipid raft protein.
GO:0005515 protein binding
IPI
PMID:16554819
The prolyl isomerase Pin1 regulates amyloid precursor protei...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16554819
The prolyl isomerase Pin1 regulates amyloid precursor protein processing and amyloid-beta production.
GO:0005515 protein binding
IPI
PMID:17112520
Aluminum inhibits proteolytic degradation of amyloid beta pe...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:17112520
Epub 2006 Nov 9. Aluminum inhibits proteolytic degradation of amyloid beta peptide by cathepsin D: a potential link between aluminum accumulation and neuritic plaque deposition.
GO:0005515 protein binding
IPI
PMID:17709753
Amyolid precursor protein mediates presynaptic localization ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:17709753
Amyolid precursor protein mediates presynaptic localization and activity of the high-affinity choline transporter.
GO:0005515 protein binding
IPI
PMID:20195357
A comprehensive resource of interacting protein regions for ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:20195357
A comprehensive resource of interacting protein regions for refining human transcription factor networks.
GO:0005515 protein binding
IPI
PMID:20811458
Gamma-secretase activating protein is a therapeutic target f...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:20811458
Gamma-secretase activating protein is a therapeutic target for Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:20817278
Iron-export ferroxidase activity of Ξ²-amyloid precursor prot...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:20817278
Iron-export ferroxidase activity of Ξ²-amyloid precursor protein is inhibited by zinc in Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:20828565
An aminopeptidase from Streptomyces sp. KK565 degrades beta ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:20828565
Epub 2010 Sep 7. An aminopeptidase from Streptomyces sp.
GO:0005515 protein binding
IPI
PMID:21163940
Interactome mapping suggests new mechanistic details underly...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:21163940
Interactome mapping suggests new mechanistic details underlying Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:2119582
Transforming growth factor-beta bound to soluble derivatives...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:2119582
Transforming growth factor-beta bound to soluble derivatives of the beta amyloid precursor protein of Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:21293490
Mediator is a transducer of amyloid-precursor-protein-depend...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:21293490
Mediator is a transducer of amyloid-precursor-protein-dependent nuclear signalling.
GO:0005515 protein binding
IPI
PMID:22730553
Open-closed motion of Mint2 regulates APP metabolism.
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:22730553
Open-closed motion of Mint2 regulates APP metabolism.
GO:0005515 protein binding
IPI
PMID:22801501
A mutation in APP protects against Alzheimer's disease and a...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:22801501
A mutation in APP protects against Alzheimer's disease and age-related cognitive decline.
GO:0005515 protein binding
IPI
PMID:23585889
Generation of amyloid-Ξ² is reduced by the interaction of cal...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:23585889
Generation of amyloid-Ξ² is reduced by the interaction of calreticulin with amyloid precursor protein, presenilin and nicastrin.
GO:0005515 protein binding
IPI
PMID:24028865
Impact of the cellular prion protein on amyloid-Ξ² and 3PO-ta...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:24028865
Impact of the cellular prion protein on amyloid-Ξ² and 3PO-tau processing.
GO:0005515 protein binding
IPI
PMID:24284412
Amyloid beta a4 precursor protein-binding family B member 1 ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:24284412
2013 Nov 27. Amyloid beta a4 precursor protein-binding family B member 1 (FE65) interactomics revealed synaptic vesicle glycoprotein 2A (SV2A) and sarcoplasmic/endoplasmic reticulum calcium ATPase 2 (SERCA2) as new binding proteins in the human brain.
GO:0005515 protein binding
IPI
PMID:24867889
sAPP modulates iron efflux from brain microvascular endothel...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:24867889
sAPP modulates iron efflux from brain microvascular endothelial cells by stabilizing the ferrous iron exporter ferroportin.
GO:0005515 protein binding
IPI
PMID:25241761
Using an in situ proximity ligation assay to systematically ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:25241761
Oct 9. Using an in situ proximity ligation assay to systematically profile endogenous protein-protein interactions in a pathway network.
GO:0005515 protein binding
IPI
PMID:25959826
Quantitative interaction proteomics of neurodegenerative dis...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:25959826
2015 May 7. Quantitative interaction proteomics of neurodegenerative disease proteins.
GO:0005515 protein binding
IPI
PMID:26496610
A human interactome in three quantitative dimensions organiz...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:26496610
Oct 22. A human interactome in three quantitative dimensions organized by stoichiometries and abundances.
GO:0005515 protein binding
IPI
PMID:29423001
Hypoxia increases amyloid-Ξ² level in exosomes by enhancing t...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:29423001
Hypoxia increases amyloid-Ξ² level in exosomes by enhancing the interaction between CD147 and Hook1.
GO:0005515 protein binding
IPI
PMID:29578633
Probing the Mint2 Protein-Protein Interaction Network Releva...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:29578633
Probing the Mint2 Protein-Protein Interaction Network Relevant to the Pathophysiology of Alzheimer's Disease.
GO:0005515 protein binding
IPI
PMID:30086173
TMEM30A is a candidate interacting partner for the Ξ²-carboxy...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:30086173
eCollection 2018. TMEM30A is a candidate interacting partner for the Ξ²-carboxyl-terminal fragment of amyloid-Ξ² precursor protein in endosomes.
GO:0005515 protein binding
IPI
PMID:30538620
Visualization of Alzheimer's Disease Related Ξ±-/Ξ²-/Ξ³-Secreta...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:30538620
eCollection 2018. Visualization of Alzheimer's Disease Related Ξ±-/Ξ²-/Ξ³-Secretase Ternary Complex by Bimolecular Fluorescence Complementation Based Fluorescence Resonance Energy Transfer.
GO:0005515 protein binding
IPI
PMID:31413325
HENA, heterogeneous network-based data set for Alzheimer's d...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:31413325
HENA, heterogeneous network-based data set for Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:32814053
Interactome Mapping Provides a Network of Neurodegenerative ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:32814053
Interactome Mapping Provides a Network of Neurodegenerative Disease Proteins and Uncovers Widespread Protein Aggregation in Affected Brains.
GO:0005515 protein binding
IPI
PMID:33961781
Dual proteome-scale networks reveal cell-specific remodeling...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:33961781
2021 May 6. Dual proteome-scale networks reveal cell-specific remodeling of the human interactome.
GO:0005515 protein binding
IPI
PMID:34446781
First identification of ITM2B interactome in the human retin...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:34446781
First identification of ITM2B interactome in the human retina.
GO:0005515 protein binding
IPI
PMID:35063084
Tau interactome maps synaptic and mitochondrial processes as...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:35063084
2022 Jan 20. Tau interactome maps synaptic and mitochondrial processes associated with neurodegeneration.
GO:0005515 protein binding
IPI
PMID:35914814
Chr21 protein-protein interactions: enrichment in proteins i...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:35914814
Chr21 protein-protein interactions: enrichment in proteins involved in intellectual disability, autism, and late-onset Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:35922511
A physical wiring diagram for the human immune system.
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:35922511
Aug 3. A physical wiring diagram for the human immune system.
GO:0005515 protein binding
IPI
PMID:40205054
Multimodal cell maps as a foundation for structural and func...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:40205054
Apr 9. Multimodal cell maps as a foundation for structural and functional genomics.
GO:0005515 protein binding
IPI
PMID:8855266
Association of a novel human FE65-like protein with the cyto...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:8855266
Association of a novel human FE65-like protein with the cytoplasmic domain of the beta-amyloid precursor protein.
GO:0005515 protein binding
IPI
PMID:8887653
The phosphotyrosine interaction domains of X11 and FE65 bind...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:8887653
The phosphotyrosine interaction domains of X11 and FE65 bind to distinct sites on the YENPTY motif of amyloid precursor protein.
GO:0005515 protein binding
IPI
PMID:9223340
Interaction between amyloid precursor protein and presenilin...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:9223340
Interaction between amyloid precursor protein and presenilins in mammalian cells: implications for the pathogenesis of Alzheimer disease.
GO:0005515 protein binding
IPI
PMID:9338779
An intracellular protein that binds amyloid-beta peptide and...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:9338779
An intracellular protein that binds amyloid-beta peptide and mediates neurotoxicity in Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:9461550
Fe65L2: a new member of the Fe65 protein family interacting ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:9461550
Fe65L2: a new member of the Fe65 protein family interacting with the intracellular domain of the Alzheimer's beta-amyloid precursor protein.
GO:0005515 protein binding
IPI
PMID:10673326
Agrin binds to beta-amyloid (Abeta), accelerates abeta fibri...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:10673326
Agrin binds to beta-amyloid (Abeta), accelerates abeta fibril formation, and is localized to Abeta deposits in Alzheimer's disease brain.
GO:0005515 protein binding
IPI
PMID:11756426
Amyloid beta binds trimers as well as monomers of the 75-kDa...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:11756426
Dec 27. Amyloid beta binds trimers as well as monomers of the 75-kDa neurotrophin receptor and activates receptor signaling.
GO:0005515 protein binding
IPI
PMID:15615705
CLAC binds to amyloid beta peptides through the positively c...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:15615705
2004 Dec 21. CLAC binds to amyloid beta peptides through the positively charged amino acid cluster within the collagenous domain 1 and inhibits formation of amyloid fibrils.
GO:0005515 protein binding
IPI
PMID:17051221
Structures of human insulin-degrading enzyme reveal a new su...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:17051221
Structures of human insulin-degrading enzyme reveal a new substrate recognition mechanism.
GO:0005515 protein binding
IPI
PMID:17116874
Blocking the apolipoprotein E/amyloid-beta interaction as a ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:17116874
Blocking the apolipoprotein E/amyloid-beta interaction as a potential therapeutic approach for Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:18806802
Cyclophilin D deficiency attenuates mitochondrial and neuron...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:18806802
Cyclophilin D deficiency attenuates mitochondrial and neuronal perturbation and ameliorates learning and memory in Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:22179788
The extracellular chaperone clusterin sequesters oligomeric ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:22179788
The extracellular chaperone clusterin sequesters oligomeric forms of the amyloid-Ξ²(1-40) peptide.
GO:0005515 protein binding
IPI
PMID:22528093
Search for amyloid-binding proteins by affinity chromatograp...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:22528093
Search for amyloid-binding proteins by affinity chromatography.
GO:0005515 protein binding
IPI
PMID:24931469
Molecular basis of substrate recognition and degradation by ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:24931469
2014 Jun 12. Molecular basis of substrate recognition and degradation by human presequence protease.
GO:0005515 protein binding
IPI
PMID:25643321
Structural basis for amyloidogenic peptide recognition by so...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:25643321
Feb 2. Structural basis for amyloidogenic peptide recognition by sorLA.
GO:0005515 protein binding
IPI
PMID:25897080
Sequential Amyloid-Ξ² Degradation by the Matrix Metalloprotea...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:25897080
2015 Apr 20. Sequential Amyloid-Ξ² Degradation by the Matrix Metalloproteases MMP-2 and MMP-9.
GO:0005515 protein binding
IPI
PMID:26618561
Direct High Affinity Interaction between AΞ²42 and GSK3Ξ± Stim...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:26618561
Epub 2015 Dec 15. Direct High Affinity Interaction between AΞ²42 and GSK3Ξ± Stimulates Hyperphosphorylation of Tau.
GO:0005515 protein binding
IPI
PMID:30158114
TLR5 decoy receptor as a novel anti-amyloid therapeutic for ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:30158114
TLR5 decoy receptor as a novel anti-amyloid therapeutic for Alzheimer's disease.
GO:0042802 identical protein binding
IPI
PMID:16286452
Gerstmann-StrΓ€ussler-Scheinker disease amyloid protein polym...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:16286452
Nov 10. Gerstmann-StrΓ€ussler-Scheinker disease amyloid protein polymerizes according to the "dock-and-lock" model.
GO:0042802 identical protein binding
IPI
PMID:18805418
In vitro perturbation of aggregation processes in beta-amylo...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:18805418
Epub 2008 Sep 19. In vitro perturbation of aggregation processes in beta-amyloid peptides: a spectroscopic study.
GO:0042802 identical protein binding
IPI
PMID:19549187
Quenched hydrogen/deuterium exchange NMR characterization of...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:19549187
2009 Jun 22. Quenched hydrogen/deuterium exchange NMR characterization of amyloid-beta peptide aggregates formed in the presence of Cu2+ or Zn2+.
GO:0042802 identical protein binding
IPI
PMID:19754881
The thioflavin T fluorescence assay for amyloid fibril detec...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:19754881
2009 Sep 15. The thioflavin T fluorescence assay for amyloid fibril detection can be biased by the presence of exogenous compounds.
GO:0042802 identical protein binding
IPI
PMID:20573181
Progressive accumulation of amyloid-beta oligomers in Alzhei...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:20573181
2010 Jun 22. Progressive accumulation of amyloid-beta oligomers in Alzheimer's disease and in amyloid precursor protein transgenic mice is accompanied by selective alterations in synaptic scaffold proteins.
GO:0042802 identical protein binding
IPI
PMID:20818335
Neurotoxicity of Alzheimer's disease AΞ² peptides is induced ...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:20818335
Neurotoxicity of Alzheimer's disease AΞ² peptides is induced by small changes in the AΞ²42 to AΞ²40 ratio.
GO:0042802 identical protein binding
IPI
PMID:21113149
Reversing EphB2 depletion rescues cognitive functions in Alz...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:21113149
Reversing EphB2 depletion rescues cognitive functions in Alzheimer model.
GO:0042802 identical protein binding
IPI
PMID:21205198
Lysophosphatidylcholine modulates fibril formation of amyloi...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:21205198
2011 Jan 17. Lysophosphatidylcholine modulates fibril formation of amyloid beta peptide.
GO:0042802 identical protein binding
IPI
PMID:21320494
Lipid matrix plays a role in Abeta fibril kinetics and morph...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:21320494
2011 Feb 12. Lipid matrix plays a role in Abeta fibril kinetics and morphology.
GO:0042802 identical protein binding
IPI
PMID:21527912
Extracellular phosphorylation of the amyloid Ξ²-peptide promo...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:21527912
Extracellular phosphorylation of the amyloid Ξ²-peptide promotes formation of toxic aggregates during the pathogenesis of Alzheimer's disease.
GO:0042802 identical protein binding
IPI
PMID:22200570
Effect of N-homocysteinylation on physicochemical and cytoto...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:22200570
2011 Dec 23. Effect of N-homocysteinylation on physicochemical and cytotoxic properties of amyloid Ξ²-peptide.
GO:0042802 identical protein binding
IPI
PMID:22584060
Dimeric structure of transmembrane domain of amyloid precurs...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:22584060
Epub 2012 May 11. Dimeric structure of transmembrane domain of amyloid precursor protein in micellar environment.
GO:0042802 identical protein binding
IPI
PMID:23103738
A comparative analysis of the aggregation behavior of amyloi...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:23103738
Epub 2012 Oct 24. A comparative analysis of the aggregation behavior of amyloid-Ξ² peptide variants.
GO:0042802 identical protein binding
IPI
PMID:23353684
Protease-activated alpha-2-macroglobulin can inhibit amyloid...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:23353684
2013 Jan 23. Protease-activated alpha-2-macroglobulin can inhibit amyloid formation via two distinct mechanisms.
GO:0042802 identical protein binding
IPI
PMID:23416305
Interaction between soluble AΞ²-(1-40) monomer and AΞ²-(1-42) ...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:23416305
2013 Feb 15. Interaction between soluble AΞ²-(1-40) monomer and AΞ²-(1-42) fibrils probed by paramagnetic relaxation enhancement.
GO:0042802 identical protein binding
IPI
PMID:23551356
N-terminal domain of PyrococcusΒ furiosus l-asparaginase func...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:23551356
N-terminal domain of Pyrococcus furiosus l-asparaginase functions as a non-specific, stable, molecular chaperone.
GO:0042802 identical protein binding
IPI
PMID:23603391
NMR characterization of the interaction of GroEL with amyloi...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:23603391
2013 Apr 18. NMR characterization of the interaction of GroEL with amyloid Ξ² as a model ligand.
GO:0042802 identical protein binding
IPI
PMID:23907009
Isobavachalcone and bavachinin from Psoraleae Fructus modula...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:23907009
Epub 2013 Jul 29. Isobavachalcone and bavachinin from Psoraleae Fructus modulate AΞ²42 aggregation process through different mechanisms in vitro.
GO:0042802 identical protein binding
IPI
PMID:24065130
Amyloid-Ξ² oligomers induce synaptic damage via Tau-dependent...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:24065130
Amyloid-Ξ² oligomers induce synaptic damage via Tau-dependent microtubule severing by TTLL6 and spastin.
GO:0042802 identical protein binding
IPI
PMID:24720730
The coexistence of an equal amount of Alzheimer's amyloid-Ξ² ...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:24720730
The coexistence of an equal amount of Alzheimer's amyloid-Ξ² 40 and 42 forms structurally stable and toxic oligomers through a distinct pathway.
GO:0042802 identical protein binding
IPI
PMID:28882996
Fibril structure of amyloid-Ξ²(1-42) by cryo-electron microsc...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:28882996
Sep 7. Fibril structure of amyloid-Ξ²(1-42) by cryo-electron microscopy.
GO:0042802 identical protein binding
IPI
PMID:17116874
Blocking the apolipoprotein E/amyloid-beta interaction as a ...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:17116874
Blocking the apolipoprotein E/amyloid-beta interaction as a potential therapeutic approach for Alzheimer's disease.
GO:0042802 identical protein binding
IPI
PMID:18059284
Evidence of fibril-like Ξ²-sheet structures in a neurotoxic a...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:18059284
Evidence of fibril-like Ξ²-sheet structures in a neurotoxic amyloid intermediate of Alzheimer's Ξ²-amyloid.
GO:0042802 identical protein binding
IPI
PMID:18483195
Paired beta-sheet structure of an Abeta(1-40) amyloid fibril...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:18483195
Paired beta-sheet structure of an Abeta(1-40) amyloid fibril revealed by electron microscopy.
GO:0042802 identical protein binding
IPI
PMID:18499799
Two-dimensional infrared spectra of isotopically diluted amy...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:18499799
Two-dimensional infrared spectra of isotopically diluted amyloid fibrils from Abeta40.
GO:0042802 identical protein binding
IPI
PMID:19304802
Synaptic transmission block by presynaptic injection of olig...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:19304802
Synaptic transmission block by presynaptic injection of oligomeric amyloid beta.
GO:0042802 identical protein binding
IPI
PMID:19458258
Alpha-helix targeting reduces amyloid-beta peptide toxicity.
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:19458258
Alpha-helix targeting reduces amyloid-beta peptide toxicity.
GO:0042802 identical protein binding
IPI
PMID:19706468
Structure-neurotoxicity relationships of amyloid beta-protei...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:19706468
Structure-neurotoxicity relationships of amyloid beta-protein oligomers.
GO:0042802 identical protein binding
IPI
PMID:19706519
Measurement of amyloid fibril mass-per-length by tilted-beam...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:19706519
Measurement of amyloid fibril mass-per-length by tilted-beam transmission electron microscopy.
GO:0042802 identical protein binding
IPI
PMID:19841277
Site-specific modification of Alzheimer's peptides by choles...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:19841277
Site-specific modification of Alzheimer's peptides by cholesterol oxidation products enhances aggregation energetics and neurotoxicity.
GO:0042802 identical protein binding
IPI
PMID:20133839
Mechanism of amyloid plaque formation suggests an intracellu...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:20133839
Mechanism of amyloid plaque formation suggests an intracellular basis of Abeta pathogenicity.
GO:0042802 identical protein binding
IPI
PMID:22036569
Arc/Arg3.1 regulates an endosomal pathway essential for acti...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:22036569
Arc/Arg3.1 regulates an endosomal pathway essential for activity-dependent Ξ²-amyloid generation.
GO:0042802 identical protein binding
IPI
PMID:22179788
The extracellular chaperone clusterin sequesters oligomeric ...
ACCEPT
Summary: Abeta self-associates forming dimers and higher oligomers.
Reason: Direct single-molecule fluorescence demonstration of Abeta oligomerization.
Supporting Evidence:
PMID:22179788
AΞ²(1-40) forms a heterogeneous distribution of small oligomers (from dimers to 50-mers)
GO:0042802 identical protein binding
IPI
PMID:25543257
Modeling an in-register, parallel "iowa" aΞ² fibril structure...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:25543257
Dec 24. Modeling an in-register, parallel "iowa" aΞ² fibril structure using solid-state NMR data from labeled samples with rosetta.
GO:0042802 identical protein binding
IPI
PMID:30158114
TLR5 decoy receptor as a novel anti-amyloid therapeutic for ...
ACCEPT
Summary: IPI annotation. APP dimerization (homodimerization) is well-established and functionally relevant for cell adhesion and processing.
Reason: APP homodimerization is a core function. More informative than generic protein binding.
Supporting Evidence:
PMID:30158114
TLR5 decoy receptor as a novel anti-amyloid therapeutic for Alzheimer's disease.
GO:0005615 extracellular space
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0006816 calcium ion transport
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: IEA annotation for calcium ion transport. APP is not a calcium transporter. Abeta peptides can form calcium-permeable pores in membranes and Abeta oligomers disrupt calcium homeostasis, but APP itself does not transport calcium. This is an indirect effect of cleavage products.
Reason: APP is not a calcium transporter. The calcium effects are indirect, mediated by Abeta pore formation and signaling disruption. Over-annotation.
GO:0007611 learning or memory
IEA
GO_REF:0000107
KEEP AS NON CORE
Summary: IEA annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
GO:0010288 response to lead ion
IEA
GO_REF:0000107
KEEP AS NON CORE
Summary: IEA annotation for response to lead ion. Lead exposure has been shown to increase APP expression and Abeta production, but this is a response to an environmental toxin rather than a core function.
Reason: Response to lead ion is an environmental response, not a core function of APP. Keep as non-core.
GO:0016504 peptidase activator activity
IEA
GO_REF:0000107
UNDECIDED
Summary: IEA annotation for peptidase activator activity. It is unclear what specific peptidase APP activates. APP is itself a substrate of multiple peptidases (alpha-, beta-, gamma-secretases) but the mechanism of direct peptidase activation is not well characterized.
Reason: Unclear molecular basis for peptidase activator activity. APP is a protease substrate, not clearly a protease activator. Needs further evidence.
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0036269 swimming behavior
IEA
GO_REF:0000107
KEEP AS NON CORE
Summary: ISS annotation for swimming behavior based on mouse APP knockout/transgenic studies. These behavioral phenotypes reflect pleiotropic downstream effects of APP loss or Abeta overexpression in mice rather than a core molecular function of APP.
Reason: Behavioral phenotype (swimming behavior) observed in mouse models. Not a core function of APP but a downstream consequence. Keep as non-core.
GO:0043523 regulation of neuron apoptotic process
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0044304 main axon
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0045471 response to ethanol
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0051247 positive regulation of protein metabolic process
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: IEA annotation for positive regulation of protein metabolic process. Very broad term that does not provide useful information about APP function.
Reason: Too broad to be informative. Over-annotation.
GO:0070555 response to interleukin-1
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: IEA annotation to a broad cytokine-response term. APP and its cleavage products can participate in inflammatory contexts, but this label is not specific enough for APP core-function curation.
Reason: Response to interleukin-1 is too broad and downstream to be promoted as an informative APP function; more specific processing, trafficking, synaptic, or fragment-specific mechanisms should be used where supported.
GO:0070851 growth factor receptor binding
IEA
GO_REF:0000107
UNDECIDED
Summary: IEA annotation for growth factor receptor binding. The specific growth factor receptor that APP binds is unclear. sAPPalpha has growth factor-like properties but the receptor is not well defined.
Reason: Unclear which growth factor receptor APP binds. Needs further evidence.
GO:0071280 cellular response to copper ion
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0071287 cellular response to manganese ion
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0071320 cellular response to cAMP
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0071874 cellular response to norepinephrine stimulus
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0097449 astrocyte projection
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0098992 neuronal dense core vesicle
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0110088 hippocampal neuron apoptotic process
IEA
GO_REF:0000107
KEEP AS NON CORE
Summary: IEA annotation for hippocampal neuron apoptotic process. This is an overly specific term for Abeta-mediated neurotoxicity. The neurotoxic effect of Abeta is well established but this is a pathological consequence, not a core function of APP.
Reason: Pathological consequence of Abeta accumulation, not a core function. Overly specific cell-type qualification. Keep as non-core.
GO:1990090 cellular response to nerve growth factor stimulus
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:1990418 response to insulin-like growth factor stimulus
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:1990761 growth cone lamellipodium
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:1990812 growth cone filopodium
IEA
GO_REF:0000107
ACCEPT
Summary: IEA annotation based on electronic inference. Consistent with APP biology.
Reason: IEA annotation consistent with known APP functions.
GO:0005794 Golgi apparatus
IDA
GO_REF:0000052
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
GO:0005615 extracellular space
NAS
P05067-PRO_0000000093
PMID:18568035
Amyloid-beta protein dimers isolated directly from Alzheimer...
ACCEPT
Summary: NAS annotation for Abeta localization in extracellular space. Shankar et al. (2008) extracted soluble Abeta oligomers from AD brain cortex, demonstrating extracellular presence.
Reason: Annotation correctly targets Abeta cleavage product (PRO_0000000093) and extracellular localization is supported by extraction from brain tissue.
Supporting Evidence:
PMID:18568035
We extracted soluble amyloid-beta protein (Abeta) oligomers directly from the cerebral cortex of subjects with Alzheimer's disease.
GO:0005886 plasma membrane
NAS
P05067-PRO_0000000093
PMID:18568035
Amyloid-beta protein dimers isolated directly from Alzheimer...
ACCEPT
Summary: NAS annotation for Abeta at plasma membrane. Abeta oligomers act at synaptic sites, consistent with membrane association.
Reason: Annotation correctly targets Abeta cleavage product. Membrane association implied by synaptic site of action, consistent with other evidence for plasma membrane localization.
Supporting Evidence:
PMID:18568035
The oligomers potently inhibited long-term potentiation (LTP), enhanced long-term depression (LTD) and reduced dendritic spine density in normal rodent hippocampus.
GO:0043408 regulation of MAPK cascade
ISS
GO_REF:0000114
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0045666 positive regulation of neuron differentiation
ISS
GO_REF:0000114
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:1900272 negative regulation of long-term synaptic potentiation
IDA
P05067-PRO_0000000093
PMID:18568035
Amyloid-beta protein dimers isolated directly from Alzheimer...
KEEP AS NON CORE
Summary: IDA annotation for Abeta-mediated LTP inhibition. Shankar et al. (2008) demonstrated that Abeta oligomers extracted directly from AD brains potently inhibited LTP in rodent hippocampus. Crucially, this effect was specifically attributable to Abeta DIMERS, not monomers or higher-order aggregates.
Reason: Well-supported IDA annotation correctly targeting Abeta cleavage product. This is a real cleavage-product synaptic effect, but it is not a core evolved full-length APP function and should be kept as non-core in this gene-level review.
Supporting Evidence:
PMID:18568035
The oligomers potently inhibited long-term potentiation (LTP), enhanced long-term depression (LTD) and reduced dendritic spine density in normal rodent hippocampus
GO:1900272 negative regulation of long-term synaptic potentiation
NAS
PMID:19242475
Cellular prion protein mediates impairment of synaptic plast...
KEEP AS NON CORE
Summary: NAS annotation based on author statement.
Reason: NAS annotation is supported by literature, but negative regulation of long-term synaptic potentiation is a cleavage-product/pathophysiological synaptic effect rather than a core evolved APP function.
Supporting Evidence:
PMID:19242475
Cellular prion protein mediates impairment of synaptic plasticity by amyloid-beta oligomers.
GO:1900454 positive regulation of long-term synaptic depression
IDA
P05067-PRO_0000000093
PMID:18568035
Amyloid-beta protein dimers isolated directly from Alzheimer...
ACCEPT
Summary: IDA annotation for Abeta-mediated LTD enhancement. Shankar et al. (2008) showed that Abeta dimers from AD brains enhanced LTD in rodent hippocampus. The mechanism requires metabotropic glutamate receptors (mGluRs).
Reason: Well-supported IDA annotation correctly targeting Abeta cleavage product. LTD enhancement is a core synaptotoxic function of Abeta dimers.
Supporting Evidence:
PMID:18568035
The oligomers potently inhibited long-term potentiation (LTP), enhanced long-term depression (LTD) and reduced dendritic spine density in normal rodent hippocampus
GO:1900454 positive regulation of long-term synaptic depression
NAS
PMID:19242475
Cellular prion protein mediates impairment of synaptic plast...
ACCEPT
Summary: NAS annotation based on author statement.
Reason: NAS annotation supported by literature.
Supporting Evidence:
PMID:19242475
Cellular prion protein mediates impairment of synaptic plasticity by amyloid-beta oligomers.
GO:1902951 negative regulation of dendritic spine maintenance
IDA
P05067-PRO_0000000093
PMID:18568035
Amyloid-beta protein dimers isolated directly from Alzheimer...
ACCEPT
Summary: IDA annotation for Abeta-mediated spine loss. Shankar et al. (2008) showed that Abeta oligomers from AD brains reduced dendritic spine density. Effects specifically attributable to Abeta dimers and require NMDA receptors.
Reason: Well-supported IDA annotation correctly targeting Abeta cleavage product. Spine loss is a core synaptotoxic function of Abeta dimers.
Supporting Evidence:
PMID:18568035
The oligomers potently inhibited long-term potentiation (LTP), enhanced long-term depression (LTD) and reduced dendritic spine density in normal rodent hippocampus
GO:1902951 negative regulation of dendritic spine maintenance
NAS
PMID:22820466
Alzheimer amyloid-Ξ² oligomer bound to postsynaptic prion pro...
ACCEPT
Summary: NAS annotation based on author statement.
Reason: NAS annotation supported by literature.
Supporting Evidence:
PMID:22820466
Alzheimer amyloid-Ξ² oligomer bound to postsynaptic prion protein activates Fyn to impair neurons.
GO:0043525 positive regulation of neuron apoptotic process
IGI
PMID:23164821
Clusterin regulates Ξ²-amyloid toxicity via Dickkopf-1-driven...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of neuron apoptotic process. Abeta and gamma-CTF fragments promote neuronal apoptosis, but this is a pathological consequence of aberrant APP processing rather than a core physiological function.
Reason: Neurotoxicity is a pathological consequence of Abeta, not a core APP function. Keep as non-core.
Supporting Evidence:
PMID:23164821
silencing of DKK1 blocks AΞ² neurotoxicity
GO:0032224 positive regulation of synaptic transmission, cholinergic
IDA
PMID:33239400
Implications of Oligomeric Amyloid-Beta (oAΞ²(42)) Signaling ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:33239400
oAΞ²42 activates both homomeric Ξ±7- and heteromeric Ξ±7Ξ²2-nAChR subtypes while preferentially enhancing Ξ±7Ξ²2-nAChR open-dwell times
GO:0043083 synaptic cleft
TAS
PMID:33239400
Implications of Oligomeric Amyloid-Beta (oAΞ²(42)) Signaling ...
ACCEPT
Summary: TAS annotation based on author statement in referenced publication.
Reason: TAS annotation supported by literature.
Supporting Evidence:
PMID:33239400
the oligomeric form of amyloid-Ξ² (oAΞ²42), interacting with Ξ±7-containing nicotinic acetylcholine receptor (nAChR) subtypes
GO:0048018 receptor ligand activity
IDA
PMID:33239400
Implications of Oligomeric Amyloid-Beta (oAΞ²(42)) Signaling ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:33239400
these data provide a molecular mechanism supporting a role for Ξ±7Ξ²2-nAChR in mediating the effects of oAΞ²42
GO:0106003 amyloid-beta complex
IDA
PMID:33239400
Implications of Oligomeric Amyloid-Beta (oAΞ²(42)) Signaling ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:33239400
the oligomeric form of amyloid-Ξ² (oAΞ²42)
GO:0031901 early endosome membrane
IDA
PMID:16174740
Neuronal sorting protein-related receptor sorLA/LR11 regulat...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:16174740
Neuronal sorting protein-related receptor sorLA/LR11 regulates processing of the amyloid precursor protein.
GO:0048018 receptor ligand activity
IDA
PMID:16174740
Neuronal sorting protein-related receptor sorLA/LR11 regulat...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:16174740
Neuronal sorting protein-related receptor sorLA/LR11 regulates processing of the amyloid precursor protein.
GO:1904646 cellular response to amyloid-beta
IDA
PMID:29518356
TREM2 Is a Receptor for Ξ²-Amyloid that Mediates Microglial F...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:29518356
TREM2 Is a Receptor for Ξ²-Amyloid that Mediates Microglial Function.
GO:1905606 regulation of presynapse assembly
IMP
PMID:19726636
Presynaptic and postsynaptic interaction of the amyloid prec...
ACCEPT
Summary: IMP annotation based on mutant phenotype analysis.
Reason: IMP annotation supported by mutant phenotype data.
Supporting Evidence:
PMID:19726636
Presynaptic and postsynaptic interaction of the amyloid precursor protein promotes peripheral and central synaptogenesis.
GO:1905606 regulation of presynapse assembly
IDA
PMID:19726636
Presynaptic and postsynaptic interaction of the amyloid prec...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:19726636
Presynaptic and postsynaptic interaction of the amyloid precursor protein promotes peripheral and central synaptogenesis.
GO:0030425 dendrite
IDA
PMID:24012003
Metabotropic glutamate receptor 5 is a coreceptor for Alzhei...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:24012003
Metabotropic glutamate receptor 5 is a coreceptor for Alzheimer aΞ² oligomer bound to cellular prion protein.
GO:0120283 protein serine/threonine kinase binding
IPI
PMID:24305806
Pharmacologic inhibition of ROCK2 suppresses amyloid-Ξ² produ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:24305806
Pharmacologic inhibition of ROCK2 suppresses amyloid-Ξ² production in an Alzheimer's disease mouse model.
GO:0055096 low-density lipoprotein particle mediated signaling
IDA
PMID:26005850
Central role for PICALM in amyloid-Ξ² blood-brain barrier tra...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:26005850
PICALM regulated PICALM/clathrin-dependent internalization of AΞ² bound to the low density lipoprotein receptor related protein-1
GO:0098989 NMDA selective glutamate receptor signaling pathway
TAS
PMID:17360908
Natural oligomers of the Alzheimer amyloid-beta protein indu...
ACCEPT
Summary: TAS annotation based on author statement in referenced publication.
Reason: TAS annotation supported by literature.
Supporting Evidence:
PMID:17360908
Natural oligomers of the Alzheimer amyloid-beta protein induce reversible synapse loss by modulating an NMDA-type glutamate receptor-dependent signaling pathway.
GO:1902993 positive regulation of amyloid precursor protein catabolic process
IGI
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
ACCEPT
Summary: RAGE-mediated Abeta signaling affects APP processing through beta-secretase activity.
Reason: Study shows RAGE inhibitor reduced beta-secretase activity and Abeta production.
Supporting Evidence:
PMID:22406537
In brain, FPS-ZM1 bound exclusively to RAGE, which inhibited Ξ²-secretase activity and AΞ² production and suppressed microglia activation and the neuroinflammatory response
GO:0050850 positive regulation of calcium-mediated signaling
IGI
PMID:22500019
Amyloid Ξ² (AΞ²) peptide directly activates amylin-3 receptor ...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of calcium-mediated signaling. Abeta disrupts calcium homeostasis. Downstream pathological effect.
Reason: Calcium signaling disruption is a downstream effect of Abeta. Keep as non-core.
Supporting Evidence:
PMID:22500019
2012 Apr 12. Amyloid Ξ² (AΞ²) peptide directly activates amylin-3 receptor subtype by triggering multiple intracellular signaling pathways.
GO:0005743 mitochondrial inner membrane
TAS
Reactome:R-HSA-9839072
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005829 cytosol
TAS
Reactome:R-HSA-9839072
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0010628 positive regulation of gene expression
IMP
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IMP annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:15457210
Double Tgs (mutant APP (mAPP)/RAGE) displayed early abnormalities in spatial learning/memory, accompanied by altered activation of markers of synaptic plasticity and exaggerated neuropathologic findings, before such changes were found in mAPP mice
GO:1900272 negative regulation of long-term synaptic potentiation
IGI
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IGI annotation from RAGE interaction study. Arancio et al. (2004) showed mAPP/RAGE double transgenics have early LTP deficits, but RAGE is the receptor mediating Abeta effects. The annotation is technically valid but the mechanism is RAGE-dependent.
Reason: While LTP inhibition occurs in mAPP transgenics, this paper demonstrates it is RAGE-mediated. Keep as non-core because it reflects Abeta/RAGE-dependent synaptic physiology rather than the defining full-length APP function.
Supporting Evidence:
PMID:15457210
RAGE is a cofactor for Abeta-induced neuronal perturbation in a model of Alzheimer's-type pathology
GO:1901224 positive regulation of non-canonical NF-kappaB signal transduction
IGI
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of non-canonical NF-kappaB signal transduction. Abeta-mediated inflammatory signaling. Downstream effect.
Reason: NF-kappaB activation is a downstream inflammatory effect of Abeta. Keep as non-core.
Supporting Evidence:
PMID:15457210
Receptor for Advanced Glycation Endproducts (RAGE), a multiligand receptor in the immunoglobulin superfamily, functions as a signal-transducing cell surface acceptor for amyloid-beta peptide (Abeta)
GO:2000406 positive regulation of T cell migration
IMP
PMID:19660551
Biochemical and immunohistochemical analysis of an Alzheimer...
KEEP AS NON CORE
Summary: IMP annotation for positive regulation of T cell migration. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of T cell migration) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:19660551
2009 Aug 4. Biochemical and immunohistochemical analysis of an Alzheimer's disease mouse model reveals the presence of multiple cerebral Abeta assembly forms throughout life.
GO:0007611 learning or memory
IGI
PMID:20164328
Loss of alpha7 nicotinic receptors enhances beta-amyloid oli...
KEEP AS NON CORE
Summary: IGI annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:20164328
Loss of alpha7 nicotinic receptors enhances beta-amyloid oligomer accumulation, exacerbating early-stage cognitive decline and septohippocampal pathology in a mouse model of Alzheimer's disease.
GO:0010468 regulation of gene expression
IGI
PMID:21857966
WNT5A signaling contributes to AΞ²-induced neuroinflammation ...
KEEP AS NON CORE
Summary: IGI annotation for regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:21857966
WNT5A signaling contributes to AΞ²-induced neuroinflammation and neurotoxicity.
GO:0030111 regulation of Wnt signaling pathway
IC
PMID:21857966
WNT5A signaling contributes to AΞ²-induced neuroinflammation ...
KEEP AS NON CORE
Summary: IC annotation for regulation of Wnt signaling pathway. APP has been reported to interact with Wnt pathway components. Not a core function.
Reason: Wnt signaling regulation is not a core function of APP. Keep as non-core.
Supporting Evidence:
PMID:21857966
WNT5A signaling contributes to AΞ²-induced neuroinflammation and neurotoxicity.
GO:0046330 positive regulation of JNK cascade
IGI
PMID:23921129
FcΞ³RIIb mediates amyloid-Ξ² neurotoxicity and memory impairme...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of JNK cascade. APP cytoplasmic domain interacts with JIP1 and can activate JNK signaling. Downstream signaling effect.
Reason: JNK cascade activation is a downstream signaling effect. Keep as non-core.
Supporting Evidence:
PMID:23921129
Neuronal FcΞ³RIIb activated ER stress and caspase-12
GO:0048169 regulation of long-term neuronal synaptic plasticity
IGI
PMID:23921129
FcΞ³RIIb mediates amyloid-Ξ² neurotoxicity and memory impairme...
KEEP AS NON CORE
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation is supported by genetic interaction data, but negative regulation of long-term synaptic potentiation is a cleavage-product or transgenic model output rather than a core evolved full-length APP function.
Supporting Evidence:
PMID:23921129
Fcgr2b deficiency ameliorated AΞ²-induced inhibition of long-term potentiation
GO:0007611 learning or memory
IGI
PMID:20445063
Memory impairment in transgenic Alzheimer mice requires cell...
KEEP AS NON CORE
Summary: IGI annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:20445063
Memory impairment in transgenic Alzheimer mice requires cellular prion protein.
GO:0007611 learning or memory
IGI
PMID:24012003
Metabotropic glutamate receptor 5 is a coreceptor for Alzhei...
KEEP AS NON CORE
Summary: IGI annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:24012003
Metabotropic glutamate receptor 5 is a coreceptor for Alzheimer aΞ² oligomer bound to cellular prion protein.
GO:0010628 positive regulation of gene expression
IGI
PMID:28008308
The Protective Role of microRNA-200c in Alzheimer's Disease ...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:28008308
eCollection 2016. The Protective Role of microRNA-200c in Alzheimer's Disease Pathologies Is Induced by Beta Amyloid-Triggered Endoplasmic Reticulum Stress.
GO:0010629 negative regulation of gene expression
IGI
PMID:28008308
The Protective Role of microRNA-200c in Alzheimer's Disease ...
KEEP AS NON CORE
Summary: IGI annotation for negative regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: negative regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:28008308
eCollection 2016. The Protective Role of microRNA-200c in Alzheimer's Disease Pathologies Is Induced by Beta Amyloid-Triggered Endoplasmic Reticulum Stress.
GO:0046982 protein heterodimerization activity
IPI
PMID:19660551
Biochemical and immunohistochemical analysis of an Alzheimer...
ACCEPT
Summary: Abeta forms SDS-stable dimers in J20 transgenic mouse brain.
Reason: Direct biochemical demonstration of Abeta dimerization.
Supporting Evidence:
PMID:19660551
Using an immunoprecipitation/Western blotting technique we find an age-dependent increase in Abeta monomer and SDS-stable dimer
GO:0050808 synapse organization
IGI
PMID:24012003
Metabotropic glutamate receptor 5 is a coreceptor for Alzhei...
ACCEPT
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation supported by genetic interaction data. Note potential cleavage product specificity.
Supporting Evidence:
PMID:24012003
Metabotropic glutamate receptor 5 is a coreceptor for Alzheimer aΞ² oligomer bound to cellular prion protein.
GO:0051247 positive regulation of protein metabolic process
IMP
PMID:11404397
Beta-amyloid activates the mitogen-activated protein kinase ...
MARK AS OVER ANNOTATED
Summary: IMP annotation based on mutant phenotype analysis, but the GO term is broad and does not identify the specific APP or amyloid-beta-dependent signaling/protein-metabolism target.
Reason: The evidence may support a downstream effect on protein metabolism, but GO:0051247 is too broad for informative APP curation and should not be promoted as a core function.
Supporting Evidence:
PMID:11404397
Beta-amyloid activates the mitogen-activated protein kinase cascade via hippocampal alpha7 nicotinic acetylcholine receptors: In vitro and in vivo mechanisms related to Alzheimer's disease.
GO:0051262 protein tetramerization
IPI
PMID:19660551
Biochemical and immunohistochemical analysis of an Alzheimer...
ACCEPT
Summary: Abeta forms multiple assembly forms including oligomers in J20 mouse brain.
Reason: Study shows multiple Abeta assembly forms detected biochemically.
Supporting Evidence:
PMID:19660551
These data demonstrate the presence of multiple assembly forms of Abeta throughout the life of J20 mice
GO:0070206 protein trimerization
IPI
PMID:19660551
Biochemical and immunohistochemical analysis of an Alzheimer...
ACCEPT
Summary: Abeta forms multiple oligomeric assembly forms in J20 mouse brain.
Reason: Study demonstrates multiple Abeta assembly forms including oligomers.
Supporting Evidence:
PMID:19660551
These data demonstrate the presence of multiple assembly forms of Abeta throughout the life of J20 mice
GO:0150003 regulation of spontaneous synaptic transmission
IGI
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
ACCEPT
Summary: Abeta-RAGE interaction affects synaptic plasticity markers in transgenic mouse models.
Reason: Study shows RAGE-mediated Abeta effects on synaptic function.
Supporting Evidence:
PMID:15457210
Double Tgs (mutant APP (mAPP)/RAGE) displayed early abnormalities in spatial learning/memory, accompanied by altered activation of markers of synaptic plasticity and exaggerated neuropathologic findings, before such changes were found in mAPP mice
GO:1905908 positive regulation of amyloid fibril formation
IMP
PMID:19660551
Biochemical and immunohistochemical analysis of an Alzheimer...
KEEP AS NON CORE
Summary: IMP annotation for positive regulation of amyloid fibril formation. While amyloid fibril formation is central to AD pathology, it is a pathological process rather than a core physiological function.
Reason: Amyloid fibril formation is pathological rather than a core physiological function. Keep as non-core.
Supporting Evidence:
PMID:19660551
biochemical fractionation and ELISA analysis revealed evidence of TBS and triton-insoluble sedimentable Abeta aggregates at the earliest ages studied
GO:0034361 very-low-density lipoprotein particle
IPI
PMID:9211985
Association of human, rat, and rabbit apolipoprotein E with ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:9211985
when equivalent amounts of apoE3 or E4 were incubated with beta-amyloid (A beta), apoE3 formed 20 times as much SDS-stable complex with the peptide as apoE4
GO:0034362 low-density lipoprotein particle
IPI
PMID:9211985
Association of human, rat, and rabbit apolipoprotein E with ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:9211985
Lipoproteins isolated from the plasma of individuals homozygous for either epsilon2 or epsilon3 were incubated with A beta(1-40)
GO:0034363 intermediate-density lipoprotein particle
IPI
PMID:9211985
Association of human, rat, and rabbit apolipoprotein E with ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:9211985
lipoprotein-associated rabbit apoE (Cys112, Arg158) did bind the peptide
GO:0034364 high-density lipoprotein particle
IPI
PMID:9211985
Association of human, rat, and rabbit apolipoprotein E with ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:9211985
ApoE2:A beta complex formation was comparable to apoE3:A beta in both native and purified preparations of apoE
GO:0042803 protein homodimerization activity
IPI
PMID:15447668
MAPK recruitment by beta-amyloid in organotypic hippocampal ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:15447668
MAPK recruitment by beta-amyloid in organotypic hippocampal slice cultures depends on physical state and exposure time.
GO:0042803 protein homodimerization activity
IPI
PMID:22179788
The extracellular chaperone clusterin sequesters oligomeric ...
ACCEPT
Summary: Abeta forms dimers as part of its oligomerization pathway.
Reason: Single-molecule fluorescence shows Abeta forms dimers to 50-mers.
Supporting Evidence:
PMID:22179788
AΞ²(1-40) forms a heterogeneous distribution of small oligomers (from dimers to 50-mers)
GO:0051260 protein homooligomerization
IPI
PMID:15447668
MAPK recruitment by beta-amyloid in organotypic hippocampal ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:15447668
MAPK recruitment by beta-amyloid in organotypic hippocampal slice cultures depends on physical state and exposure time.
GO:0051260 protein homooligomerization
IPI
PMID:18602473
Aggregation and catabolism of disease-associated intra-Abeta...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:18602473
2008 Jun 17. Aggregation and catabolism of disease-associated intra-Abeta mutations: reduced proteolysis of AbetaA21G by neprilysin.
GO:0051260 protein homooligomerization
IPI
PMID:22179788
The extracellular chaperone clusterin sequesters oligomeric ...
ACCEPT
Summary: Abeta self-associates forming a range of oligomeric species from dimers to 50-mers.
Reason: Direct single-molecule fluorescence characterization of Abeta oligomerization.
Supporting Evidence:
PMID:22179788
AΞ²(1-40) forms a heterogeneous distribution of small oligomers (from dimers to 50-mers)
GO:0010628 positive regulation of gene expression
IGI
PMID:23164821
Clusterin regulates Ξ²-amyloid toxicity via Dickkopf-1-driven...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:23164821
AΞ² induces the neuronal expression of the canonical wnt antagonist, Dickkopf-1 (Dkk1)
GO:1904591 positive regulation of protein import
IDA
PMID:23164821
Clusterin regulates Ξ²-amyloid toxicity via Dickkopf-1-driven...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:23164821
We demonstrate that AΞ² rapidly targets the clusterin protein, causing its intracellular accumulation possibly by blocking its exit from neurons
GO:1990000 amyloid fibril formation
EXP
PMID:26138908
High-resolution NMR characterization of low abundance oligom...
ACCEPT
Summary: EXP annotation based on experimental evidence.
Reason: EXP annotation supported by direct experimental data.
Supporting Evidence:
PMID:26138908
High-resolution NMR characterization of low abundance oligomers of amyloid-Ξ² without purification.
GO:1990000 amyloid fibril formation
EXP
PMID:9737846
Solution structure of methionine-oxidized amyloid beta-pepti...
ACCEPT
Summary: EXP annotation based on experimental evidence.
Reason: EXP annotation supported by direct experimental data.
Supporting Evidence:
PMID:9737846
Solution structure of methionine-oxidized amyloid beta-peptide (1-40).
GO:0007611 learning or memory
IMP
PMID:11880515
The relationship between Abeta and memory in the Tg2576 mous...
KEEP AS NON CORE
Summary: IMP annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:11880515
The relationship between Abeta and memory in the Tg2576 mouse model of Alzheimer's disease.
GO:0007612 learning
IMP
PMID:11140684
A learning deficit related to age and beta-amyloid plaques i...
KEEP AS NON CORE
Summary: IMP annotation for learning. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:11140684
A learning deficit related to age and beta-amyloid plaques in a mouse model of Alzheimer's disease.
GO:0005515 protein binding
IPI
PMID:14527950
Generation of the beta-amyloid peptide and the amyloid precu...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:14527950
2003 Oct 3. Generation of the beta-amyloid peptide and the amyloid precursor protein C-terminal fragment gamma are potentiated by FE65L1.
GO:0005769 early endosome
IDA
PMID:14527950
Generation of the beta-amyloid peptide and the amyloid precu...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:14527950
2003 Oct 3. Generation of the beta-amyloid peptide and the amyloid precursor protein C-terminal fragment gamma are potentiated by FE65L1.
GO:0005783 endoplasmic reticulum
IDA
PMID:14527950
Generation of the beta-amyloid peptide and the amyloid precu...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:14527950
2003 Oct 3. Generation of the beta-amyloid peptide and the amyloid precursor protein C-terminal fragment gamma are potentiated by FE65L1.
GO:0005794 Golgi apparatus
IDA
PMID:14527950
Generation of the beta-amyloid peptide and the amyloid precu...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:14527950
2003 Oct 3. Generation of the beta-amyloid peptide and the amyloid precursor protein C-terminal fragment gamma are potentiated by FE65L1.
GO:0005615 extracellular space
IDA
PMID:29518356
TREM2 Is a Receptor for Ξ²-Amyloid that Mediates Microglial F...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:29518356
TREM2 Is a Receptor for Ξ²-Amyloid that Mediates Microglial Function.
GO:0048018 receptor ligand activity
IDA
PMID:29518356
TREM2 Is a Receptor for Ξ²-Amyloid that Mediates Microglial F...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:29518356
TREM2 Is a Receptor for Ξ²-Amyloid that Mediates Microglial Function.
GO:0014005 microglia development
IGI
PMID:22198949
TLR2 is a primary receptor for Alzheimer's amyloid Ξ² peptide...
KEEP AS NON CORE
Summary: IGI annotation for microglia development. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (microglia development) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:22198949
Microglia activated by extracellularly deposited amyloid Ξ² peptide (AΞ²) act as a two-edged sword in Alzheimer's disease pathogenesis
GO:0032760 positive regulation of tumor necrosis factor production
IGI
PMID:22198949
TLR2 is a primary receptor for Alzheimer's amyloid Ξ² peptide...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of tumor necrosis factor production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of tumor necrosis factor production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:22198949
they damage neurons by releasing neurotoxic proinflammatory mediators (M1 activation)
GO:0005515 protein binding
IPI
PMID:12054541
A secreted form of human ADAM9 has an alpha-secretase activi...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:12054541
A secreted form of human ADAM9 has an alpha-secretase activity for APP.
GO:0005515 protein binding
IPI
PMID:9774383
Evidence that tumor necrosis factor alpha converting enzyme ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:9774383
Evidence that tumor necrosis factor alpha converting enzyme is involved in regulated alpha-secretase cleavage of the Alzheimer amyloid protein precursor.
GO:0019899 enzyme binding
IPI
PMID:17112471
ADAM19 is tightly associated with constitutive Alzheimer's d...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:17112471
ADAM19 is tightly associated with constitutive Alzheimer's disease APP alpha-secretase in A172 cells.
GO:0050729 positive regulation of inflammatory response
IMP
PMID:29961672
miR-15b reduces amyloid-Ξ² accumulation in SH-SY5Y cell line ...
KEEP AS NON CORE
Summary: IMP annotation for positive regulation of inflammatory response. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of inflammatory response) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:29961672
2018 Dec 21. miR-15b reduces amyloid-Ξ² accumulation in SH-SY5Y cell line through targetting NF-ΞΊB signaling and BACE1.
GO:1901224 positive regulation of non-canonical NF-kappaB signal transduction
IMP
PMID:29961672
miR-15b reduces amyloid-Ξ² accumulation in SH-SY5Y cell line ...
KEEP AS NON CORE
Summary: IMP annotation for positive regulation of non-canonical NF-kappaB signal transduction. Abeta-mediated inflammatory signaling. Downstream effect.
Reason: NF-kappaB activation is a downstream inflammatory effect of Abeta. Keep as non-core.
Supporting Evidence:
PMID:29961672
2018 Dec 21. miR-15b reduces amyloid-Ξ² accumulation in SH-SY5Y cell line through targetting NF-ΞΊB signaling and BACE1.
GO:0010468 regulation of gene expression
IMP
PMID:29274751
Reduced expression of Na(+)/Ca(2+) exchangers is associated ...
KEEP AS NON CORE
Summary: IMP annotation for regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:29274751
Reduced expression of Na(+)/Ca(2+) exchangers is associated with cognitive deficits seen in Alzheimer's disease model mice.
GO:0005515 protein binding
IPI
PMID:23973487
Two Ξ²-strands of RAGE participate in the recognition and tra...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:23973487
Two Ξ²-strands of RAGE participate in the recognition and transport of amyloid-Ξ² peptide across the blood brain barrier.
GO:0010468 regulation of gene expression
IGI
PMID:26200696
Dual pathways mediate Ξ²-amyloid stimulated glutathione relea...
KEEP AS NON CORE
Summary: IGI annotation for regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:26200696
Dual pathways mediate Ξ²-amyloid stimulated glutathione release from astrocytes.
GO:0010628 positive regulation of gene expression
IDA
PMID:26006083
The multidrug resistance pump ABCB1 is a substrate for the u...
KEEP AS NON CORE
Summary: IDA annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:26006083
2015 May 26. The multidrug resistance pump ABCB1 is a substrate for the ubiquitin ligase NEDD4-1.
GO:0010629 negative regulation of gene expression
IDA
PMID:26006083
The multidrug resistance pump ABCB1 is a substrate for the u...
KEEP AS NON CORE
Summary: IDA annotation for negative regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: negative regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:26006083
2015 May 26. The multidrug resistance pump ABCB1 is a substrate for the ubiquitin ligase NEDD4-1.
GO:0106003 amyloid-beta complex
TAS
PMID:22500019
Amyloid Ξ² (AΞ²) peptide directly activates amylin-3 receptor ...
ACCEPT
Summary: TAS annotation based on author statement in referenced publication.
Reason: TAS annotation supported by literature.
Supporting Evidence:
PMID:22500019
2012 Apr 12. Amyloid Ξ² (AΞ²) peptide directly activates amylin-3 receptor subtype by triggering multiple intracellular signaling pathways.
GO:0005886 plasma membrane
IDA
PMID:28164773
Apolipoprotein E-mediated Modulation of ADAM10 in Alzheimer'...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:28164773
Apolipoprotein E-mediated Modulation of ADAM10 in Alzheimer's Disease.
GO:0001774 microglial cell activation
IGI
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IGI annotation for microglial cell activation. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (microglial cell activation) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:15457210
RAGE is a cofactor for Abeta-induced neuronal perturbation in a model of Alzheimer's-type pathology
GO:0001774 microglial cell activation
IGI
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
KEEP AS NON CORE
Summary: IGI annotation for microglial cell activation. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (microglial cell activation) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-mediated brain disorder in a mouse model of Alzheimer disease.
GO:0048143 astrocyte activation
IGI
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IGI annotation for astrocyte activation. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (astrocyte activation) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:15457210
RAGE is a cofactor for Abeta-induced neuronal perturbation in a model of Alzheimer's-type pathology
GO:0032729 positive regulation of type II interferon production
IGI
PMID:17255335
Interferon-gamma and tumor necrosis factor-alpha regulate am...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of type II interferon production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of type II interferon production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:17255335
Interferon-gamma and tumor necrosis factor-alpha regulate amyloid-beta plaque deposition and beta-secretase expression in Swedish mutant APP transgenic mice.
GO:0005886 plasma membrane
IDA
PMID:28855300
An Alzheimer-associated TREM2 variant occurs at the ADAM cle...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:28855300
An Alzheimer-associated TREM2 variant occurs at the ADAM cleavage site and affects shedding and phagocytic function.
GO:0010628 positive regulation of gene expression
IGI
PMID:29061364
Inflammatory microglia are glycolytic and iron retentive and...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:29061364
genotype-related increases in glycolysis, accompanied by increased PFKFB3, and an increase in the expression of ferritin
GO:0010629 negative regulation of gene expression
IGI
PMID:29061364
Inflammatory microglia are glycolytic and iron retentive and...
KEEP AS NON CORE
Summary: IGI annotation for negative regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: negative regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:29061364
microglia prepared from wildtype mice and from transgenic mice that overexpress amyloid precursor protein (APP) and presenilin 1 (PS1; APP/PS1)
GO:0032760 positive regulation of tumor necrosis factor production
IGI
PMID:29061364
Inflammatory microglia are glycolytic and iron retentive and...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of tumor necrosis factor production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of tumor necrosis factor production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:29061364
retention of iron in microglia increased TNFΞ± expression
GO:0045821 positive regulation of glycolytic process
IGI
PMID:29061364
Inflammatory microglia are glycolytic and iron retentive and...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of glycolytic process. Abeta-mediated metabolic effects in cells. Not a core function of APP.
Reason: Metabolic effects downstream of Abeta. Not core APP function. Keep as non-core.
Supporting Evidence:
PMID:29061364
increases in tumor necrosis factor-Ξ± (TNFΞ±) and nitric oxide synthase 2 (NOS2) were accompanied by increased glycolysis
GO:0070555 response to interleukin-1
ISS
GO_REF:0000024
MARK AS OVER ANNOTATED
Summary: ISS annotation based on sequence similarity to characterized ortholog, but the GO term is too broad to identify APP-specific biology.
Reason: The inferred biology should be represented with more specific APP processing, trafficking, synaptic, inflammatory, or fragment-specific regulatory terms rather than this broad cytokine-response term.
GO:0005515 protein binding
IPI
PMID:28720718
Phosphorylation of amyloid precursor protein by mutant LRRK2...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:28720718
Phosphorylation of amyloid precursor protein by mutant LRRK2 promotes AICD activity and neurotoxicity in Parkinson's disease.
GO:1900272 negative regulation of long-term synaptic potentiation
IGI
PMID:16636059
Neprilysin-sensitive synapse-associated amyloid-beta peptide...
KEEP AS NON CORE
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation supported by genetic interaction data, but the phenotype reflects neprilysin-sensitive amyloid-beta oligomer effects on plasticity rather than the core evolved function of full-length APP.
Supporting Evidence:
PMID:16636059
2006 Apr 24. Neprilysin-sensitive synapse-associated amyloid-beta peptide oligomers impair neuronal plasticity and cognitive function.
GO:0032722 positive regulation of chemokine production
IGI
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of chemokine production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of chemokine production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:22406537
In brain, FPS-ZM1 bound exclusively to RAGE, which inhibited Ξ²-secretase activity and AΞ² production and suppressed microglia activation and the neuroinflammatory response
GO:0032731 positive regulation of interleukin-1 beta production
IGI
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of interleukin-1 beta production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of interleukin-1 beta production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:22406537
Receptor for advanced glycation end products (RAGE) mediates AΞ²-induced perturbations in cerebral vessels, neurons, and microglia in AD
GO:0032755 positive regulation of interleukin-6 production
IGI
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of interleukin-6 production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of interleukin-6 production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:22406537
Receptor for advanced glycation end products (RAGE) mediates AΞ²-induced perturbations in cerebral vessels, neurons, and microglia in AD
GO:0032760 positive regulation of tumor necrosis factor production
IGI
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of tumor necrosis factor production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of tumor necrosis factor production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:22406537
Receptor for advanced glycation end products (RAGE) mediates AΞ²-induced perturbations in cerebral vessels, neurons, and microglia in AD
GO:0032760 positive regulation of tumor necrosis factor production
IGI
PMID:12808450
RAGE mediates amyloid-beta peptide transport across the bloo...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of tumor necrosis factor production. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (positive regulation of tumor necrosis factor production) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:12808450
RAGE mediates amyloid-beta peptide transport across the blood-brain barrier and accumulation in brain.
GO:1903523 negative regulation of blood circulation
IGI
PMID:12808450
RAGE mediates amyloid-beta peptide transport across the bloo...
KEEP AS NON CORE
Summary: IGI annotation for negative regulation of blood circulation. Vascular effects of Abeta peptides including vasoconstriction and endothelin production. These are pathological consequences of Abeta accumulation rather than core APP functions.
Reason: Vascular annotation (negative regulation of blood circulation) is a downstream Abeta-mediated pathological effect. Keep as non-core.
Supporting Evidence:
PMID:12808450
RAGE mediates amyloid-beta peptide transport across the blood-brain barrier and accumulation in brain.
GO:1904472 positive regulation of endothelin production
IGI
PMID:12808450
RAGE mediates amyloid-beta peptide transport across the bloo...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of endothelin production. Vascular effects of Abeta peptides including vasoconstriction and endothelin production. These are pathological consequences of Abeta accumulation rather than core APP functions.
Reason: Vascular annotation (positive regulation of endothelin production) is a downstream Abeta-mediated pathological effect. Keep as non-core.
Supporting Evidence:
PMID:12808450
RAGE mediates amyloid-beta peptide transport across the blood-brain barrier and accumulation in brain.
GO:0050786 RAGE receptor binding
IPI
P05067-PRO_0000000093
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
ACCEPT
Summary: IPI annotation for Abeta-RAGE binding. Deane et al. (2012) showed a RAGE inhibitor (FPS-ZM1) blocks Abeta binding to the V domain of RAGE, preventing Abeta-induced cellular stress. This is a core molecular interaction of Abeta.
Reason: Well-documented Abeta-RAGE interaction. Annotation correctly applies to Abeta cleavage product. RAGE binding is key to Abeta neurotoxicity mechanism.
Supporting Evidence:
PMID:22406537
we identified a high-affinity RAGE-specific inhibitor (FPS-ZM1) that blocked Abeta binding to the V domain of RAGE
GO:1901224 positive regulation of non-canonical NF-kappaB signal transduction
IDA
PMID:22406537
A multimodal RAGE-specific inhibitor reduces amyloid Ξ²-media...
KEEP AS NON CORE
Summary: IDA annotation for positive regulation of non-canonical NF-kappaB signal transduction. Abeta-mediated inflammatory signaling. Downstream effect.
Reason: NF-kappaB activation is a downstream inflammatory effect of Abeta. Keep as non-core.
Supporting Evidence:
PMID:22406537
Receptor for advanced glycation end products (RAGE) mediates AΞ²-induced perturbations in cerebral vessels, neurons, and microglia in AD
GO:0005798 Golgi-associated vesicle
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0055037 recycling endosome
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0005739 mitochondrion
IDA
PMID:23525105
Transcriptional regulation of insulin-degrading enzyme modul...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:23525105
2013 Mar 22. Transcriptional regulation of insulin-degrading enzyme modulates mitochondrial amyloid Ξ² (AΞ²) peptide catabolism and functionality.
GO:0005769 early endosome
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0050890 cognition
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: ISS annotation for cognition. Downstream behavioral phenotype of APP/Abeta biology. Not a core molecular function.
Reason: Cognition is a high-level phenotype downstream of APP biology. Keep as non-core.
GO:0005829 cytosol
TAS
Reactome:R-HSA-9617595
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0051087 protein-folding chaperone binding
IPI
PMID:23106396
Amyloid-Ξ² oligomers are sequestered by both intracellular an...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:23106396
Amyloid-Ξ² oligomers are sequestered by both intracellular and extracellular chaperones.
GO:0106003 amyloid-beta complex
IPI
PMID:22179788
The extracellular chaperone clusterin sequesters oligomeric ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:22179788
The extracellular chaperone clusterin sequesters oligomeric forms of the amyloid-Ξ²(1-40) peptide.
GO:0031904 endosome lumen
TAS
PMID:24305806
Pharmacologic inhibition of ROCK2 suppresses amyloid-Ξ² produ...
ACCEPT
Summary: TAS annotation based on author statement in referenced publication.
Reason: TAS annotation supported by literature.
Supporting Evidence:
PMID:24305806
Pharmacologic inhibition of ROCK2 suppresses amyloid-Ξ² production in an Alzheimer's disease mouse model.
GO:0010628 positive regulation of gene expression
IGI
PMID:27853422
ROCK1 Is Associated with Alzheimer's Disease-Specific Plaque...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:27853422
eCollection 2016. ROCK1 Is Associated with Alzheimer's Disease-Specific Plaques, as well as Enhances Autophagosome Formation But not Autophagic AΞ² Clearance.
GO:0010628 positive regulation of gene expression
IMP
PMID:27853422
ROCK1 Is Associated with Alzheimer's Disease-Specific Plaque...
KEEP AS NON CORE
Summary: IMP annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:27853422
eCollection 2016. ROCK1 Is Associated with Alzheimer's Disease-Specific Plaques, as well as Enhances Autophagosome Formation But not Autophagic AΞ² Clearance.
GO:0010629 negative regulation of gene expression
IGI
PMID:27853422
ROCK1 Is Associated with Alzheimer's Disease-Specific Plaque...
KEEP AS NON CORE
Summary: IGI annotation for negative regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: negative regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:27853422
eCollection 2016. ROCK1 Is Associated with Alzheimer's Disease-Specific Plaques, as well as Enhances Autophagosome Formation But not Autophagic AΞ² Clearance.
GO:0007611 learning or memory
IMP
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IMP annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:15457210
Double Tgs (mutant APP (mAPP)/RAGE) displayed early abnormalities in spatial learning/memory, accompanied by altered activation of markers of synaptic plasticity and exaggerated neuropathologic findings, before such changes were found in mAPP mice
GO:0007611 learning or memory
IGI
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IGI annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:15457210
Tg mice bearing a dominant-negative RAGE construct targeted to neurons crossed with mAPP animals displayed preservation of spatial learning/memory
GO:0009986 cell surface
NAS
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
ACCEPT
Summary: RAGE functions as a cell surface receptor for Abeta.
Reason: Paper describes RAGE as signal-transducing cell surface acceptor for Abeta.
Supporting Evidence:
PMID:15457210
Receptor for Advanced Glycation Endproducts (RAGE), a multiligand receptor in the immunoglobulin superfamily, functions as a signal-transducing cell surface acceptor for amyloid-beta peptide (Abeta)
GO:0070374 positive regulation of ERK1 and ERK2 cascade
IGI
PMID:15457210
RAGE potentiates Abeta-induced perturbation of neuronal func...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of ERK1 and ERK2 cascade. Abeta activates MAPK/ERK signaling in various cell types. Downstream signaling effect, not core APP function.
Reason: ERK cascade activation is a downstream effect of Abeta. Keep as non-core.
Supporting Evidence:
PMID:15457210
Receptor for Advanced Glycation Endproducts (RAGE), a multiligand receptor in the immunoglobulin superfamily, functions as a signal-transducing cell surface acceptor for amyloid-beta peptide (Abeta)
GO:1990535 neuron projection maintenance
IGI
PMID:20445063
Memory impairment in transgenic Alzheimer mice requires cell...
ACCEPT
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation supported by genetic interaction data. Note potential cleavage product specificity.
Supporting Evidence:
PMID:20445063
Memory impairment in transgenic Alzheimer mice requires cellular prion protein.
GO:0007611 learning or memory
IGI
PMID:24052308
Human LilrB2 is a Ξ²-amyloid receptor and its murine homolog ...
KEEP AS NON CORE
Summary: IGI annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:24052308
Human LilrB2 is a Ξ²-amyloid receptor and its murine homolog PirB regulates synaptic plasticity in an Alzheimer's model.
GO:0005178 integrin binding
IDA
PMID:21126803
Perlecan domain V inhibits Ξ±2 integrin-mediated amyloid-Ξ² ne...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:21126803
Perlecan domain V inhibits Ξ±2 integrin-mediated amyloid-Ξ² neurotoxicity.
GO:0005615 extracellular space
IMP
PMID:23640054
Brain interstitial oligomeric amyloid Ξ² increases with age a...
ACCEPT
Summary: IMP annotation based on mutant phenotype analysis.
Reason: IMP annotation supported by mutant phenotype data.
Supporting Evidence:
PMID:23640054
Brain interstitial oligomeric amyloid Ξ² increases with age and is resistant to clearance from brain in a mouse model of Alzheimer's disease.
GO:0106003 amyloid-beta complex
IMP
PMID:23640054
Brain interstitial oligomeric amyloid Ξ² increases with age a...
ACCEPT
Summary: IMP annotation based on mutant phenotype analysis.
Reason: IMP annotation supported by mutant phenotype data.
Supporting Evidence:
PMID:23640054
Brain interstitial oligomeric amyloid Ξ² increases with age and is resistant to clearance from brain in a mouse model of Alzheimer's disease.
GO:0050750 low-density lipoprotein particle receptor binding
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0030425 dendrite
IDA NOT
PMID:17251419
Abeta oligomer-induced aberrations in synapse composition, s...
ACCEPT
Summary: NOT annotation - Lacor et al. (2007) showed Abeta oligomers (ADDLs) bind to dendritic spines, not dendrite shafts. The annotation indicates where full-length APP or its products are NOT found. This study focused on Abeta oligomer binding specificity to excitatory pyramidal neurons.
Reason: The negated annotation accurately captures the spatial specificity of Abeta/ADDL binding shown in PMID:17251419.
Supporting Evidence:
PMID:17251419
ADDLs bound to neurons with specificity, attaching to presumed excitatory pyramidal neurons but not GABAergic neurons... consistent with observed attachment of ADDLs to dendritic spines.
GO:0032590 dendrite membrane
TAS NOT
PMID:20032460
Inhibition of calcineurin-mediated endocytosis and alpha-ami...
ACCEPT
Summary: NOT annotation - Zhao et al. (2010) showed that Abeta oligomers (ADDLs) bind specifically to dendritic spines expressing surface AMPA receptors (particularly GluR2), not the general dendrite membrane. The specificity is for postsynaptic compartments.
Reason: The negated annotation accurately reflects the spatial selectivity of ADDL binding shown in PMID:20032460.
Supporting Evidence:
PMID:20032460
ADDL binding occurs in dendritic spines that express surface AMPA receptors, particularly the calcium-impermeable type II AMPA receptor subunit (GluR2).
GO:0005576 extracellular region
TAS
Reactome:R-HSA-9010034
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005886 plasma membrane
TAS
Reactome:R-HSA-9010034
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005886 plasma membrane
TAS
Reactome:R-HSA-9010091
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-5692495
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-9010096
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005615 extracellular space
IDA
PMID:23921129
FcΞ³RIIb mediates amyloid-Ξ² neurotoxicity and memory impairme...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:23921129
soluble AΞ² oligomers interact with FcΞ³RIIb in vitro and in AD brains
GO:0045944 positive regulation of transcription by RNA polymerase II
IGI
PMID:23921129
FcΞ³RIIb mediates amyloid-Ξ² neurotoxicity and memory impairme...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of transcription by RNA polymerase II. AICD has been reported to regulate transcription through Fe65/Tip60 complex, but this remains controversial and applies to a cleavage product rather than full-length APP.
Reason: Transcriptional regulation by AICD is controversial and represents a cleavage product function. Keep as non-core.
Supporting Evidence:
PMID:23921129
FcΞ³RIIb is significantly upregulated in the hippocampus of AD brains and neuronal cells exposed to synthetic AΞ²
GO:0007611 learning or memory
IGI
PMID:21113149
Reversing EphB2 depletion rescues cognitive functions in Alz...
KEEP AS NON CORE
Summary: IGI annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:21113149
Reversing EphB2 depletion rescues cognitive functions in Alzheimer model.
GO:0097645 amylin binding
TAS
PMID:22500019
Amyloid Ξ² (AΞ²) peptide directly activates amylin-3 receptor ...
ACCEPT
Summary: TAS annotation based on author statement in referenced publication.
Reason: TAS annotation supported by literature.
Supporting Evidence:
PMID:22500019
2012 Apr 12. Amyloid Ξ² (AΞ²) peptide directly activates amylin-3 receptor subtype by triggering multiple intracellular signaling pathways.
GO:0010628 positive regulation of gene expression
IGI
PMID:22198949
TLR2 is a primary receptor for Alzheimer's amyloid Ξ² peptide...
KEEP AS NON CORE
Summary: IGI annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:22198949
TLR2-mediated AΞ²42-triggered inflammatory activation
GO:0010629 negative regulation of gene expression
IGI
PMID:22198949
TLR2 is a primary receptor for Alzheimer's amyloid Ξ² peptide...
KEEP AS NON CORE
Summary: IGI annotation for negative regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: negative regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:22198949
TLR2 deficiency in microglia shifts M1- to M2-inflammatory activation in vivo
GO:0005769 early endosome
IDA
PMID:26005850
Central role for PICALM in amyloid-Ξ² blood-brain barrier tra...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:26005850
guided AΞ² trafficking to Rab5 and Rab11
GO:0070381 endosome to plasma membrane transport vesicle
IDA
PMID:26005850
Central role for PICALM in amyloid-Ξ² blood-brain barrier tra...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:26005850
leading to AΞ² endothelial transcytosis and clearance
GO:0005615 extracellular space
IDA
PMID:26005850
Central role for PICALM in amyloid-Ξ² blood-brain barrier tra...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:26005850
AΞ² clearance across the murine blood-brain barrier (BBB)
GO:0048143 astrocyte activation
IGI
PMID:20445063
Memory impairment in transgenic Alzheimer mice requires cell...
KEEP AS NON CORE
Summary: IGI annotation for astrocyte activation. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (astrocyte activation) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20445063
Memory impairment in transgenic Alzheimer mice requires cellular prion protein.
GO:0005109 frizzled binding
IPI
PMID:18234671
Amyloid-beta binds to the extracellular cysteine-rich domain...
ACCEPT
Summary: Abeta binds to the Frizzled cysteine-rich domain at or near the Wnt-binding site.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:18234671
Abeta binds to the Fz cysteine-rich domain at or in close proximity to the Wnt-binding site and inhibits the canonical Wnt signaling pathway
GO:0010629 negative regulation of gene expression
IGI
PMID:18234671
Amyloid-beta binds to the extracellular cysteine-rich domain...
KEEP AS NON CORE
Summary: IGI annotation for negative regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: negative regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:18234671
Amyloid-beta binds to the extracellular cysteine-rich domain of Frizzled and inhibits Wnt/beta-catenin signaling
GO:0090090 negative regulation of canonical Wnt signaling pathway
IDA
PMID:18234671
Amyloid-beta binds to the extracellular cysteine-rich domain...
KEEP AS NON CORE
Summary: IDA annotation for negative regulation of canonical Wnt signaling pathway. APP/Abeta interaction with Wnt signaling components. Not core function.
Reason: Wnt signaling regulation is not a core function of APP. Keep as non-core.
Supporting Evidence:
PMID:18234671
Abeta binds to the Fz cysteine-rich domain at or in close proximity to the Wnt-binding site and inhibits the canonical Wnt signaling pathway
GO:1900181 negative regulation of protein localization to nucleus
IGI
PMID:18234671
Amyloid-beta binds to the extracellular cysteine-rich domain...
ACCEPT
Summary: By inhibiting Wnt signaling, Abeta prevents beta-catenin nuclear localization required for Wnt target gene activation.
Reason: IGI annotation reflects Abeta blocking beta-catenin nuclear translocation by inhibiting Wnt signaling.
Supporting Evidence:
PMID:18234671
Amyloid-beta binds to the extracellular cysteine-rich domain of Frizzled and inhibits Wnt/beta-catenin signaling
GO:0002265 astrocyte activation involved in immune response
IGI
PMID:23152628
LRP1 in brain vascular smooth muscle cells mediates local cl...
KEEP AS NON CORE
Summary: IGI annotation for astrocyte activation involved in immune response. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (astrocyte activation involved in immune response) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:23152628
LRP1 in brain vascular smooth muscle cells mediates local clearance of Alzheimer's amyloid-Ξ².
GO:0005764 lysosome
IDA
PMID:23152628
LRP1 in brain vascular smooth muscle cells mediates local cl...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:23152628
LRP1 in brain vascular smooth muscle cells mediates local clearance of Alzheimer's amyloid-Ξ².
GO:0043395 heparan sulfate proteoglycan binding
IMP
PMID:21289173
Heparan sulphate proteoglycan and the low-density lipoprotei...
ACCEPT
Summary: IMP annotation based on mutant phenotype analysis.
Reason: IMP annotation supported by mutant phenotype data.
Supporting Evidence:
PMID:21289173
Heparan sulphate proteoglycan and the low-density lipoprotein receptor-related protein 1 constitute major pathways for neuronal amyloid-beta uptake.
GO:1904399 heparan sulfate binding
TAS
PMID:21289173
Heparan sulphate proteoglycan and the low-density lipoprotei...
ACCEPT
Summary: TAS annotation based on author statement in referenced publication.
Reason: TAS annotation supported by literature.
Supporting Evidence:
PMID:21289173
Heparan sulphate proteoglycan and the low-density lipoprotein receptor-related protein 1 constitute major pathways for neuronal amyloid-beta uptake.
GO:1904646 cellular response to amyloid-beta
IGI
PMID:23152628
LRP1 in brain vascular smooth muscle cells mediates local cl...
ACCEPT
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation supported by genetic interaction data. Note potential cleavage product specificity.
Supporting Evidence:
PMID:23152628
LRP1 in brain vascular smooth muscle cells mediates local clearance of Alzheimer's amyloid-Ξ².
GO:0032991 protein-containing complex
IDA
PMID:9228033
Interaction of apolipoprotein J-amyloid beta-peptide complex...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:9228033
Interaction of apolipoprotein J-amyloid beta-peptide complex with low density lipoprotein receptor-related protein-2/megalin.
GO:0034185 apolipoprotein binding
IPI
PMID:22138302
Preferential interactions between ApoE-containing lipoprotei...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:22138302
Preferential interactions between ApoE-containing lipoproteins and AΞ² revealed by a detection method that combines size exclusion chromatography with non-reducing gel-shift.
GO:0034363 intermediate-density lipoprotein particle
IDA
PMID:22138302
Preferential interactions between ApoE-containing lipoprotei...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:22138302
Preferential interactions between ApoE-containing lipoproteins and AΞ² revealed by a detection method that combines size exclusion chromatography with non-reducing gel-shift.
GO:0034364 high-density lipoprotein particle
IDA
PMID:22138302
Preferential interactions between ApoE-containing lipoprotei...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:22138302
Preferential interactions between ApoE-containing lipoproteins and AΞ² revealed by a detection method that combines size exclusion chromatography with non-reducing gel-shift.
GO:0051087 protein-folding chaperone binding
IPI
PMID:9228033
Interaction of apolipoprotein J-amyloid beta-peptide complex...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:9228033
Interaction of apolipoprotein J-amyloid beta-peptide complex with low density lipoprotein receptor-related protein-2/megalin.
GO:1990777 lipoprotein particle
IDA
PMID:22138302
Preferential interactions between ApoE-containing lipoprotei...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:22138302
Preferential interactions between ApoE-containing lipoproteins and AΞ² revealed by a detection method that combines size exclusion chromatography with non-reducing gel-shift.
GO:0010628 positive regulation of gene expression
IMP
PMID:23164821
Clusterin regulates Ξ²-amyloid toxicity via Dickkopf-1-driven...
KEEP AS NON CORE
Summary: IMP annotation for positive regulation of gene expression. Gene expression changes are downstream effects of APP processing and Abeta signaling. Some may be mediated by AICD transcriptional regulation (controversial). Not core APP function.
Reason: positive regulation of gene expression is a downstream effect. Keep as non-core.
Supporting Evidence:
PMID:23164821
AΞ² induction of DKK1 and all five of the common genes, including EGR1, NAB2 and KLF10, was significantly blocked by the silencing of CLU
GO:0008285 negative regulation of cell population proliferation
IDA
PMID:22944668
Antimicrobial activity of human islet amyloid polypeptides: ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:22944668
Antimicrobial activity of human islet amyloid polypeptides: an insight into amyloid peptides' connection with antimicrobial peptides.
GO:0034185 apolipoprotein binding
IPI
PMID:9211985
Association of human, rat, and rabbit apolipoprotein E with ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:9211985
These binding studies provide one possible explanation for protective effects of both apoE2 and E3 against the development of Alzheimer's disease
GO:0042157 lipoprotein metabolic process
IC
PMID:9211985
Association of human, rat, and rabbit apolipoprotein E with ...
ACCEPT
Summary: IC annotation inferred by curator based on available evidence.
Reason: IC annotation supported by curator judgment.
Supporting Evidence:
PMID:9211985
In humans, apolipoprotein E (apoE) has three major isoforms
GO:0098815 modulation of excitatory postsynaptic potential
IGI
PMID:20974225
Activation of nicotinic Ξ±(7) acetylcholine receptor enhances...
ACCEPT
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation supported by genetic interaction data. Note potential cleavage product specificity.
Supporting Evidence:
PMID:20974225
Epub 2010 Oct 23. Activation of nicotinic Ξ±(7) acetylcholine receptor enhances long term potentation in wild type mice but not in APP(swe)/PS1Ξ”E9 mice.
GO:1900273 positive regulation of long-term synaptic potentiation
IGI
PMID:20974225
Activation of nicotinic Ξ±(7) acetylcholine receptor enhances...
ACCEPT
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation supported by genetic interaction data. Note potential cleavage product specificity.
Supporting Evidence:
PMID:20974225
Epub 2010 Oct 23. Activation of nicotinic Ξ±(7) acetylcholine receptor enhances long term potentation in wild type mice but not in APP(swe)/PS1Ξ”E9 mice.
GO:0097060 synaptic membrane
IDA NOT
PMID:17308309
Abeta oligomers induce neuronal oxidative stress through an ...
ACCEPT
Summary: NOT annotation - De Felice et al. (2007) showed Abeta oligomers (ADDLs) bind specifically at or near NMDA receptors, not the general synaptic membrane. The study showed ADDLs co-immunoprecipitate with NMDA-R subunits and require NMDA-R activation for their effects.
Reason: The negated annotation accurately captures the receptor-specific binding of ADDLs shown in PMID:17308309, distinguishing binding specificity from general synaptic membrane localization.
Supporting Evidence:
PMID:17308309
ADDLs that were bound to detergent-extracted synaptosomal membranes co-immunoprecipitated with NMDA-R subunits... ADDLs bind to or in close proximity to NMDA-Rs, triggering neuronal damage through NMDA-R-dependent calcium flux.
GO:0032991 protein-containing complex
IPI
P05067-PRO_0000000093
PMID:18568035
Amyloid-beta protein dimers isolated directly from Alzheimer...
ACCEPT
Summary: IPI annotation for Abeta complex formation. Shankar et al. (2008) showed that Abeta dimers (Abeta42-Abeta40 complexes) are the minimal synaptotoxic species. The IPI annotation correctly captures that Abeta42 forms complexes with Abeta40.
Reason: Well-supported IPI annotation correctly targeting Abeta cleavage product. Dimerization is essential for synaptotoxicity.
Supporting Evidence:
PMID:18568035
These various effects were specifically attributable to Abeta dimers
GO:0061844 antimicrobial humoral immune response mediated by antimicrobial peptide
IMP
PMID:20209079
The Alzheimer's disease-associated amyloid beta-protein is a...
KEEP AS NON CORE
Summary: IMP annotation for antimicrobial humoral immune response mediated by antimicrobial peptide. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (antimicrobial humoral immune response mediated by antimicrobial peptide) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20209079
Abeta exerts antimicrobial activity against eight common and clinically relevant microorganisms with a potency equivalent to, and in some cases greater than, LL-37
GO:0046982 protein heterodimerization activity
IPI
P05067-PRO_0000000093
PMID:18568035
Amyloid-beta protein dimers isolated directly from Alzheimer...
ACCEPT
Summary: IPI annotation for Abeta heterodimerization. GOA shows Abeta42 (PRO_0000000093) heterodimerizes with Abeta40 (PRO_0000000092). Shankar et al. (2008) demonstrated that Abeta dimers are the smallest synaptotoxic species.
Reason: Well-supported IPI annotation correctly targeting Abeta42. The Abeta42-Abeta40 heterodimer is the pathogenic species.
Supporting Evidence:
PMID:18568035
These various effects were specifically attributable to Abeta dimers
GO:0051247 positive regulation of protein metabolic process
ISS
GO_REF:0000024
MARK AS OVER ANNOTATED
Summary: ISS annotation based on sequence similarity to characterized ortholog, but the term is very broad and does not identify the specific APP-dependent processing, trafficking, or fragment-mediated mechanism.
Reason: GO:0051247 is too broad for informative APP curation and should not be promoted as a core function when more specific APP biology is available.
GO:0005886 plasma membrane
IDA
PMID:20164328
Loss of alpha7 nicotinic receptors enhances beta-amyloid oli...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:20164328
Loss of alpha7 nicotinic receptors enhances beta-amyloid oligomer accumulation, exacerbating early-stage cognitive decline and septohippocampal pathology in a mouse model of Alzheimer's disease.
GO:0005788 endoplasmic reticulum lumen
TAS
Reactome:R-HSA-8952289
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0007611 learning or memory
IGI
PMID:19587288
Deletion of the alpha 7 nicotinic acetylcholine receptor gen...
KEEP AS NON CORE
Summary: IGI annotation for learning or memory. APP and its cleavage products (especially Abeta oligomers) affect learning and memory, but this is a downstream phenotypic consequence of APP processing rather than a core molecular function.
Reason: learning or memory is a downstream consequence of APP/Abeta biology. Important for disease relevance but not a core function. Keep as non-core.
Supporting Evidence:
PMID:19587288
Deletion of the alpha 7 nicotinic acetylcholine receptor gene improves cognitive deficits and synaptic pathology in a mouse model of Alzheimer's disease.
GO:0050808 synapse organization
IGI
PMID:19587288
Deletion of the alpha 7 nicotinic acetylcholine receptor gen...
ACCEPT
Summary: IGI annotation based on genetic interaction evidence. NOTE: Many IGI annotations for APP involve Abeta-specific effects from transgenic mouse studies and may not represent full-length APP function.
Reason: IGI annotation supported by genetic interaction data. Note potential cleavage product specificity.
Supporting Evidence:
PMID:19587288
Deletion of the alpha 7 nicotinic acetylcholine receptor gene improves cognitive deficits and synaptic pathology in a mouse model of Alzheimer's disease.
GO:0005796 Golgi lumen
TAS
Reactome:R-HSA-8871506
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:1990000 amyloid fibril formation
IMP
PMID:25620700
A genome-wide gene-expression analysis and database in trans...
ACCEPT
Summary: IMP annotation based on mutant phenotype analysis.
Reason: IMP annotation supported by mutant phenotype data.
Supporting Evidence:
PMID:25620700
2015 Jan 22. A genome-wide gene-expression analysis and database in transgenic mice during development of amyloid or tau pathology.
GO:0001878 response to yeast
IMP
PMID:20209079
The Alzheimer's disease-associated amyloid beta-protein is a...
KEEP AS NON CORE
Summary: IMP annotation for response to yeast. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (response to yeast) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20209079
anti-Abeta immunoreactive material in AD whole brain homogenates is active against Candida albicans, the pathogen we identified as most sensitive to synthetic Abeta
GO:0019731 antibacterial humoral response
IDA
PMID:20209079
The Alzheimer's disease-associated amyloid beta-protein is a...
KEEP AS NON CORE
Summary: IDA annotation for antibacterial humoral response. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (antibacterial humoral response) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20209079
Abeta exerts antimicrobial activity against eight common and clinically relevant microorganisms with a potency equivalent to, and in some cases greater than, LL-37
GO:0019732 antifungal humoral response
IMP
PMID:20209079
The Alzheimer's disease-associated amyloid beta-protein is a...
KEEP AS NON CORE
Summary: IMP annotation for antifungal humoral response. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (antifungal humoral response) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20209079
anti-Abeta immunoreactive material in AD whole brain homogenates is active against Candida albicans, the pathogen we identified as most sensitive to synthetic Abeta
GO:0045087 innate immune response
IMP
PMID:20209079
The Alzheimer's disease-associated amyloid beta-protein is a...
KEEP AS NON CORE
Summary: IMP annotation for innate immune response. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (innate immune response) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20209079
Our findings suggest Abeta is a hitherto unrecognized AMP that may normally function in the innate immune system
GO:0050829 defense response to Gram-negative bacterium
IDA
PMID:20209079
The Alzheimer's disease-associated amyloid beta-protein is a...
KEEP AS NON CORE
Summary: IDA annotation for defense response to Gram-negative bacterium. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (defense response to Gram-negative bacterium) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20209079
The synthetic Abeta peptides demonstrated antibiotic activity against Gram-negative and Gram-positive bacteria and the yeast C. albicans
GO:0050830 defense response to Gram-positive bacterium
IDA
PMID:20209079
The Alzheimer's disease-associated amyloid beta-protein is a...
KEEP AS NON CORE
Summary: IDA annotation for defense response to Gram-positive bacterium. These immune/inflammatory effects are primarily mediated by Abeta cleavage products activating innate immune cells (microglia, astrocytes) rather than representing core functions of full-length APP.
Reason: Immune/inflammatory annotation (defense response to Gram-positive bacterium) reflects downstream Abeta-mediated effects. Not a core function of APP itself. Keep as non-core.
Supporting Evidence:
PMID:20209079
The synthetic Abeta peptides demonstrated antibiotic activity against Gram-negative and Gram-positive bacteria and the yeast C. albicans
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-6783332
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005515 protein binding
IPI
PMID:11238726
Fibulin-1 binds the amino-terminal head of beta-amyloid prec...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:11238726
Fibulin-1 binds the amino-terminal head of beta-amyloid precursor protein and modulates its physiological function.
GO:0005768 endosome
IDA
PMID:18353773
A novel sorting nexin modulates endocytic trafficking and al...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:18353773
2008 Mar 19. A novel sorting nexin modulates endocytic trafficking and alpha-secretase cleavage of the amyloid precursor protein.
GO:0009986 cell surface
IDA
PMID:18353773
A novel sorting nexin modulates endocytic trafficking and al...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:18353773
2008 Mar 19. A novel sorting nexin modulates endocytic trafficking and alpha-secretase cleavage of the amyloid precursor protein.
GO:0005515 protein binding
IPI
PMID:24336208
Rare coding variants in the phospholipase D3 gene confer ris...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:24336208
Rare coding variants in the phospholipase D3 gene confer risk for Alzheimer's disease.
GO:0005615 extracellular space
HDA
PMID:16502470
Human colostrum: identification of minor proteins in the aqu...
ACCEPT
Summary: HDA annotation from high-throughput direct assay.
Reason: HDA annotation supported by experimental data.
Supporting Evidence:
PMID:16502470
Human colostrum: identification of minor proteins in the aqueous phase by proteomics.
GO:0019899 enzyme binding
IPI
PMID:24499793
FKBP12 regulates the localization and processing of amyloid ...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:24499793
FKBP12 regulates the localization and processing of amyloid precursor protein in human cell lines.
GO:0045121 membrane raft
IDA
PMID:24499793
FKBP12 regulates the localization and processing of amyloid ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:24499793
FKBP12 regulates the localization and processing of amyloid precursor protein in human cell lines.
GO:0005515 protein binding
IPI
PMID:16407538
Interaction of the cytosolic domains of sorLA/LR11 with the ...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:16407538
Interaction of the cytosolic domains of sorLA/LR11 with the amyloid precursor protein (APP) and beta-secretase beta-site APP-cleaving enzyme.
GO:0005641 nuclear envelope lumen
IDA
PMID:21989385
Quantitative modelling of amyloidogenic processing and its i...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:21989385
Quantitative modelling of amyloidogenic processing and its influence by SORLA in Alzheimer's disease.
GO:0043235 receptor complex
IDA
PMID:23382219
Structural basis for endosomal trafficking of diverse transm...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:23382219
Structural basis for endosomal trafficking of diverse transmembrane cargos by PX-FERM proteins.
GO:0070062 extracellular exosome
HDA
PMID:19199708
Proteomic analysis of human parotid gland exosomes by multid...
ACCEPT
Summary: HDA annotation from high-throughput direct assay.
Reason: HDA annotation supported by experimental data.
Supporting Evidence:
PMID:19199708
Proteomic analysis of human parotid gland exosomes by multidimensional protein identification technology (MudPIT).
GO:0005794 Golgi apparatus
IDA
PMID:20427278
The novel membrane protein TMEM59 modulates complex glycosyl...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:20427278
2010 Apr 28. The novel membrane protein TMEM59 modulates complex glycosylation, cell surface expression, and secretion of the amyloid precursor protein.
GO:0005886 plasma membrane
IDA
PMID:20427278
The novel membrane protein TMEM59 modulates complex glycosyl...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:20427278
2010 Apr 28. The novel membrane protein TMEM59 modulates complex glycosylation, cell surface expression, and secretion of the amyloid precursor protein.
GO:0048471 perinuclear region of cytoplasm
IDA
PMID:20427278
The novel membrane protein TMEM59 modulates complex glycosyl...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:20427278
2010 Apr 28. The novel membrane protein TMEM59 modulates complex glycosylation, cell surface expression, and secretion of the amyloid precursor protein.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-481007
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005829 cytosol
TAS
Reactome:R-HSA-1296421
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005829 cytosol
TAS
Reactome:R-HSA-844440
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005829 cytosol
TAS
Reactome:R-HSA-844610
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005829 cytosol
TAS
Reactome:R-HSA-844612
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0031093 platelet alpha granule lumen
TAS
Reactome:R-HSA-481007
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-5229111
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-8871494
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-8871506
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0031904 endosome lumen
TAS
Reactome:R-HSA-9010091
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0032588 trans-Golgi network membrane
TAS
Reactome:R-HSA-5229111
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0032588 trans-Golgi network membrane
TAS
Reactome:R-HSA-5229132
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-2467665
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-6783332
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-879411
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-976734
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-977136
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-NUL-997411
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-379048
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-380073
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-391913
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-749448
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-749452
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-749454
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-749456
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005576 extracellular region
TAS
Reactome:R-HSA-8870710
ACCEPT
Summary: TAS annotation from Reactome pathway database.
Reason: Reactome annotation consistent with known APP biology and pathway involvement.
GO:0005515 protein binding
IPI
PMID:18468999
Regulation of FE65 nuclear translocation and function by amy...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:18468999
2008 May 9. Regulation of FE65 nuclear translocation and function by amyloid beta-protein precursor in osmotically stressed cells.
GO:0005886 plasma membrane
IDA
PMID:12805363
Autosomal recessive hypercholesterolemia protein interacts w...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:12805363
2003 Jun 12. Autosomal recessive hypercholesterolemia protein interacts with and regulates the cell surface level of Alzheimer's amyloid beta precursor protein.
GO:0051425 PTB domain binding
IPI
PMID:12805363
Autosomal recessive hypercholesterolemia protein interacts w...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:12805363
2003 Jun 12. Autosomal recessive hypercholesterolemia protein interacts with and regulates the cell surface level of Alzheimer's amyloid beta precursor protein.
GO:0005515 protein binding
IPI
PMID:18509662
Close association of water channel AQP1 with amyloid-beta de...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:18509662
2008 May 29. Close association of water channel AQP1 with amyloid-beta deposition in Alzheimer disease brains.
GO:0005737 cytoplasm
IDA
PMID:18509662
Close association of water channel AQP1 with amyloid-beta de...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:18509662
2008 May 29. Close association of water channel AQP1 with amyloid-beta deposition in Alzheimer disease brains.
GO:0005102 signaling receptor binding
IPI
PMID:19849849
CD74 interacts with APP and suppresses the production of Abe...
ACCEPT
Summary: IPI annotation showing specific protein interaction.
Reason: IPI annotation with specific molecular function is more informative than generic protein binding.
Supporting Evidence:
PMID:19849849
CD74 interacts with APP and suppresses the production of Abeta.
GO:0005515 protein binding
IPI
PMID:19849849
CD74 interacts with APP and suppresses the production of Abe...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:19849849
CD74 interacts with APP and suppresses the production of Abeta.
GO:0005515 protein binding
IPI
PMID:19901339
RAGE-mediated signaling contributes to intraneuronal transpo...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:19901339
RAGE-mediated signaling contributes to intraneuronal transport of amyloid-beta and neuronal dysfunction.
GO:0043197 dendritic spine
IDA
PMID:11988176
The acid-activated ion channel ASIC contributes to synaptic ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:11988176
The acid-activated ion channel ASIC contributes to synaptic plasticity, learning, and memory.
GO:0043198 dendritic shaft
IDA
PMID:11988176
The acid-activated ion channel ASIC contributes to synaptic ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:11988176
The acid-activated ion channel ASIC contributes to synaptic plasticity, learning, and memory.
GO:0045202 synapse
IDA
PMID:11988176
The acid-activated ion channel ASIC contributes to synaptic ...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:11988176
The acid-activated ion channel ASIC contributes to synaptic plasticity, learning, and memory.
GO:0003677 DNA binding
ISS
GO_REF:0000024
UNDECIDED
Summary: ISS annotation for DNA binding. The AICD fragment has been reported to associate with transcription factor complexes (Fe65/Tip60) and regulate gene expression, but whether AICD itself directly binds DNA remains controversial. Most evidence suggests AICD acts as a transcriptional co-activator through protein-protein interactions rather than direct DNA binding.
Reason: The claim that APP/AICD directly binds DNA is not well-supported. AICD associates with DNA-binding complexes but may not bind DNA directly. This annotation needs further experimental validation.
GO:0005737 cytoplasm
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0005794 Golgi apparatus
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0006417 regulation of translation
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0006878 intracellular copper ion homeostasis
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0006897 endocytosis
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0007409 axonogenesis
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0007617 mating behavior
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: ISS annotation for mating behavior based on mouse APP knockout/transgenic studies. These behavioral phenotypes reflect pleiotropic downstream effects of APP loss or Abeta overexpression in mice rather than a core molecular function of APP.
Reason: Behavioral phenotype (mating behavior) observed in mouse models. Not a core function of APP but a downstream consequence. Keep as non-core.
GO:0007626 locomotory behavior
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: ISS annotation for locomotory behavior based on mouse APP knockout/transgenic studies. These behavioral phenotypes reflect pleiotropic downstream effects of APP loss or Abeta overexpression in mice rather than a core molecular function of APP.
Reason: Behavioral phenotype (locomotory behavior) observed in mouse models. Not a core function of APP but a downstream consequence. Keep as non-core.
GO:0008088 axo-dendritic transport
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0008344 adult locomotory behavior
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: ISS annotation for adult locomotory behavior based on mouse APP knockout/transgenic studies. These behavioral phenotypes reflect pleiotropic downstream effects of APP loss or Abeta overexpression in mice rather than a core molecular function of APP.
Reason: Behavioral phenotype (adult locomotory behavior) observed in mouse models. Not a core function of APP but a downstream consequence. Keep as non-core.
GO:0008542 visual learning
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: ISS annotation for visual learning based on mouse APP knockout/transgenic studies. These behavioral phenotypes reflect pleiotropic downstream effects of APP loss or Abeta overexpression in mice rather than a core molecular function of APP.
Reason: Behavioral phenotype (visual learning) observed in mouse models. Not a core function of APP but a downstream consequence. Keep as non-core.
GO:0016020 membrane
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0016199 axon midline choice point recognition
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0016322 neuron remodeling
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0016358 dendrite development
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0030198 extracellular matrix organization
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0031175 neuron projection development
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0035235 ionotropic glutamate receptor signaling pathway
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0040014 regulation of multicellular organism growth
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0045931 positive regulation of mitotic cell cycle
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: ISS annotation for positive regulation of mitotic cell cycle. Some evidence suggests AICD can regulate cell cycle genes, but this is not a core function of APP in neurons (which are post-mitotic).
Reason: Cell cycle regulation is not a core function of APP, particularly in neurons which are post-mitotic. Keep as non-core.
GO:0048669 collateral sprouting in absence of injury
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0050803 regulation of synapse structure or activity
ISS
GO_REF:0000024
ACCEPT
Summary: ISS annotation based on sequence similarity to characterized ortholog.
Reason: ISS annotation consistent with known APP functions.
GO:0005515 protein binding
IPI
PMID:18026102
Cystatin C modulates cerebral beta-amyloidosis.
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:18026102
Cystatin C modulates cerebral beta-amyloidosis.
GO:0005515 protein binding
IPI
PMID:14557245
APP-BP1 mediates APP-induced apoptosis and DNA synthesis and...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:14557245
APP-BP1 mediates APP-induced apoptosis and DNA synthesis and is increased in Alzheimer's disease brain.
GO:0005515 protein binding
IPI
PMID:8626687
APP-BP1, a novel protein that binds to the carboxyl-terminal...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:8626687
APP-BP1, a novel protein that binds to the carboxyl-terminal region of the amyloid precursor protein.
GO:0004867 serine-type endopeptidase inhibitor activity
IDA
PMID:10652580
Production of amyloid beta protein precursor as a proteinase...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:10652580
Production of amyloid beta protein precursor as a proteinase inhibitor by human astrocytic tumors.
GO:0009986 cell surface
IDA
PMID:7593229
Serine proteinase inhibitors in human skeletal muscle: expre...
ACCEPT
Summary: IDA annotation based on direct experimental assay.
Reason: IDA annotation supported by direct experimental evidence.
Supporting Evidence:
PMID:7593229
Serine proteinase inhibitors in human skeletal muscle: expression of beta-amyloid protein precursor and alpha 1-antichymotrypsin in vivo and during myogenesis in vitro.
GO:0005886 plasma membrane
TAS
PMID:10806211
Phosphorylation of the beta-amyloid precursor protein at the...
ACCEPT
Summary: TAS annotation based on author statement in referenced publication.
Reason: TAS annotation supported by literature.
Supporting Evidence:
PMID:10806211
Phosphorylation of the beta-amyloid precursor protein at the cell surface by ectocasein kinases 1 and 2.
GO:0005515 protein binding
IPI
PMID:10081969
Molecular cloning of human Fe65L2 and its interaction with t...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:10081969
Molecular cloning of human Fe65L2 and its interaction with the Alzheimer's beta-amyloid precursor protein.
GO:0005515 protein binding
IPI
PMID:10049767
X11L2, a new member of the X11 protein family, interacts wit...
MARK AS OVER ANNOTATED
Summary: IPI protein binding annotation. Generic protein binding does not provide specific functional information.
Reason: Generic protein binding uninformative - should use more specific MF terms.
Supporting Evidence:
PMID:10049767
X11L2, a new member of the X11 protein family, interacts with Alzheimer's beta-amyloid precursor protein.
GO:0098631 cell adhesion mediator activity
TAS
file:human/APP/APP-uniprot.txt
NEW
Summary: NEW annotation proposed in this second-pass review. Full-length APP functions at the neuronal cell surface as an adhesion/receptor-like molecule that promotes cell-cell contact and synaptogenesis.
Reason: This molecular function is already used in the APP core-function synthesis but was missing from the existing annotation block. It captures full-length APP biology more directly than generic cell adhesion process terms.
Supporting Evidence:
file:human/APP/APP-uniprot.txt
Functions as a cell surface receptor
file:human/APP/APP-uniprot.txt
neuronal adhesion and axonogenesis
GO:0050839 cell adhesion molecule binding
TAS
file:human/APP/APP-uniprot.txt
NEW
Summary: NEW annotation proposed in this second-pass review. APP molecules and APP-family ectodomains participate in adhesion-associated interactions at the cell surface and synapse.
Reason: This term is present in the APP core-function synthesis but absent from GOA-derived annotations. It represents APP adhesion-associated binding better than generic protein-binding annotations.
Supporting Evidence:
file:human/APP/APP-deep-research-falcon.md
cell adhesion
file:human/APP/APP-uniprot.txt
promotes synaptogenesis
GO:0005507 copper ion binding
TAS
file:human/APP/APP-uniprot.txt
NEW
Summary: NEW annotation proposed in this second-pass review. APP and amyloid-beta fragments bind copper through extracellular metal-binding regions and are linked to copper reduction/homeostasis.
Reason: Existing annotations include broad metal and transition-metal binding, but the APP core-function synthesis uses the more specific copper ion binding term. UniProt supports copper binding/reduction directly, so the specific MF term should be represented.
Supporting Evidence:
file:human/APP/APP-uniprot.txt
Extracellular binding and reduction of copper
file:human/APP/APP-uniprot.txt
Amyloid-beta peptides are lipophilic metal chelators

Core Functions

Full-length APP functions as a cell surface adhesion molecule. APP molecules on neighboring cells engage in trans-dimerization to promote synaptogenesis and cell-cell contact. This is a physiological function of full-length APP at the plasma membrane.

Directly Involved In:
Supporting Evidence:
  • file:human/APP/APP-deep-research-falcon.md

APP regulates axon development through multiple mechanisms. The sAPPalpha ectodomain promotes neurite outgrowth acting as a signaling ligand, while full-length APP interacts with Fe65/Mena to guide axon growth. APP knockout mice show defects in axonogenesis.

Supporting Evidence:
  • file:human/APP/APP-deep-research-falcon.md

APP is highly expressed at synapses and plays physiological roles in synapse formation, maintenance, and plasticity. APP trans-dimerization across the synaptic cleft mediates cell-cell adhesion that contributes to synapse structure. APP knockout models show synaptic deficits.

Supporting Evidence:
  • file:human/APP/APP-deep-research-falcon.md

APP binds copper and zinc ions via its ectodomain (GFLD/copper-binding domain) and participates in copper homeostasis and reduction of Cu(2+) to Cu(+). This is a direct molecular function of the APP ectodomain.

Supporting Evidence:
  • file:human/APP/APP-deep-research-falcon.md

ISOFORM-SPECIFIC: The Kunitz protease inhibitor (KPI) domain in APP751/770 isoforms confers serine protease inhibitor activity (Protease nexin-II function). Absent from the neuronal APP695 isoform.

Supporting Evidence:
  • file:human/APP/APP-deep-research-falcon.md

CLEAVAGE PRODUCT FUNCTION: Abeta peptides (particularly Abeta42) self-assemble into amyloid fibrils via identical protein binding. This is a defining biochemical property of the Abeta cleavage products of APP and is central to Alzheimer disease pathology. Both full-length APP and Abeta cleavage products engage in homodimerization.

Supporting Evidence:
  • file:human/APP/APP-deep-research-falcon.md

APP ectodomain binds heparin and heparan sulfate proteoglycans. This interaction promotes APP dimerization, influences neurite outgrowth, and modulates cell adhesion functions.

Molecular Function:
heparin binding
Directly Involved In:
Supporting Evidence:
  • file:human/APP/APP-deep-research-falcon.md

References

Loading supporting content…

Download this section (compressed HTML)

Suggested Questions for Experts

Q: Which APP isoforms and proteolytic fragments mediate normal in-vivo synaptic adhesion, neurite outgrowth, and axon guidance in adult neurons versus development?

Suggested experts: APP neurobiology expert, synapse development expert, neuronal cell-adhesion expert

Q: What endogenous receptor or partner mechanisms mediate sAPPalpha trophic signaling in vivo, and which functions are separable from full-length APP cell-adhesion activity?

Suggested experts: APP processing expert, neurotrophic signaling expert

Q: How do APP copper and zinc binding or redox activities operate under physiological neuronal and endosomal conditions, and which functions belong to full-length APP versus amyloid-beta fragments?

Suggested experts: neuronal metal homeostasis expert, APP biochemist

Q: Which APP intracellular-domain transcriptional or signaling effects are direct evolved signaling functions rather than secondary consequences of altered trafficking or proteolysis?

Suggested experts: APP intracellular signaling expert, neuronal trafficking expert

Suggested Experiments

Experiment: Compare endogenous APP isoform and fragment rescue in APP-deficient neurons or knock-in mice, separating APP695 from KPI-containing APP751/770 and measuring synapse formation, neurite outgrowth, axon guidance, and plasticity.

Hypothesis: Distinct APP isoforms and cleavage products make separable physiological contributions to adhesion, trophic signaling, and axon/synapse development.

Type: endogenous rescue and isoform-specific knock-in genetics

Experiment: Generate cleavage-resistant and fragment-selective APP alleles at the endogenous locus to separate full-length adhesion, sAPPalpha trophic signaling, amyloid-beta production, and APP intracellular-domain functions in vivo.

Hypothesis: Full-length APP, soluble ectodomain, amyloid-beta, and intracellular fragments each account for different subsets of the observed neuronal phenotypes.

Type: knock-in allele series with in-vivo phenotyping

Experiment: Test APP copper/zinc-binding-site mutants at endogenous expression levels while measuring neuronal metal homeostasis, redox state, endosomal physiology, synaptic function, and APP trafficking.

Hypothesis: APP metal-binding motifs contribute to physiological neuronal metal/redox homeostasis independently of overexpression or aggregate toxicity.

Type: endogenous mutagenesis with biochemical and physiological assays

Deep Research

Falcon

(APP-deep-research-falcon.md)

Loading supporting content…

Download this section (compressed HTML)

πŸ“š Additional Documentation

Notes

(APP-notes.md)

Loading supporting content…

Download this section (compressed HTML)

Bioreason Rl Predictions

(APP-bioreason-rl-predictions.md)

Loading supporting content…

Download this section (compressed HTML)

Bioreason Rl Review

(APP-bioreason-rl-review.md)

Loading supporting content…

Download this section (compressed HTML)

πŸ“„ View Raw YAML

Loading supporting content…

Download this section (compressed HTML)