Mapk1

UniProt ID: P63086
Organism: Rattus norvegicus
Review Status: INITIALIZED
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Gene Description

Mapk1 (also known as Erk2, Prkm1, p42-MAPK) encodes ERK2, the rat ortholog of the extracellular signal-regulated kinase 2. It is a proline-directed serine/threonine protein kinase (EC 2.7.11.24) of the CMGC group and the terminal effector kinase of the canonical RAS-RAF-MEK-ERK (ERK1/2) MAPK cascade. ERK2 is activated by dual phosphorylation on the TEY activation-loop motif (Thr183/Tyr185 in rat numbering, equivalent to the TEY threonine/tyrosine pair) by the upstream MAP2Ks MEK1/MEK2 (MAP2K1/MAP2K2), downstream of receptor tyrosine kinases (EGFR and other growth factor receptors), G-protein-coupled receptors, and other stimuli that activate RAS. Once activated, ERK2 phosphorylates a Ser/Thr-Pro consensus motif on hundreds of cytoplasmic and nuclear substrates (e.g., RSK kinases, ELK1 and other transcription factors, translation-control nodes, cytoskeletal and membrane scaffold proteins such as NHE1/SLC9A1). Its core molecular function is protein serine/threonine (MAP) kinase activity using ATP, and its core biological role is transduction of the ERK1/2 MAPK cascade. Subcellular localization (cytoplasm versus nucleus) is a key regulatory feature: activated ERK2 translocates to the nucleus to drive transcriptional programs, and is sequestered/exported by binding partners such as PEA-15. Because ERK2 is an extremely pleiotropic signaling hub, it is annotated to a very large number of downstream and developmental processes; most of these are context-specific consequences of cascade activity rather than the core function of the protein.

Existing Annotations Review

GO Term Evidence Action Reason
GO:0005634 nucleus
IBA
GO_REF:0000033
ACCEPT
Summary: Activated ERK2 translocates to the nucleus where it phosphorylates transcription factors; nuclear localization is well established and a core site of action.
Reason: Core localization. Activated ERK2 accumulates in the nucleus to drive transcription; supported by the phylogenetic inference and by direct evidence in this review.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
transcriptional outcomes often requiring nuclear ERK
GO:0005737 cytoplasm
IBA
GO_REF:0000033
ACCEPT
Summary: ERK2 resides in the cytoplasm in the basal state and is activated there by the cytoplasmic MEK1/2; cytoplasmic localization is a core feature.
Reason: Core localization. ERK2 is cytoplasmic in resting cells and is subject to cytoplasmic sequestration; this is the compartment of initial activation.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
NHE1/Slc9a1** can act as a **membrane scaffold** for ERK2
GO:0035556 intracellular signal transduction
IBA
GO_REF:0000033
KEEP AS NON CORE
Summary: ERK2 is a central intracellular signal-transducing kinase. This is a generic parent of the more specific ERK1/2 cascade terms.
Reason: Correct but generic. The more specific GO:0070371 (ERK1 and ERK2 cascade) better captures the core biological process; this broad parent is retained as non-core.
GO:0004674 protein serine/threonine kinase activity
IBA
GO_REF:0000033
ACCEPT
Summary: ERK2 is a proline-directed serine/threonine protein kinase. This is a core molecular function (parent of MAP kinase activity).
Reason: Core molecular function. ERK2 phosphorylates Ser/Thr-Pro motifs on substrates; well supported phylogenetically and experimentally.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
ERK family proteins are annotated under a **serine/threonine kinase domain category**
GO:0007166 cell surface receptor signaling pathway
IBA
GO_REF:0000033
KEEP AS NON CORE
Summary: ERK2 acts downstream of cell-surface receptors (RTKs, GPCRs), but this broad term is a generic parent of the specific cascade/receptor pathways.
Reason: Generic parent. The specific receptor pathways and the ERK1/2 cascade term capture this better; kept as non-core context.
GO:0004672 protein kinase activity
IEA
GO_REF:0000002
MARK AS OVER ANNOTATED
Summary: Generic parent of protein serine/threonine kinase / MAP kinase activity.
Reason: Over-general. The specific MF terms (MAP kinase activity, protein serine/threonine kinase activity) are present and preferred.
GO:0004707 MAP kinase activity
IEA
GO_REF:0000120
ACCEPT
Summary: ERK2 IS a MAP kinase; this is the most specific and accurate molecular function term for this protein.
Reason: Core molecular function. ERK2 is the canonical MAP kinase; this term is the precise MF.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
Mapk1 encodes ERK2**, a serine/threonine MAP kinase in the canonical RAS→RAF→MEK→ERK cascade
GO:0005524 ATP binding
IEA
GO_REF:0000002
ACCEPT
Summary: ERK2 binds ATP in its kinase domain and transfers the gamma-phosphate to substrates; a core molecular function of the enzyme.
Reason: Core molecular function. ATP binding is required for the phosphotransfer reaction; experimentally demonstrated (PMID:15027896) and assay-confirmed in the deep research.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
an in vitro kinase assay with active TEY-phosphorylated ERK2 and an ATPγS analog
GO:0005634 nucleus
IEA
GO_REF:0000044
ACCEPT
Summary: Nuclear localization (duplicate of the IBA nucleus annotation).
Reason: Core localization, consistent with the IBA annotation and direct evidence.
GO:0005654 nucleoplasm
IEA
GO_REF:0000117
ACCEPT
Summary: Nucleoplasm is a more specific child of nucleus; ERK2 acts within the nucleoplasm on transcription factors.
Reason: Consistent specific nuclear localization; supported by IDA evidence (PMID:7889942) elsewhere in this review.
GO:0005737 cytoplasm
IEA
GO_REF:0000044
ACCEPT
Summary: Cytoplasmic localization (duplicate of the IBA cytoplasm annotation).
Reason: Core localization.
GO:0005769 early endosome
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: ERK signaling can be organized on endosomal compartments, but early endosome is a minor/context-specific localization, not a core site.
Reason: Context-specific localization tied to endosomal signaling scaffolds; not a core compartment for ERK2 function.
GO:0005770 late endosome
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: Context-specific endosomal localization (see early endosome).
Reason: Minor/context-specific localization, not core.
GO:0005794 Golgi apparatus
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: Golgi-localized ERK pools exist and ERK can regulate Golgi dynamics, but this is a specialized localization rather than the core site of action.
Reason: Specialized localized signaling pool; non-core.
GO:0005813 centrosome
IEA
GO_REF:0000044
KEEP AS NON CORE
Summary: Centrosomal localization is reported in mitotic contexts; specialized, not core.
Reason: Context-specific localization (mitosis); non-core.
GO:0005819 spindle
IEA
GO_REF:0000044
KEEP AS NON CORE
Summary: Spindle localization in mitosis is a specialized, context-specific site.
Reason: Context-specific mitotic localization; non-core.
GO:0005901 caveola
IEA
GO_REF:0000044
KEEP AS NON CORE
Summary: ERK can be recruited to caveolae (e.g., via MURC/Cavin-4) in specialized signaling, supported by IDA (PMID:24567387); specialized localization.
Reason: Context-specific membrane microdomain localization; non-core but experimentally supported.
GO:0005925 focal adhesion
IEA
GO_REF:0000120
KEEP AS NON CORE
Summary: ERK localizes to focal adhesions in migration contexts; specialized localization.
Reason: Context-specific localization linked to cell migration; non-core.
GO:0006357 regulation of transcription by RNA polymerase II
IEA
GO_REF:0000108
KEEP AS NON CORE
Summary: Nuclear ERK2 regulates Pol II transcription by phosphorylating transcription factors (e.g., ELK1). This is a downstream consequence of cascade activity rather than the core function.
Reason: Genuine but downstream/indirect process; ERK2 regulates transcription via substrate phosphorylation. Kept as non-core.
GO:0032872 regulation of stress-activated MAPK cascade
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: ERK2 can cross-regulate stress-activated MAPK (p38/JNK) cascades, but this is a secondary crosstalk role, not core.
Reason: Crosstalk/regulatory role; non-core relative to the ERK1/2 cascade itself.
GO:0035094 response to nicotine
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: ERK activation downstream of nicotinic receptors is a stimulus-specific response, not a core function.
Reason: Stimulus-specific response (also supported by IGI PMID:11404397); non-core.
GO:0045727 positive regulation of translation
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: ERK2 promotes translation via downstream nodes (e.g., RSK/MNK, eIF4E pathway, EIF4EBP1, EEF2K). This is a downstream consequence of cascade activity.
Reason: Downstream regulatory consequence (also IMP PMID:15027896); non-core.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
ERK2 is also linked to translation-control nodes including Eif4ebp1 and Eef2k
GO:0046697 decidualization
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: Decidualization is a tissue-specific developmental process downstream of MAPK activation; not a core ERK2 function.
Reason: Tissue-specific developmental process (also IDA PMID:21248290); non-core.
GO:0051493 regulation of cytoskeleton organization
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: ERK2 phosphorylates cytoskeletal regulators, influencing cytoskeleton organization; a downstream effect.
Reason: Downstream effector consequence; non-core.
GO:0070371 ERK1 and ERK2 cascade
IEA
GO_REF:0000117
ACCEPT
Summary: This is the defining biological process for ERK2 - it IS one of the two terminal kinases of the ERK1/2 cascade. Core BP.
Reason: Core biological process. ERK2 is a defining component of the ERK1 and ERK2 cascade.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
ERK1/2 (MAPK3/MAPK1) are described as **terminal kinases** in the canonical **RAS→RAF→MEK→ERK** cascade
GO:0071375 cellular response to peptide hormone stimulus
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: ERK activation downstream of peptide hormones is a stimulus-specific response.
Reason: Stimulus-specific response; non-core.
GO:0071396 cellular response to lipid
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: Stimulus-specific cellular response.
Reason: Stimulus-specific response; non-core.
GO:0072584 caveolin-mediated endocytosis
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: A specialized endocytosis process where ERK has been implicated; downstream/context-specific.
Reason: Context-specific process; non-core.
GO:0090170 regulation of Golgi inheritance
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: ERK2 has been implicated in mitotic Golgi partitioning; specialized downstream process.
Reason: Specialized mitotic process; non-core.
GO:0106310 protein serine kinase activity
IEA
GO_REF:0000116
ACCEPT
Summary: ERK2 phosphorylates serine residues; a more specific child of protein serine/threonine kinase activity. Accurate.
Reason: Accurate specific MF; ERK2 is a Ser/Thr (proline-directed) kinase.
GO:2000641 regulation of early endosome to late endosome transport
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: Specialized endosomal trafficking process linked to ERK; downstream.
Reason: Context-specific process; non-core.
GO:0005515 protein binding
IPI
PMID:21070949
Phosphorylation of DCC by ERK2 is facilitated by direct dock...
MARK AS OVER ANNOTATED
Summary: This IPI annotation reflects the ERK2-DCC docking interaction (ERK2 phosphorylates DCC via direct docking). The generic protein binding term is uninformative.
Reason: The protein binding term is non-informative per curation guidelines. The underlying interaction (DCC docking/substrate) is better captured by the kinase activity and substrate-docking functions.
GO:0106310 protein serine kinase activity
IMP
PMID:29959233
Desmoplakin maintains gap junctions by inhibiting Ras/MAPK a...
ACCEPT
Summary: ERK2 serine kinase activity demonstrated in the context of Ras/MAPK regulation of connexin-43/gap junctions. Accurate MF.
Reason: Accurate specific molecular function with experimental support.
Supporting Evidence:
PMID:29959233
increased phosphorylation of S279/282 of Cx43, which signals clathrin-mediated internalization and subsequent lysosomal degradation of Cx43
GO:0045880 positive regulation of smoothened signaling pathway
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: Crosstalk between ERK and Hedgehog/Smoothened signaling is reported but indirect; not a core ERK2 function and based on sequence-similarity transfer.
Reason: Indirect crosstalk role from ISS transfer; non-core.
GO:0042802 identical protein binding
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Refers to ERK2 homodimerization. While ERK2 can dimerize, this is a relatively uninformative interaction term.
Reason: ERK2 homodimerization is documented but its functional relevance is debated; retained as non-core rather than core function.
GO:0005654 nucleoplasm
ISO
GO_REF:0000121
ACCEPT
Summary: Nucleoplasm localization (ISO duplicate). Consistent.
Reason: Consistent specific nuclear localization.
GO:0005829 cytosol
ISO
GO_REF:0000121
ACCEPT
Summary: Cytosolic localization; consistent with cytoplasmic localization and the site of basal ERK2 and MEK-mediated activation.
Reason: Core localization (cytosolic pool), consistent with TAS and other evidence.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
NHE1/Slc9a1** can act as a **membrane scaffold** for ERK2
GO:0004707 MAP kinase activity
IDA
PMID:7889942
ERK phosphorylation potentiates Elk-1-mediated ternary compl...
ACCEPT
Summary: Direct demonstration of ERK MAP kinase activity (Elk-1 phosphorylation / ternary complex). Core MF with strong experimental support.
Reason: Core molecular function with direct experimental evidence.
GO:0150078 positive regulation of neuroinflammatory response
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: A tissue/context-specific downstream process inferred by orthology; not a core ERK2 function.
Reason: Context-specific downstream process from ISO transfer; non-core.
GO:0061514 interleukin-34-mediated signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK acts downstream of IL-34/CSF1R signaling; a stimulus-specific pathway inferred by orthology.
Reason: Stimulus-specific signaling context; non-core.
GO:0000165 MAPK cascade
ISO
GO_REF:0000121
ACCEPT
Summary: ERK2 is a core component of the MAPK cascade; this is the generic parent of the ERK1/2 cascade term.
Reason: Core biological process (generic parent of ERK1/2 cascade). ERK2 is a terminal MAPK of this cascade.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
concludes that EGF activates the canonical MAPK pathway in this native rat tissue context
GO:0007173 epidermal growth factor receptor signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 is a key effector of EGFR signaling; this is a major upstream pathway that activates the ERK1/2 cascade. Well supported in rat tissue.
Reason: Genuine and important upstream-receptor pathway, but it is the receptor context that activates ERK2 rather than ERK2's own core function. Kept as non-core; strongly corroborated by rat IMCD EGF data.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
pathway enrichment confirms engagement of **RAF–MEK–ERK signaling**
GO:0032206 positive regulation of telomere maintenance
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Downstream/indirect process inferred by orthology; not a core function.
Reason: Indirect downstream process; non-core.
GO:0004707 MAP kinase activity
ISO
GO_REF:0000121
ACCEPT
Summary: MAP kinase activity (ISO duplicate). Core MF.
Reason: Core molecular function (orthology-inferred duplicate of the IDA/IEA MAP kinase activity annotations).
GO:0045542 positive regulation of cholesterol biosynthetic process
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Indirect downstream metabolic process inferred by orthology.
Reason: Indirect downstream process; non-core.
GO:0061431 cellular response to methionine
IEP
PMID:22676582
Activation of Nrf2 is required for up-regulation of the π cl...
KEEP AS NON CORE
Summary: ERK activation under methionine starvation (Nrf2/GST context); a stimulus-specific cellular response inferred from expression/phenotype.
Reason: Stimulus-specific response (IEP); non-core.
GO:0071380 cellular response to prostaglandin E stimulus
IEP
PMID:11875501
Prostaglandin E2 transactivates EGF receptor: a novel mechan...
KEEP AS NON CORE
Summary: ERK activation downstream of PGE2/EGFR transactivation; stimulus-specific response.
Reason: Stimulus-specific response (IEP); non-core.
GO:0071320 cellular response to cAMP
IEP
PMID:8223435
cAMP antagonizes p21ras-directed activation of extracellular...
KEEP AS NON CORE
Summary: cAMP modulates ERK2 activation (cAMP antagonizes Ras-directed ERK2 activation); stimulus-specific response.
Reason: Stimulus-specific response/crosstalk (IEP); non-core.
GO:0014069 postsynaptic density
IEP
PMID:7478291
ERK2-type mitogen-activated protein kinase (MAPK) and its su...
KEEP AS NON CORE
Summary: ERK2 detected in postsynaptic density fractions from rat brain; a neuronal localization. Specialized.
Reason: Tissue-specific neuronal localization; non-core but experimentally observed in rat brain.
GO:0014069 postsynaptic density
IDA
PMID:7478291
ERK2-type mitogen-activated protein kinase (MAPK) and its su...
KEEP AS NON CORE
Summary: Direct observation of ERK2 in postsynaptic density fractions (rat brain).
Reason: Tissue-specific neuronal localization with direct evidence; non-core.
GO:0032355 response to estradiol
IEP
PMID:15893655
17-Beta estradiol rapidly enhances extracellular signal-regu...
KEEP AS NON CORE
Summary: Estradiol rapidly enhances ERK2 phosphorylation in rat brain; stimulus-specific response.
Reason: Stimulus-specific response (IEP); non-core.
GO:0036120 cellular response to platelet-derived growth factor stimulus
IEP
PMID:8246947
Epidermal growth factor induces phosphorylation of extracell...
KEEP AS NON CORE
Summary: ERK2 is activated downstream of PDGF; a growth-factor-specific response.
Reason: Stimulus-specific response (IEP); non-core.
GO:0071364 cellular response to epidermal growth factor stimulus
IEP
PMID:8246947
Epidermal growth factor induces phosphorylation of extracell...
KEEP AS NON CORE
Summary: ERK2 is activated downstream of EGF; well supported in rat tissue (IMCD EGF phosphoproteomics shows TEY phosphorylation of Mapk1). Stimulus response.
Reason: Stimulus-specific response, but strongly corroborated; non-core relative to the cascade itself.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
Dual phosphorylation in the TEY activation segment region** is directly observed for rat Mapk1/ERK2
GO:0033574 response to testosterone
IEP
PMID:22265242
Extracellular signal-regulated kinase 2 signaling in the hip...
KEEP AS NON CORE
Summary: ERK2 in dentate gyrus mediates antidepressant effects of testosterone; stimulus-specific.
Reason: Stimulus-specific response (IEP); non-core.
GO:0044849 estrous cycle
IEP
PMID:22521590
Sex differences in social interaction behaviors in rats are ...
KEEP AS NON CORE
Summary: ERK2 expression correlates with estrous-cycle-related behavior; an organism-level physiological context, not a molecular role.
Reason: Physiological/behavioral context (IEP); non-core.
GO:0042220 response to cocaine
IEP
PMID:19457111
Signaling pathway adaptations and novel protein kinase A sub...
KEEP AS NON CORE
Summary: ERK signaling adaptations in cocaine sensitization; stimulus-specific response.
Reason: Stimulus-specific response (IEP); non-core.
GO:0042542 response to hydrogen peroxide
IEP
PMID:11679970
Defective mitogen-activated protein kinase (ERK2) signaling ...
KEEP AS NON CORE
Summary: ERK2 signaling altered by oxidative stress; stimulus-specific response.
Reason: Stimulus-specific response (IEP); non-core.
GO:0097305 response to alcohol
IEP
PMID:21790671
Elevated activation of ERK1 and ERK2 accompany enhanced live...
KEEP AS NON CORE
Summary: ERK1/2 activation accompanies alcohol-induced liver injury; stimulus-specific response.
Reason: Stimulus-specific response (IEP); non-core.
GO:1990314 cellular response to insulin-like growth factor stimulus
IEP
PMID:9235900
Insulin-like growth factor-I rapidly activates multiple sign...
KEEP AS NON CORE
Summary: IGF-I rapidly activates ERK2 in cardiac myocytes; growth-factor-specific response.
Reason: Stimulus-specific response (IEP); non-core.
GO:0048009 insulin-like growth factor receptor signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 is an effector of IGF-1R signaling; an upstream receptor pathway context inferred by orthology.
Reason: Upstream-receptor pathway context; non-core.
GO:0008286 insulin receptor signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 is an effector of insulin receptor signaling; upstream pathway context inferred by orthology.
Reason: Upstream-receptor pathway context; non-core.
GO:0014044 Schwann cell development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: A developmental process where ERK signaling is required; tissue/lineage specific, downstream of the cascade.
Reason: Developmental process inferred by orthology; non-core.
GO:0042552 myelination
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process where ERK signaling participates; downstream and tissue-specific.
Reason: Developmental process inferred by orthology; non-core.
GO:0038133 ERBB2-ERBB3 signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 is an effector of ERBB2-ERBB3 signaling; upstream receptor pathway context inferred by orthology.
Reason: Upstream-receptor pathway context; non-core.
GO:0005634 nucleus
ISO
GO_REF:0000121
ACCEPT
Summary: Nuclear localization (ISO duplicate). Consistent core localization.
Reason: Core localization, consistent with other nucleus annotations.
GO:0010759 positive regulation of macrophage chemotaxis
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: A cell-type-specific downstream process inferred by orthology.
Reason: Cell-type-specific downstream process; non-core.
GO:0120041 positive regulation of macrophage proliferation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: A cell-type-specific downstream process inferred by orthology.
Reason: Cell-type-specific downstream process; non-core.
GO:0042307 positive regulation of protein import into nucleus
IMP
PMID:19524539
LysRS serves as a key signaling molecule in the immune respo...
KEEP AS NON CORE
Summary: From the LysRS/Ap4A study; ERK2 phosphorylation of LysRS affecting its nuclear function. A specific downstream regulatory effect.
Reason: Specific downstream regulatory effect (IMP); non-core.
GO:0060045 positive regulation of cardiac muscle cell proliferation
IMP
PMID:26884868
MAPK1 up-regulates the expression of MALAT1 to promote the p...
KEEP AS NON CORE
Summary: MAPK1 promotes cardiomyocyte proliferation via MALAT1/PI3K-AKT; a cell-type-specific downstream process.
Reason: Cell-type-specific downstream process (IMP); non-core.
GO:0003690 double-stranded DNA binding
IDA
PMID:26950759
Phosphorylation or Mutation of the ERK2 Activation Loop Alte...
KEEP AS NON CORE
Summary: The cited study shows that ERK2 activation-loop phosphorylation/mutation alters oligonucleotide binding; ERK2 can bind DNA. This is an unusual, non-catalytic moonlighting activity, not the core kinase function.
Reason: Experimentally observed but non-canonical moonlighting DNA-binding activity; not the core kinase function. Retained as non-core.
GO:0006468 protein phosphorylation
IDA
PMID:26950759
Phosphorylation or Mutation of the ERK2 Activation Loop Alte...
KEEP AS NON CORE
Summary: Generic protein phosphorylation; the catalytic output of ERK2 kinase activity. Accurate but generic relative to the MF terms.
Reason: Generic BP that is the direct output of the kinase activity; the MF terms (MAP kinase activity) capture this more precisely. Non-core.
GO:0046697 decidualization
IDA
PMID:21248290
Ovarian steroid receptors and activated MAPK in the regional...
KEEP AS NON CORE
Summary: MAPK activation in regional decidualization in rats; tissue-specific developmental process.
Reason: Tissue-specific developmental process; non-core.
GO:0019902 phosphatase binding
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 binds dual-specificity phosphatases (DUSPs/MKPs) that dephosphorylate it; a genuine regulatory interaction but not a core function.
Reason: Regulatory protein interaction (with MKPs); non-core, more informative than generic protein binding.
GO:0004674 protein serine/threonine kinase activity
ISO
GO_REF:0000121
ACCEPT
Summary: Protein serine/threonine kinase activity (ISO duplicate). Core MF.
Reason: Core molecular function (orthology-inferred duplicate).
GO:0071356 cellular response to tumor necrosis factor
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Stimulus-specific cellular response inferred by orthology.
Reason: Stimulus-specific response; non-core.
GO:0030641 regulation of cellular pH
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Reflects ERK2 phosphorylation of the NHE1/SLC9A1 Na+/H+ exchanger; a specific downstream effect, corroborated in rat IMCD (ERK2 phosphorylates NHE1 at Ser727/Ser730).
Reason: Specific downstream effector consequence (NHE1 phosphorylation); non-core but corroborated.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
NHE1/Slc9a1** can act as a **membrane scaffold** for ERK2
GO:0005515 protein binding
IPI
PMID:24567387
MURC/Cavin-4 facilitates recruitment of ERK to caveolae and ...
MARK AS OVER ANNOTATED
Summary: ERK interaction with MURC/Cavin-4 (caveolar recruitment). The generic protein binding term is uninformative.
Reason: The protein binding term is non-informative per curation guidelines; the caveolar localization is captured by the caveola term.
GO:0005737 cytoplasm
IDA
PMID:24567387
MURC/Cavin-4 facilitates recruitment of ERK to caveolae and ...
ACCEPT
Summary: Cytoplasmic localization with direct evidence. Core localization.
Reason: Core localization with direct experimental support.
GO:0005886 plasma membrane
IDA
PMID:24567387
MURC/Cavin-4 facilitates recruitment of ERK to caveolae and ...
KEEP AS NON CORE
Summary: ERK recruited to plasma membrane/caveolae in cardiac hypertrophy context; a specialized localized pool.
Reason: Context-specific membrane recruitment; non-core.
GO:0005901 caveola
IDA
PMID:24567387
MURC/Cavin-4 facilitates recruitment of ERK to caveolae and ...
KEEP AS NON CORE
Summary: Direct evidence of ERK recruitment to caveolae via MURC/Cavin-4. Specialized localization.
Reason: Context-specific membrane microdomain localization with direct evidence; non-core.
GO:0005515 protein binding
IPI
PMID:12944431
DOC1R: a MAP kinase substrate that control microtubule organ...
MARK AS OVER ANNOTATED
Summary: DOC1R interaction (a MAP kinase substrate in oocytes). The generic protein binding term is uninformative.
Reason: The protein binding term is non-informative; the substrate relationship is captured by kinase activity.
GO:0035094 response to nicotine
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Stimulus-specific response (ISO duplicate of the nicotine annotations).
Reason: Stimulus-specific response; non-core.
GO:0035094 response to nicotine
IGI
PMID:11404397
Beta-amyloid activates the mitogen-activated protein kinase ...
KEEP AS NON CORE
Summary: Beta-amyloid activates MAPK cascade via alpha7 nicotinic receptors; stimulus-specific response with genetic-interaction evidence.
Reason: Stimulus-specific response (IGI); non-core.
GO:0034198 cellular response to amino acid starvation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Stimulus-specific cellular response inferred by orthology.
Reason: Stimulus-specific response; non-core.
GO:0051403 stress-activated MAPK cascade
ISO
GO_REF:0000121
MARK AS OVER ANNOTATED
Summary: ERK2 is not part of the stress-activated (p38/JNK) MAPK cascade itself; this annotation conflates the ERK cascade with stress-activated cascades.
Reason: ERK2 is the terminal kinase of the ERK1/2 (mitogen-activated) cascade, not a component of the stress-activated (p38/JNK) cascade. This orthology-inferred term likely over-annotates; ERK2's relationship to stress cascades is regulatory crosstalk (captured by GO:0032872), not membership.
Propagation Review
Root cause: TERM SCOPING PROBLEM
Failure modes: ROLE CONFLATION
Sources checked:
UniProtKB:P28482 · human MAPK1 SUPPORTS SOURCE BUT NOT TARGET
Human MAPK1 carries the term by IDA (PMID:11096076), but ERK2's relationship to the stress-activated cascades is crosstalk; membership in the p38/JNK cascade does not transfer.
GO:0004707 MAP kinase activity
IMP
PMID:19524539
LysRS serves as a key signaling molecule in the immune respo...
ACCEPT
Summary: MAP kinase activity demonstrated via LysRS phosphorylation. Core MF.
Reason: Core molecular function with experimental support.
GO:0015966 diadenosine tetraphosphate biosynthetic process
IMP
PMID:19524539
LysRS serves as a key signaling molecule in the immune respo...
KEEP AS NON CORE
Summary: ERK2 phosphorylation of LysRS triggers Ap4A production in immune signaling; an indirect downstream consequence, not an ERK2 enzymatic activity.
Reason: Indirect downstream consequence via substrate (LysRS); ERK2 does not itself synthesize Ap4A. Non-core.
GO:0045893 positive regulation of DNA-templated transcription
IMP
PMID:19524539
LysRS serves as a key signaling molecule in the immune respo...
KEEP AS NON CORE
Summary: ERK2 promotes transcription via substrate phosphorylation; downstream regulatory consequence.
Reason: Downstream transcriptional regulation via substrates; non-core.
GO:0070371 ERK1 and ERK2 cascade
IMP
PMID:19524539
LysRS serves as a key signaling molecule in the immune respo...
ACCEPT
Summary: ERK1/2 cascade (IMP). Core biological process.
Reason: Core biological process with experimental support.
GO:0030278 regulation of ossification
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process where ERK signaling participates; tissue-specific, downstream.
Reason: Developmental process inferred by orthology; non-core.
GO:0007507 heart development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK1/2 signaling is required for heart development; a pleiotropic developmental process downstream of the cascade.
Reason: Developmental process inferred by orthology; non-core.
GO:0014032 neural crest cell development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process where ERK signaling participates; downstream.
Reason: Developmental process inferred by orthology; non-core.
GO:0030878 thyroid gland development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process inferred by orthology; downstream.
Reason: Developmental process; non-core.
GO:0042473 outer ear morphogenesis
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process inferred by orthology (RASopathy-related); downstream.
Reason: Developmental process; non-core.
GO:0048538 thymus development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process inferred by orthology; downstream.
Reason: Developmental process; non-core.
GO:0060324 face development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process inferred by orthology (RASopathy-related); downstream.
Reason: Developmental process; non-core.
GO:0061308 cardiac neural crest cell development involved in heart development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process inferred by orthology; downstream.
Reason: Developmental process; non-core.
GO:0060020 Bergmann glial cell differentiation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Cell-type-specific developmental process inferred by orthology; downstream.
Reason: Developmental process; non-core.
GO:0070371 ERK1 and ERK2 cascade
ISO
GO_REF:0000121
ACCEPT
Summary: ERK1/2 cascade (ISO duplicate). Core biological process.
Reason: Core biological process (orthology-inferred duplicate).
GO:0006468 protein phosphorylation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Generic protein phosphorylation (the catalytic output). Generic relative to the MF terms.
Reason: Generic BP output of kinase activity; non-core.
GO:0060425 lung morphogenesis
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process inferred by orthology; downstream.
Reason: Developmental process; non-core.
GO:0060440 trachea formation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Developmental process inferred by orthology; downstream.
Reason: Developmental process; non-core.
GO:0060291 long-term synaptic potentiation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK signaling contributes to LTP; a neuronal physiological process downstream of the cascade.
Reason: Neuronal physiological process inferred by orthology; non-core.
GO:0005737 cytoplasm
ISS
GO_REF:0000024
ACCEPT
Summary: Cytoplasmic localization (ISS duplicate). Core localization.
Reason: Core localization.
GO:0072686 mitotic spindle
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: Mitotic spindle localization (specific child of spindle). Specialized mitotic localization.
Reason: Context-specific mitotic localization; non-core.
GO:0004707 MAP kinase activity
IMP
PMID:16955078
Alterations in mammalian target of rapamycin signaling pathw...
ACCEPT
Summary: MAP kinase activity (mTOR signaling/TBI context). Core MF.
Reason: Core molecular function with experimental support.
GO:0018105 peptidyl-serine phosphorylation
IMP
PMID:16955078
Alterations in mammalian target of rapamycin signaling pathw...
KEEP AS NON CORE
Summary: ERK2 phosphorylates serine residues on substrates; a specific child of protein phosphorylation describing the catalytic output.
Reason: Describes the catalytic output (serine phosphorylation); the MF terms capture this more precisely. Non-core.
GO:0019901 protein kinase binding
IPI
PMID:16943189
cGMP-dependent protein kinase type I inhibits TAB1-p38 mitog...
KEEP AS NON CORE
Summary: ERK2 binds upstream/partner kinases (e.g., TAB1 context); a more informative interaction term than generic protein binding.
Reason: Informative protein-interaction term reflecting ERK2 binding to kinases in its signaling module; non-core.
GO:0005654 nucleoplasm
TAS
Reactome:R-NUL-3245934
ACCEPT
Summary: Nucleoplasm localization, from a Reactome reaction (Mapk1 phosphorylates ERF). Consistent core nuclear localization.
Reason: Consistent specific nuclear localization (TAS from Reactome).
GO:0038127 ERBB signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 is an effector of ERBB receptor signaling; upstream pathway context inferred by orthology.
Reason: Upstream-receptor pathway context; non-core.
GO:0005737 cytoplasm
ISO
GO_REF:0000121
ACCEPT
Summary: Cytoplasmic localization (ISO duplicate). Core localization.
Reason: Core localization.
GO:0070849 response to epidermal growth factor
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: ERK2 responds to EGF; strongly supported in rat tissue (IMCD EGF phosphoproteomics). Stimulus response.
Reason: Stimulus-specific response; non-core but well corroborated.
Supporting Evidence:
file:rat/Mapk1/Mapk1-deep-research-falcon.md
concludes that EGF activates the canonical MAPK pathway in this native rat tissue context
GO:0070849 response to epidermal growth factor
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Response to EGF (ISO duplicate). Stimulus response.
Reason: Stimulus-specific response; non-core.
GO:0018105 peptidyl-serine phosphorylation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Serine phosphorylation output (ISO duplicate). Generic catalytic output.
Reason: Describes the catalytic output; non-core relative to MF terms.
GO:0018105 peptidyl-serine phosphorylation
IDA
PMID:7768935
Phosphorylation of tristetraprolin, a potential zinc finger ...
KEEP AS NON CORE
Summary: Direct demonstration of ERK2 serine phosphorylation of tristetraprolin in vitro. Catalytic output.
Reason: Direct evidence for the catalytic output (serine phosphorylation); the MF terms capture this more precisely. Non-core.
GO:0005634 nucleus
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
ACCEPT
Summary: Nuclear localization from a review of ERK signaling across compartments. Core localization.
Reason: Core localization (TAS).
GO:0005739 mitochondrion
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: A mitochondrial ERK pool is reported; a minor specialized localization.
Reason: Minor/specialized localization; non-core.
GO:0005769 early endosome
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: Endosomal ERK signaling pool; context-specific localization.
Reason: Context-specific localization; non-core.
GO:0005770 late endosome
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: Endosomal ERK signaling pool; context-specific localization.
Reason: Context-specific localization; non-core.
GO:0005794 Golgi apparatus
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: Golgi-associated ERK pool; specialized localization.
Reason: Specialized localization; non-core.
GO:0005829 cytosol
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
ACCEPT
Summary: Cytosolic localization. Core localization (the basal pool).
Reason: Core localization (cytosolic pool, TAS).
GO:0005856 cytoskeleton
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: ERK associates with cytoskeletal structures in some contexts; specialized localization.
Reason: Context-specific localization; non-core.
GO:0005901 caveola
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: Caveolar ERK pool; specialized localization.
Reason: Specialized localization; non-core.
GO:0005925 focal adhesion
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: Focal-adhesion-associated ERK pool; specialized localization.
Reason: Specialized localization; non-core.
GO:0032872 regulation of stress-activated MAPK cascade
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: ERK crosstalk regulating stress-activated MAPK cascades; secondary regulatory role.
Reason: Crosstalk/regulatory role; non-core.
GO:0051493 regulation of cytoskeleton organization
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: ERK phosphorylation of cytoskeletal regulators; downstream effect.
Reason: Downstream effector consequence; non-core.
GO:0072584 caveolin-mediated endocytosis
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: Specialized endocytic process where ERK is implicated; downstream.
Reason: Context-specific process; non-core.
GO:0090170 regulation of Golgi inheritance
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: ERK role in mitotic Golgi partitioning; specialized process.
Reason: Specialized mitotic process; non-core.
GO:2000641 regulation of early endosome to late endosome transport
TAS
PMID:19565474
The ERK signaling cascade--views from different subcellular ...
KEEP AS NON CORE
Summary: Specialized endosomal trafficking process linked to ERK; downstream.
Reason: Context-specific process; non-core.
GO:0005515 protein binding
IPI
PMID:19200235
Dopamine promotes striatal neuronal apoptotic death via ERK ...
MARK AS OVER ANNOTATED
Summary: Generic protein binding from a dopamine/ERK apoptosis study; uninformative.
Reason: The protein binding term is non-informative per curation guidelines.
GO:0010800 positive regulation of peptidyl-threonine phosphorylation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: A downstream regulatory consequence (promoting threonine phosphorylation of targets) inferred by orthology.
Reason: Downstream regulatory consequence; non-core.
GO:0031143 pseudopodium
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Pseudopodium localization inferred by orthology (migration context); specialized localization.
Reason: Context-specific localization; non-core.
GO:0005739 mitochondrion
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Mitochondrial ERK pool (ISO duplicate); minor specialized localization.
Reason: Minor/specialized localization; non-core.
GO:0033598 mammary gland epithelial cell proliferation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Cell-type-specific downstream proliferation process inferred by orthology.
Reason: Cell-type-specific downstream process; non-core.
GO:0008353 RNA polymerase II CTD heptapeptide repeat kinase activity
ISO
GO_REF:0000121
MARK AS OVER ANNOTATED
Summary: This term implies ERK2 phosphorylates the Pol II CTD as a CTD kinase. ERK2 is a proline-directed kinase and can phosphorylate Ser-Pro sites including in the CTD, but assigning a dedicated CTD-kinase MF (typically reserved for CDKs) is likely an over-annotation by orthology transfer.
Reason: ERK2's role as a bona fide Pol II CTD kinase is not its established core function; this orthology-inferred specific MF over-annotates the protein. The canonical CTD kinases are CDK7/CDK9/CDK12. Marked as over-annotated.
Propagation Review
Root cause: TERM SCOPING PROBLEM
Failure modes: GRANULARITY MISMATCH
Sources checked:
MGI:MGI:1346858 · mouse Mapk1 SUPPORTS SOURCE BUT NOT TARGET
The mouse donor (UniProtKB:P63085) carries a single GO:0008353 annotation, an IDA cited to PMID:12721286 (verified against QuickGO; that paper is titled for the SCP1 CTD phosphatase, and the cached record here is abstract-only, so the ERK2 assay supporting the IDA is visible to the curator but not in this cache). ERK2 being proline-directed makes such an in vitro CTD-phosphorylation result unsurprising, but a dedicated Pol II CTD-kinase molecular function over-reads that single donor IDA for the rat gene.
GO:0009636 response to toxic substance
IDA
PMID:17651772
MAPK-ERK activation in kidney of male rats chronically fed o...
KEEP AS NON CORE
Summary: ERK activation in kidney upon ochratoxin A exposure; stimulus-specific response.
Reason: Stimulus-specific response; non-core.
GO:0004674 protein serine/threonine kinase activity
IDA
PMID:7768935
Phosphorylation of tristetraprolin, a potential zinc finger ...
ACCEPT
Summary: Direct evidence of ERK2 Ser/Thr kinase activity (TTP phosphorylation). Core MF. The deep research notes that ERK1/2 substrates contain a Ser/Thr-Pro consensus.
Reason: Core molecular function with direct experimental support.
GO:0060716 labyrinthine layer blood vessel development
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Placental developmental process inferred by orthology; downstream.
Reason: Developmental process; non-core.
GO:0005654 nucleoplasm
IDA
PMID:7889942
ERK phosphorylation potentiates Elk-1-mediated ternary compl...
ACCEPT
Summary: Direct evidence of nucleoplasmic ERK (Elk-1 phosphorylation context). Core nuclear localization.
Reason: Core nuclear localization with direct evidence.
GO:0005515 protein binding
IPI
PMID:15781236
Caveolin-2 regulation of the cell cycle in response to insul...
MARK AS OVER ANNOTATED
Summary: Caveolin-2/insulin/cell-cycle interaction context; the generic protein binding term is uninformative.
Reason: The protein binding term is non-informative per curation guidelines.
GO:0032991 protein-containing complex
IDA
PMID:15781236
Caveolin-2 regulation of the cell cycle in response to insul...
MARK AS OVER ANNOTATED
Summary: ERK in a protein complex; generic and uninformative as a cellular component.
Reason: Generic component term that adds little functional information; the specific complexes/scaffolds are not characterized here.
GO:0031435 mitogen-activated protein kinase kinase kinase binding
IPI
PMID:12049732
The PHD domain of MEKK1 acts as an E3 ubiquitin ligase and m...
KEEP AS NON CORE
Summary: ERK2 interacts with MEKK1 (a MAP3K) which ubiquitinates ERK1/2. An informative interaction within the cascade module.
Reason: Informative protein-interaction term reflecting ERK2 binding within the MAPK module; non-core.
IDA
PMID:9714150
Immunolocalization of the mitogen-activated protein kinases ...
KEEP AS NON CORE
Summary: ERK2 (p42MAPK) immunolocalized to axons in rat CNS; neuronal subcellular localization.
Reason: Tissue-specific neuronal localization with direct evidence; non-core.
GO:0032839 dendrite cytoplasm
IDA
PMID:9714150
Immunolocalization of the mitogen-activated protein kinases ...
KEEP AS NON CORE
Summary: ERK2 immunolocalized to dendritic cytoplasm in rat CNS; neuronal localization.
Reason: Tissue-specific neuronal localization with direct evidence; non-core.
GO:0043204 perikaryon
IDA
PMID:9714150
Immunolocalization of the mitogen-activated protein kinases ...
KEEP AS NON CORE
Summary: ERK2 immunolocalized to the perikaryon (neuronal cell body) in rat CNS.
Reason: Tissue-specific neuronal localization with direct evidence; non-core.
GO:0005829 cytosol
TAS
Reactome:R-NUL-997411
ACCEPT
Summary: Cytosolic localization from a Reactome reaction (AGER binds rat ERK1/2). Core localization.
Reason: Core localization (cytosolic pool, TAS).
GO:0050853 B cell receptor signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 is an effector downstream of the B cell receptor; immune-cell pathway context inferred by orthology.
Reason: Cell-type-specific upstream pathway context; non-core.
GO:0050852 T cell receptor signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK2 is an effector downstream of the T cell receptor; immune-cell pathway context inferred by orthology.
Reason: Cell-type-specific upstream pathway context; non-core.
GO:0004674 protein serine/threonine kinase activity
IC
PMID:15027896
Angiotensin II-induced ERK1/ERK2 activation and protein synt...
ACCEPT
Summary: Ser/Thr kinase activity inferred by curator. Core MF.
Reason: Core molecular function.
GO:0004707 MAP kinase activity
IDA
PMID:15027896
Angiotensin II-induced ERK1/ERK2 activation and protein synt...
ACCEPT
Summary: Direct evidence of ERK1/2 (MAP kinase) activation in mesangial cells. Core MF.
Reason: Core molecular function with direct evidence.
GO:0005524 ATP binding
IDA
PMID:15027896
Angiotensin II-induced ERK1/ERK2 activation and protein synt...
ACCEPT
Summary: ATP binding/use directly demonstrated. Core MF. The deep research independently describes an in vitro kinase assay using active TEY-phosphorylated ERK2 and an ATP-gamma-S analog.
Reason: Core molecular function with direct experimental support.
GO:0006468 protein phosphorylation
IDA
PMID:15027896
Angiotensin II-induced ERK1/ERK2 activation and protein synt...
KEEP AS NON CORE
Summary: Generic protein phosphorylation (catalytic output) with direct evidence.
Reason: Generic BP output of kinase activity; the MF terms capture this more precisely. Non-core.
GO:0045727 positive regulation of translation
IMP
PMID:15027896
Angiotensin II-induced ERK1/ERK2 activation and protein synt...
KEEP AS NON CORE
Summary: ERK promotes protein synthesis in mesangial cells; downstream consequence.
Reason: Downstream regulatory consequence; non-core.
GO:0000165 MAPK cascade
IMP
PMID:17310240
Growth factor-induced MAPK network topology shapes Erk respo...
ACCEPT
Summary: ERK response within the growth-factor-induced MAPK network. Core BP.
Reason: Core biological process (generic parent of ERK1/2 cascade) with experimental support.
GO:0031663 lipopolysaccharide-mediated signaling pathway
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK acts downstream of LPS/TLR signaling; stimulus-specific pathway context inferred by orthology.
Reason: Stimulus-specific pathway context; non-core.
GO:0032496 response to lipopolysaccharide
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Stimulus-specific cellular response inferred by orthology.
Reason: Stimulus-specific response; non-core.
GO:0043330 response to exogenous dsRNA
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Stimulus-specific cellular response inferred by orthology.
Reason: Stimulus-specific response; non-core.
GO:0045596 negative regulation of cell differentiation
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK signaling modulates differentiation; a pleiotropic, context-dependent downstream process inferred by orthology.
Reason: Context-dependent downstream process; non-core.
GO:0008284 positive regulation of cell population proliferation
IEP
PMID:15583728
The indazole derivative YD-3 inhibits thrombin-induced vascu...
KEEP AS NON CORE
Summary: ERK1/2 drives proliferation (thrombin-induced VSMC proliferation context). A major but downstream pleiotropic outcome of cascade activity.
Reason: Major downstream consequence of ERK activity, but context-dependent and not the protein's core molecular role. Kept as non-core.
GO:0030335 positive regulation of cell migration
IEP
PMID:15917991
Reactive oxygen species and ERK 1/2 mediate monocyte chemota...
KEEP AS NON CORE
Summary: ERK1/2 promotes cell migration (MCP-1-stimulated VSMC migration). A downstream pleiotropic outcome.
Reason: Downstream consequence of ERK activity; non-core.
GO:0043627 response to estrogen
IDA
PMID:11751611
Impact of progestins on estrogen-induced neuroprotection: sy...
KEEP AS NON CORE
Summary: ERK2 activation in estrogen-induced neuroprotection; stimulus-specific response.
Reason: Stimulus-specific response; non-core.
GO:0097237 cellular response to toxic substance
IDA
PMID:12487375
Acrolein activates mitogen-activated protein kinase signal t...
KEEP AS NON CORE
Summary: ERK activation by acrolein in vascular smooth muscle; stimulus-specific response.
Reason: Stimulus-specific response; non-core.
GO:0016301 kinase activity
ISO
GO_REF:0000121
MARK AS OVER ANNOTATED
Summary: Generic parent of the specific kinase MF terms.
Reason: Over-general MF; the specific MAP kinase / protein serine/threonine kinase terms are present and preferred.
Propagation Review
Root cause: TERM SCOPING PROBLEM
Failure modes: GRANULARITY MISMATCH
Sources checked:
MGI:MGI:1346858 · mouse Mapk1 SOURCE STALE OR MISSING
The current mouse Mapk1 record carries no generic kinase activity annotation (QuickGO, checked 2026-08); its evidence is for MAP kinase and protein serine/threonine kinase activity.
GO:0019858 cytosine metabolic process
ISO
GO_REF:0000121
REMOVE
Summary: ERK2 has no established role in cytosine metabolism as a function it executes; the donor mouse Mapk1 annotation is experimentally grounded (IDA, PMID:15284227), but the term does not describe an ERK2 function.
Reason: ERK2 is a protein kinase; it does not execute a function in pyrimidine/cytosine metabolism, so the term fails the review standard for a process annotation regardless of the donor evidence. Source tracing shows the mouse donor annotation rests on a real IDA (PMID:15284227, an MKP3/CK2alpha study), so the defect is the term choice/transfer, not a fabricated source; REMOVE stands on the biology.
Propagation Review
Root cause: PROPAGATION BAD
Sources checked:
MGI:MGI:1346858 · mouse Mapk1 SUPPORTS SOURCE BUT NOT TARGET
The mouse donor does carry this term (IDA, PMID:15284227, a study of MKP3 and CK2alpha), but nothing in ERK2 biology connects it to cytosine metabolism, so the transfer is unsafe for the rat gene.
GO:0019233 sensory perception of pain
IMP
PMID:11356865
Metabotropic glutamate receptor subtypes 1 and 5 are activat...
KEEP AS NON CORE
Summary: ERK signaling required for inflammatory pain (via mGluR1/5); an organism-level physiological process downstream of the cascade.
Reason: Physiological process; non-core.
GO:0006974 DNA damage response
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: ERK signaling participates in DNA damage responses in some contexts; downstream/context-specific.
Reason: Context-specific downstream process; non-core.
GO:0004707 MAP kinase activity
TAS
PMID:9779826
Expression of mitogen-activated protein kinase pathways duri...
ACCEPT
Summary: MAP kinase activity (TAS, postnatal heart development study). Core MF.
Reason: Core molecular function.
GO:0006468 protein phosphorylation
TAS
PMID:9779826
Expression of mitogen-activated protein kinase pathways duri...
KEEP AS NON CORE
Summary: Generic protein phosphorylation (catalytic output, TAS).
Reason: Generic BP output; non-core relative to MF terms.
GO:0016301 kinase activity
TAS
PMID:11687663
Cyclic changes in estradiol regulate synaptic plasticity thr...
MARK AS OVER ANNOTATED
Summary: Generic kinase activity (TAS). Over-general.
Reason: Over-general MF; specific kinase terms preferred.
GO:0035556 intracellular signal transduction
IDA
PMID:12072413
1alpha,25-dihydroxyvitamin D(3) and 24R,25-dihydroxyvitamin ...
KEEP AS NON CORE
Summary: ERK1/2 in vitamin-D-modulated chondrocyte signaling; generic signal-transduction parent.
Reason: Generic BP parent; the ERK1/2 cascade term is preferred. Non-core.
GO:0035556 intracellular signal transduction
TAS
PMID:9779826
Expression of mitogen-activated protein kinase pathways duri...
KEEP AS NON CORE
Summary: Generic intracellular signal transduction (TAS).
Reason: Generic BP parent; non-core.
GO:0004672 protein kinase activity
ISO
GO_REF:0000121
MARK AS OVER ANNOTATED
Summary: Generic parent of the specific kinase MF terms (ISO duplicate).
Reason: Over-general MF; specific MAP kinase / Ser/Thr kinase terms preferred.
Propagation Review
Root cause: TERM SCOPING PROBLEM
Failure modes: GRANULARITY MISMATCH
Sources checked:
MGI:MGI:1346858 · mouse Mapk1 SUPPORTS SOURCE BUT NOT TARGET
The mouse donor carries the term by IDA (PMID:14744933), but the specific MAP kinase and serine/threonine kinase terms are already present on the rat gene and are preferred.
GO:0001784 phosphotyrosine residue binding
ISO
GO_REF:0000121
MARK AS OVER ANNOTATED
Summary: This implies ERK2 binds phosphotyrosine residues. ERK2 does engage phosphorylated docking partners, but a dedicated phosphotyrosine-binding MF is not an established ERK2 function and likely over-annotates by orthology transfer.
Reason: Not an established ERK2 molecular function; ERK2 lacks a canonical phosphotyrosine-binding module (e.g., SH2/PTB). Likely an erroneous/over-broad orthology transfer.
Propagation Review
Root cause: PROPAGATION BAD
Failure modes: GRANULARITY MISMATCH
Sources checked:
MGI:MGI:1346858 · mouse Mapk1 SUPPORTS SOURCE BUT NOT TARGET
The mouse donor support is an IMP (PMID:14636584) reflecting engagement with phosphorylated partners; ERK2 has no canonical phosphotyrosine-binding module, so a dedicated molecular function over-reads the donor.
GO:0009887 animal organ morphogenesis
ISO
GO_REF:0000121
KEEP AS NON CORE
Summary: Generic developmental morphogenesis process inferred by orthology; pleiotropic and downstream.
Reason: Generic developmental process; non-core.

Core Functions

ERK2 is the terminal serine/threonine protein kinase of the canonical RAS-RAF-MEK-ERK (ERK1/2) MAPK cascade. Activated by MEK1/2-mediated dual phosphorylation of its TEY activation-loop motif, it uses ATP to phosphorylate Ser/Thr-Pro motifs on a broad set of cytoplasmic and nuclear substrates, transducing signals from growth factor receptors and other stimuli into cellular responses such as proliferation and differentiation.

Molecular Function:
MAP kinase activity
Cellular Locations:
Supporting Evidence:
  • PMID:15027896
    Angiotensin II-induced ERK1/ERK2 activation
  • file:rat/Mapk1/Mapk1-deep-research-falcon.md
    Mapk1 encodes ERK2**, a serine/threonine MAP kinase in the canonical RAS→RAF→MEK→ERK cascade
  • file:rat/Mapk1/Mapk1-deep-research-falcon.md
    ERK1/2 substrates contain a **Ser/Thr‑Pro** consensus

ERK2 binds ATP in its kinase domain and transfers the gamma-phosphate to Ser/Thr residues of substrate proteins; ATP binding is required for the phosphotransfer reaction that underlies all ERK2 signaling.

Molecular Function:
ATP binding
Directly Involved In:
Cellular Locations:
Supporting Evidence:
  • PMID:15027896
    Angiotensin II-induced ERK1/ERK2 activation and protein synthesis are redox-dependent in glomerular mesangial cells
  • file:rat/Mapk1/Mapk1-deep-research-falcon.md
    an in vitro kinase assay with active TEY-phosphorylated ERK2 and an ATPγS analog

References

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Suggested Questions for Experts

Q: To what extent are the many ISO-inferred developmental and tissue-specific process annotations (e.g., thyroid/thymus/face/lung development) representative of an endogenous rat Mapk1 requirement versus general ERK1/2 pathway pleiotropy shared redundantly with Mapk3/ERK1?

Q: Which ERK2 substrates and localized signaling pools are most relevant in rat-specific physiology (e.g., the IMCD EGF-ERK network and NHE1/SLC9A1 phosphorylation), and how does ERK2 nuclear translocation versus cytoplasmic sequestration (PEA-15) shape these outputs?

Suggested Experiments

Experiment: Use compartment-restricted ERK2 (constitutively nuclear vs. cytoplasm-tethered) in a relevant rat cell system and perform RNA-seq plus phosphoproteomics to dissect which downstream processes require nuclear ERK2 versus cytoplasmic ERK2 activity.

Hypothesis: Endogenous rat ERK2 (Mapk1) activation drives a defined transcriptional program through nuclear translocation, separable from cytoplasmic substrate phosphorylation.

Deep Research

Falcon

(Mapk1-deep-research-falcon.md)

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📚 Additional Documentation

Bioreason Rl Predictions

(Mapk1-bioreason-rl-predictions.md)

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Bioreason Rl Review

(Mapk1-bioreason-rl-review.md)

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📄 View Raw YAML

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