G6PC3

UniProt ID: Q9BUM1
Organism: Homo sapiens
Review Status: COMPLETE
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Gene Description

G6PC3 encodes the ubiquitously expressed catalytic subunit 3 of glucose-6-phosphatase (glucose-6-phosphatase-beta / G6Pase-beta; EC 3.1.3.9), a multi-pass integral membrane protein of the endoplasmic reticulum and a paralog of the liver/kidney/intestine-restricted G6PC1. It hydrolyses glucose-6-phosphate to glucose and inorganic phosphate (and the metabolite 1,5-anhydroglucitol-6-phosphate) with its active site facing the ER lumen, forming a covalent phosphohistidine intermediate at His167. It functions together with the ER glucose-6-phosphate transporter SLC37A4 (G6PT) to support intracellular glucose production and energy homeostasis, and is ~8x less active than G6Pase-alpha. Loss of G6PC3 causes severe congenital neutropenia type 4 (SCN4 / Dursun syndrome), in which neutrophils show endoplasmic-reticulum stress and enhanced apoptosis, accompanied by congenital cardiac and urogenital malformations and a prominent superficial venous pattern; unlike G6PC1 deficiency it is not a classic hepatic glycogen storage disease.

Existing Annotations Review

GO Term Evidence Action Reason
GO:0005783 endoplasmic reticulum
IBA
GO_REF:0000033
ACCEPT
Summary: IBA localization of G6PC3 to the endoplasmic reticulum. Correct but a generic parent of the more precise ER membrane assignment.
Reason: G6PC3 is an ER-resident enzyme with its active site facing the ER lumen; ER localization is well supported experimentally, so the phylogenetic call is sound. The more specific term is endoplasmic reticulum membrane (GO:0005789), captured elsewhere and used in core_functions.
Supporting Evidence:
PMID:25492228
G6Pase-Ξ² is an enzyme embedded in the endoplasmic reticulum membrane that catalyzes the hydrolysis of glucose-6-phosphate (G6P) to glucose and phosphate.
GO:0006094 gluconeogenesis
IBA
GO_REF:0000033
KEEP AS NON CORE
Summary: IBA involvement in gluconeogenesis, inherited from the glucose-6-phosphatase family (including hepatic orthologs).
Reason: Gluconeogenesis is a family/pathway-level assignment (the terminal dephosphorylation step is shared with the liver enzyme G6PC1). G6PC3 is ubiquitously expressed and its deficiency causes neutropenia rather than fasting hypoglycemia/glycogen storage disease, so systemic gluconeogenesis is not its core physiological role. Its ubiquitous complex with SLC37A4/G6PT supports local intracellular glucose production and energy homeostasis rather than hepatic glucose output. Retained as a valid but non-core process.
Supporting Evidence:
PMID:25492228
the ubiquitous G6Pase-Ξ²/G6PT complex maintains energy homeostasis and functionality in neutrophils and macrophages
GO:0004346 glucose-6-phosphatase activity
IBA
GO_REF:0000033
ACCEPT
Summary: IBA glucose-6-phosphatase activity, the core molecular function of G6PC3, concordant with experimental evidence.
Reason: This is the defining, experimentally established molecular function of G6PC3 (EC 3.1.3.9). It is corroborated by direct catalytic assays and mutagenesis of the active-site residues, and by the disease-mutation functional analysis. Represents the core molecular function.
Supporting Evidence:
PMID:14718531
Glc-6-Pase-beta is also a nine-transmembrane domain protein that forms a covalently bound phosphoryl enzyme intermediate during Glc-6-P hydrolysis.
GO:0016020 membrane
IBA
GO_REF:0000033
MARK AS OVER ANNOTATED
Summary: IBA generic membrane localization. Correct but uninformative given the well-established ER membrane localization.
Reason: G6PC3 is a multi-pass ER membrane protein, so "membrane" is not wrong, but it is a generic parent superseded by the specific endoplasmic reticulum membrane (GO:0005789) annotation. Marked as over-annotated in favor of the specific term.
Propagation Review
Root cause: TERM SCOPING PROBLEM
Failure modes: GRANULARITY MISMATCH
Supporting Evidence:
file:human/G6PC3/G6PC3-uniprot.txt
Multi-pass membrane protein
GO:0004346 glucose-6-phosphatase activity
IEA
GO_REF:0000120
ACCEPT
Summary: Electronic (ARBA/InterPro/RHEA/EC) assignment of glucose-6-phosphatase activity, matching the experimentally established function.
Reason: The IEA mapping (EC 3.1.3.9, RHEA:16689, InterPro glucose-6-phosphatase family) agrees with the direct experimental molecular function. Correct.
Supporting Evidence:
file:human/G6PC3/G6PC3-uniprot.txt
Reaction=D-glucose 6-phosphate + H2O = D-glucose + phosphate;
GO:0005789 endoplasmic reticulum membrane
IEA
GO_REF:0000044
ACCEPT
Summary: UniProt subcellular-location keyword mapping to ER membrane, the precise localization of G6PC3.
Reason: G6PC3 is a multi-pass ER membrane protein; this specific localization is well supported experimentally and by topology studies. This is the core cellular component.
Supporting Evidence:
file:human/G6PC3/G6PC3-uniprot.txt
SUBCELLULAR LOCATION: Endoplasmic reticulum membrane
PMID:25492228
G6Pase-Ξ² is an enzyme embedded in the endoplasmic reticulum membrane that catalyzes the hydrolysis of glucose-6-phosphate (G6P) to glucose and phosphate.
GO:0005783 endoplasmic reticulum
IEA
GO_REF:0000107
ACCEPT
Summary: Ensembl orthology-based transfer of ER localization. Correct but a generic parent of ER membrane.
Reason: ER localization is well established for G6PC3. Correct, though the specific ER membrane term is more informative and captured elsewhere.
Supporting Evidence:
PMID:25492228
G6Pase-Ξ² is an enzyme embedded in the endoplasmic reticulum membrane that catalyzes the hydrolysis of glucose-6-phosphate (G6P) to glucose and phosphate.
GO:0006094 gluconeogenesis
IEA
GO_REF:0000120
KEEP AS NON CORE
Summary: Electronic (UniPathway/ortholog) assignment of gluconeogenesis, a family/pathway-level process.
Reason: Same rationale as the IBA gluconeogenesis annotation: a valid pathway-level assignment shared across the glucose-6-phosphatase family, but not the core physiological role of the ubiquitous G6PC3, whose deficiency causes neutropenia rather than a hepatic glucose-homeostasis disorder. Kept as non-core.
Supporting Evidence:
file:human/G6PC3/G6PC3-uniprot.txt
Carbohydrate biosynthesis; gluconeogenesis.
GO:0051156 glucose 6-phosphate metabolic process
IEA
GO_REF:0000107
ACCEPT
Summary: Ortholog-based assignment of glucose 6-phosphate metabolic process, the direct metabolic process performed by G6PC3.
Reason: G6PC3 directly hydrolyses glucose-6-phosphate, so it participates in glucose 6-phosphate metabolism. This is the most directly supported biological process and is used as the core process in core_functions.
Supporting Evidence:
PMID:25492228
Both phosphatases catalyze the hydrolysis of glucose-6-phosphate (G6P) to glucose and phosphate and both are key enzymes for intracellular glucose production.
GO:0006094 gluconeogenesis
TAS
Reactome:R-HSA-70263
KEEP AS NON CORE
Summary: Reactome pathway (Gluconeogenesis) traceable assignment placing G6PC3 in the gluconeogenesis pathway.
Reason: Reactome places G6PC3 in the gluconeogenesis pathway (the terminal G6P dephosphorylation step). Valid at pathway level but non-core for the ubiquitous G6PC3, per the rationale above.
Supporting Evidence:
file:human/G6PC3/G6PC3-uniprot.txt
Carbohydrate biosynthesis; gluconeogenesis.
GO:0004346 glucose-6-phosphatase activity
EXP
PMID:14718531
Histidine 167 is the phosphate acceptor in glucose-6-phospha...
ACCEPT
Summary: Experimental demonstration of glucose-6-phosphatase (G6P hydrolase) activity, with identification of His167 as the catalytic phosphate acceptor.
Reason: Direct experimental evidence: G6Pase-beta forms a covalent phosphoryl enzyme intermediate during G6P hydrolysis, and His167 (lumenal, with active-site Arg79 and His114) is the phosphate acceptor; active-site mutants lose the intermediate. Core molecular function.
Supporting Evidence:
PMID:14718531
we demonstrated that the phosphate acceptor in Glc-6-Pase-beta is His(167) and that it lies inside the ER lumen with the active site residues, Arg(79) and His(114).
GO:0004346 glucose-6-phosphatase activity
TAS
Reactome:R-HSA-3282876
ACCEPT
Summary: Reactome traceable assignment of glucose-6-phosphatase activity (context: defective G6PC3 does not hydrolyze G6P), consistent with the core function.
Reason: Reactome records G6PC3 as the enzyme that hydrolyzes G6P; the paired "defective G6PC3" reaction underscores that loss of this activity is the disease mechanism. Consistent with the experimentally established function.
Supporting Evidence:
PMID:25492228
Fourteen missense mutations completely abolish G6Pase-Ξ² enzymatic activity
GO:0005783 endoplasmic reticulum
IDA
GO_REF:0000052
ACCEPT
Summary: Human Protein Atlas immunofluorescence (IDA) localizing G6PC3 to the endoplasmic reticulum.
Reason: Direct immunofluorescence localization to the ER, concordant with the established ER membrane residence of G6PC3. Correct; the specific ER membrane term is captured in core_functions.
Supporting Evidence:
PMID:25492228
G6Pase-Ξ² is an enzyme embedded in the endoplasmic reticulum membrane that catalyzes the hydrolysis of glucose-6-phosphate (G6P) to glucose and phosphate.
GO:0004346 glucose-6-phosphatase activity
IMP
PMID:25492228
Functional analysis of mutations in a severe congenital neut...
ACCEPT
Summary: IMP for glucose-6-phosphatase activity: functional analysis of SCN4 disease mutations shows they abolish or reduce G6P hydrolase activity.
Reason: Mutational functional analysis in a sensitive recombinant expression assay: 14 of 16 SCN4 missense mutants completely abolish G6P hydrolytic activity (S139I and R189Q retain ~49%/45%), directly establishing that G6PC3 encodes glucose-6-phosphatase activity and that loss of this activity is pathogenic. Core molecular function.
Supporting Evidence:
PMID:25492228
Fourteen missense mutations completely abolish G6Pase-Ξ² enzymatic activity while the p.S139I and p.R189Q mutations retain 49% and 45%, respectively of wild type G6Pase-Ξ² activity.
GO:0016020 membrane
HDA
PMID:19946888
Defining the membrane proteome of NK cells.
MARK AS OVER ANNOTATED
Summary: High-throughput MS membrane-proteome survey of an NK-like cell line (PMID:19946888) detecting G6PC3 among membrane proteins.
Reason: This is a generic "membrane" localization from a large-scale membrane proteomics dataset (1843 proteins identified) rather than a G6PC3-specific study. G6PC3 is specifically an ER membrane protein; the generic parent term is uninformative and superseded by endoplasmic reticulum membrane (GO:0005789). Marked as over-annotated.
Supporting Evidence:
PMID:19946888
spectrometric analysis identified 1843 proteins with high confidence scores.
GO:0005789 endoplasmic reticulum membrane
TAS
Reactome:R-HSA-3282876
ACCEPT
Summary: Reactome traceable assignment of ER membrane localization for G6PC3.
Reason: ER membrane is the precise, well-supported localization of the multi-pass G6PC3 protein. Core cellular component.
Supporting Evidence:
file:human/G6PC3/G6PC3-uniprot.txt
SUBCELLULAR LOCATION: Endoplasmic reticulum membrane
GO:0005789 endoplasmic reticulum membrane
TAS
Reactome:R-HSA-3262512
ACCEPT
Summary: Reactome traceable assignment of ER membrane localization (reaction: G6PC3 hydrolyzes G6P to form Glc and Pi, ubiquitous).
Reason: Duplicate ER membrane localization from a second Reactome reaction; correct and consistent with the multi-pass ER membrane residence of G6PC3.
Supporting Evidence:
file:human/G6PC3/G6PC3-uniprot.txt
SUBCELLULAR LOCATION: Endoplasmic reticulum membrane

Core Functions

Glucose-6-phosphatase activity: hydrolysis of glucose-6-phosphate to glucose and inorganic phosphate at the luminal face of the endoplasmic reticulum membrane, via a covalent phosphohistidine (His167) intermediate, contributing to glucose 6-phosphate metabolism and intracellular glucose production in concert with the ER G6P transporter SLC37A4.

Supporting Evidence:
  • PMID:14718531
    we demonstrated that the phosphate acceptor in Glc-6-Pase-beta is His(167) and that it lies inside the ER lumen with the active site residues, Arg(79) and His(114).
  • PMID:25492228
    Both phosphatases catalyze the hydrolysis of glucose-6-phosphate (G6P) to glucose and phosphate and both are key enzymes for intracellular glucose production.

References

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Notes

(G6PC3-notes.md)

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