CDK5

UniProt ID: Q00535
Organism: Homo sapiens
Review Status: COMPLETE
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Gene Description

CDK5 encodes a proline-directed serine/threonine kinase activated by CDK5R1/p35, CDK5R1/p25, and CDK5R2/p39 family regulators, with major functions in neuronal development, neurite and axon growth, cytoskeletal and dendritic-spine dynamics, synaptic vesicle cycling, synaptic plasticity, and p25-linked neurodegenerative apoptosis as a stress/disease context. Human CDK5 also regulates induced neuronal autophagy through phosphorylation of SH3GLB1/endophilin B1. Beyond the nervous system, CDK5 partners with cyclin B1 in proliferating cells and is active during mitosis, where it acts as a canonical CDK-cyclin kinase required for mitotic fidelity.

Existing Annotations Review

GO Term Evidence Action Reason
GO:0000307 cyclin-dependent protein kinase holoenzyme complex
IBA
GO_REF:0000033
ACCEPT
Summary: cyclin-dependent protein kinase holoenzyme complex is a supported CDK5 kinase-complex annotation.
Reason: CDK5 functions as a catalytic subunit in heterodimeric CDK5R-containing kinase complexes.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0005737 cytoplasm
IBA
GO_REF:0000033
ACCEPT
Summary: cytoplasm is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0004693 cyclin-dependent protein serine/threonine kinase activity
IBA
GO_REF:0000033
ACCEPT
Summary: cyclin-dependent protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:1901987 regulation of cell cycle phase transition
IBA
GO_REF:0000033
ACCEPT
Summary: regulation of cell cycle phase transition is a core CDK5 process. CDK5 was long classified as an atypical CDK with no direct cell-cycle role, but Zheng et al. 2024 (Nature) demonstrated that CDK5 is active during mitosis, partners with cyclin B1, and is required for mitotic fidelity - a direct, enzymatically-mediated function rather than over-propagation.
Reason: Experimentally established direct function- CDK5-cyclin B1 acts as a canonical CDK-cyclin complex that phosphorylates mitotic substrates to ensure mitotic fidelity (Zheng et al. 2024, PMID:39232161). This is a bona fide core CDK5 kinase function operating in proliferating cells via cyclin B1, complementary to (not subordinate to) its p35/p39-activated neuronal kinase role.
Supporting Evidence:
PMID:39232161
CDK5 is active throughout mitosis
PMID:39232161
cyclin B1 is a mitotic co-factor of CDK5
file:human/CDK5/CDK5-deep-research-falcon.md
CDK5 can form a complex with cyclin B1 and regulate mitotic fidelity, challenging the traditional view that CDK5 has no cell cycle function
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
GO:0007409 axonogenesis
IBA
GO_REF:0000033
ACCEPT
Summary: axonogenesis is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0048489 synaptic vesicle transport
IBA
GO_REF:0000033
ACCEPT
Summary: synaptic vesicle transport is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0051402 neuron apoptotic process
IBA
GO_REF:0000033
KEEP AS NON CORE
Summary: Keep neuron apoptotic process as a non-core p25-linked neurotoxicity/stress annotation rather than canonical core CDK5 neuronal kinase biology.
Reason: The strongest apoptosis evidence is pathological calpain cleavage of CDK5R1/p35 to p25, causing constitutive and mislocalized CDK5 activity in neurodegenerative stress models; this is not the core developmental/synaptic CDK5 function.
Supporting Evidence:
PMID:10604467
p25, a truncated form of p35, accumulates in neurons in the brains of patients with Alzheimer's disease
PMID:10604467
p25/Cdk5 complex in cultured primary neurons induces cytoskeletal disruption, morphological degeneration and apoptosis
PMID:10604467
cleavage of p35, followed by accumulation of p25, may be involved in the pathogenesis of cytoskeletal abnormalities and neuronal death in neurodegenerative diseases
GO:0004672 protein kinase activity
IEA
GO_REF:0000120
MODIFY
Summary: protein kinase activity is correct but too broad for CDK5.
Reason: Replace the broad kinase parent with the more informative cyclin-dependent protein serine/threonine kinase activity term.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004674 protein serine/threonine kinase activity
IEA
GO_REF:0000120
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0005524 ATP binding
IEA
GO_REF:0000002
ACCEPT
Summary: ATP binding is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0005634 nucleus
IEA
GO_REF:0000120
ACCEPT
Summary: nucleus is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0005737 cytoplasm
IEA
GO_REF:0000120
ACCEPT
Summary: cytoplasm is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0005886 plasma membrane
IEA
GO_REF:0000044
ACCEPT
Summary: plasma membrane is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0007409 axonogenesis
IEA
GO_REF:0000117
ACCEPT
Summary: axonogenesis is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0014069 postsynaptic density
IEA
GO_REF:0000044
ACCEPT
Summary: Accept postsynaptic density as a supported synaptic CDK5 localization.
Reason: UniProt gives a specific postsynaptic density localization by similarity, consistent with CDK5 synaptic substrate regulation.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Postsynaptic density
GO:0030027 lamellipodium
IEA
GO_REF:0000120
ACCEPT
Summary: Accept lamellipodium as a specific CDK5 cell-projection localization supported by UniProt.
Reason: The UniProt subcellular-location line explicitly includes lamellipodium in the cell-projection context.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Perikaryon. Cell projection, lamellipodium
GO:0030426 growth cone
IEA
GO_REF:0000044
ACCEPT
Summary: growth cone is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0043204 perikaryon
IEA
GO_REF:0000044
ACCEPT
Summary: Accept perikaryon as a specific CDK5 neuronal-cell-body localization supported by UniProt.
Reason: The UniProt subcellular-location line explicitly includes perikaryon.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Perikaryon. Cell projection, lamellipodium
GO:0045202 synapse
IEA
GO_REF:0000044
ACCEPT
Summary: synapse is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0051649 establishment of localization in cell
IEA
GO_REF:0000117
KEEP AS NON CORE
Summary: establishment of localization in cell is a secondary or broad CDK5 process annotation.
Reason: The term reflects a true downstream or disease/stress context, but it is broader or less central than CDK5 kinase activity and neuronal/synaptic substrate regulation.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0051726 regulation of cell cycle
IEA
GO_REF:0000117
ACCEPT
Summary: regulation of cell cycle is a core CDK5 process. Historically CDK5 was thought to lack a direct cell-cycle role; Zheng et al. 2024 (Nature) showed CDK5 is active during mitosis and, with cyclin B1, is required for mitotic fidelity, establishing this as a genuine direct function.
Reason: Experimentally established by the demonstration that CDK5 forms a functional CDK-cyclin complex with cyclin B1 and ensures mitotic fidelity (Zheng et al. 2024, PMID:39232161). Treated as a core CDK5 kinase function in proliferating cells, complementary to its p35/p39-activated neuronal/synaptic signaling.
Supporting Evidence:
PMID:39232161
CDK5 is active throughout mitosis
PMID:39232161
cyclin B1 is a mitotic co-factor of CDK5
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
GO:0098793 presynapse
IEA
GO_REF:0000120
KEEP AS NON CORE
Summary: Keep presynapse as non-core synaptic localization context.
Reason: The accessible UniProt text supports synapse broadly, but not presynapse specifically; the core localization should remain broader synapse/postsynaptic density/growth cone/neuron projection contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Synapse
GO:0106310 protein serine kinase activity
IEA
GO_REF:0000116
MODIFY
Summary: Protein serine kinase activity is too narrow/incomplete for CDK5.
Reason: CDK5 phosphorylates both serine and threonine residues, so protein serine/threonine kinase activity is the better molecular-function term.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0005515 protein binding
IPI
PMID:14521924
Apoptosis-associated tyrosine kinase is a Cdk5 activator p35...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:15689152
Mechanism of CDK5/p25 binding by CDK inhibitors.
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:15890360
Molecular basis for the specificity of p27 toward cyclin-dep...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:17078951
PKA modulates GSK-3beta- and cdk5-catalyzed phosphorylation ...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:20133653
No difference in kinetics of tau or histone phosphorylation ...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:20559324
Cables1 protects p63 from proteasomal degradation to ensure ...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:21220307
Phosphorylation of glutamyl-prolyl tRNA synthetase by cyclin...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:22078880
Adipocyte NCoR knockout decreases PPARΞ³ phosphorylation and ...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:23455922
Interlaboratory reproducibility of large-scale human protein...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:23543736
Ubiquitin C-terminal hydrolase L1 (UCH-L1) acts as a novel p...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:23602568
The protein interaction landscape of the human CMGC kinase g...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:25416956
A proteome-scale map of the human interactome network.
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:25852190
Integrative analysis of kinase networks in TRAIL-induced apo...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:26871637
Widespread Expansion of Protein Interaction Capabilities by ...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:27107012
Pooled-matrix protein interaction screens using Barcode Fusi...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:28514442
Architecture of the human interactome defines protein commun...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:30833792
A protein-interaction network of interferon-stimulated genes...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:32296183
A reference map of the human binary protein interactome.
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:32707033
Kinase Interaction Network Expands Functional and Disease Ro...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:32812023
Phosphorylated tau interactome in the human Alzheimer's dise...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:32814053
Interactome Mapping Provides a Network of Neurodegenerative ...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:33961781
Dual proteome-scale networks reveal cell-specific remodeling...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:34591612
A protein interaction landscape of breast cancer.
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:35016035
Identification and functional characterization of transcript...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:35063084
Tau interactome maps synaptic and mitochondrial processes as...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005515 protein binding
IPI
PMID:35271311
OpenCell: Endogenous tagging for the cartography of human ce...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0002039 p53 binding
IEA
GO_REF:0000107
KEEP AS NON CORE
Summary: p53 binding is a specific substrate/regulator binding context, not the core molecular function.
Reason: This binding annotation is more specific than generic protein binding, but CDK5 should primarily be represented by kinase activity and substrate phosphorylation/regulation terms.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Interacts with P53/TP53 in neurons
GO:0005176 ErbB-2 class receptor binding
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: ErbB-2 class receptor binding overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0005829 cytosol
IEA
GO_REF:0000107
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0016533 protein kinase 5 complex
IEA
GO_REF:0000120
ACCEPT
Summary: protein kinase 5 complex is a supported CDK5 kinase-complex annotation.
Reason: CDK5 functions as a catalytic subunit in heterodimeric CDK5R-containing kinase complexes.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0030175 filopodium
IEA
GO_REF:0000107
KEEP AS NON CORE
Summary: Keep filopodium as non-core fine cell-projection localization context.
Reason: The accessible evidence supports CDK5 at cell projections and lamellipodia/growth cones, but not a specific filopodium localization as a core CDK5 compartment.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Perikaryon. Cell projection, lamellipodium
IEA
GO_REF:0000107
ACCEPT
Summary: axon is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0030547 signaling receptor inhibitor activity
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: signaling receptor inhibitor activity overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0030549 acetylcholine receptor activator activity
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: acetylcholine receptor activator activity overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0043125 ErbB-3 class receptor binding
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: ErbB-3 class receptor binding overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0051879 Hsp90 protein binding
IEA
GO_REF:0000107
MARK AS OVER ANNOTATED
Summary: Hsp90 protein binding overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0051966 regulation of synaptic transmission, glutamatergic
IEA
GO_REF:0000107
ACCEPT
Summary: regulation of synaptic transmission, glutamatergic is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0061001 regulation of dendritic spine morphogenesis
IEA
GO_REF:0000107
ACCEPT
Summary: regulation of dendritic spine morphogenesis is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:1903076 regulation of protein localization to plasma membrane
IEA
GO_REF:0000107
ACCEPT
Summary: regulation of protein localization to plasma membrane is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0000307 cyclin-dependent protein kinase holoenzyme complex
IPI
PMID:16039528
Defining Cdk5 ligand chemical space with small molecule inhi...
ACCEPT
Summary: cyclin-dependent protein kinase holoenzyme complex is a supported CDK5 kinase-complex annotation.
Reason: CDK5 functions as a catalytic subunit in heterodimeric CDK5R-containing kinase complexes.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0016533 protein kinase 5 complex
IPI
PMID:15689152
Mechanism of CDK5/p25 binding by CDK inhibitors.
ACCEPT
Summary: protein kinase 5 complex is a supported CDK5 kinase-complex annotation.
Reason: CDK5 functions as a catalytic subunit in heterodimeric CDK5R-containing kinase complexes.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0016533 protein kinase 5 complex
IPI
PMID:16039528
Defining Cdk5 ligand chemical space with small molecule inhi...
ACCEPT
Summary: protein kinase 5 complex is a supported CDK5 kinase-complex annotation.
Reason: CDK5 functions as a catalytic subunit in heterodimeric CDK5R-containing kinase complexes.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0005654 nucleoplasm
IDA
GO_REF:0000052
KEEP AS NON CORE
Summary: nucleoplasm is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005886 plasma membrane
IDA
GO_REF:0000052
ACCEPT
Summary: plasma membrane is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0004674 protein serine/threonine kinase activity
TAS
Reactome:R-HSA-399944
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004674 protein serine/threonine kinase activity
TAS
Reactome:R-HSA-8863007
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004674 protein serine/threonine kinase activity
TAS
Reactome:R-HSA-8863011
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004674 protein serine/threonine kinase activity
TAS
Reactome:R-HSA-8863014
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004693 cyclin-dependent protein serine/threonine kinase activity
TAS
Reactome:R-HSA-180047
ACCEPT
Summary: cyclin-dependent protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004674 protein serine/threonine kinase activity
IDA
PMID:24607229
Memory enhancement by targeting Cdk5 regulation of NR2B.
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0030547 signaling receptor inhibitor activity
IMP
PMID:24607229
Memory enhancement by targeting Cdk5 regulation of NR2B.
MARK AS OVER ANNOTATED
Summary: signaling receptor inhibitor activity overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0035255 ionotropic glutamate receptor binding
IPI
PMID:24607229
Memory enhancement by targeting Cdk5 regulation of NR2B.
KEEP AS NON CORE
Summary: ionotropic glutamate receptor binding is a specific substrate/regulator binding context, not the core molecular function.
Reason: This binding annotation is more specific than generic protein binding, but CDK5 should primarily be represented by kinase activity and substrate phosphorylation/regulation terms.
Supporting Evidence:
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
GO:0005634 nucleus
EXP
PMID:12691662
Cdk5-mediated inhibition of the protective effects of transc...
ACCEPT
Summary: nucleus is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0005737 cytoplasm
EXP
PMID:12691662
Cdk5-mediated inhibition of the protective effects of transc...
ACCEPT
Summary: cytoplasm is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0005886 plasma membrane
EXP
PMID:17009320
cdk5 modulates beta- and delta-catenin/Pin1 interactions in ...
ACCEPT
Summary: plasma membrane is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0014069 postsynaptic density
ISS
GO_REF:0000024
ACCEPT
Summary: Accept postsynaptic density as a supported synaptic CDK5 localization.
Reason: UniProt gives a specific postsynaptic density localization by similarity, consistent with CDK5 synaptic substrate regulation.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Postsynaptic density
GO:0045202 synapse
ISS
GO_REF:0000024
ACCEPT
Summary: synapse is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0099533 positive regulation of presynaptic cytosolic calcium concentration
ISS
GO_REF:0000024
ACCEPT
Summary: positive regulation of presynaptic cytosolic calcium concentration is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:1903234 negative regulation of calcium ion-dependent exocytosis of neurotransmitter
ISS
GO_REF:0000024
ACCEPT
Summary: negative regulation of calcium ion-dependent exocytosis of neurotransmitter is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0004674 protein serine/threonine kinase activity
TAS
PMID:17491008
Microtubule association of the neuronal p35 activator of Cdk...
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0030036 actin cytoskeleton organization
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: actin cytoskeleton organization is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0005515 protein binding
IPI
PMID:8090221
p35 is a neural-specific regulatory subunit of cyclin-depend...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0048156 tau protein binding
NAS
PMID:28386764
Roles of tau protein in health and disease.
KEEP AS NON CORE
Summary: tau protein binding is a specific substrate/regulator binding context, not the core molecular function.
Reason: This binding annotation is more specific than generic protein binding, but CDK5 should primarily be represented by kinase activity and substrate phosphorylation/regulation terms.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
MAPT/TAU, MAP2, MAP1B
file:human/CDK5/CDK5-uniprot.txt
microtubule-binding proteins (e.g. MAPT/TAU, MAP2, MAP1B)
GO:0050321 tau-protein kinase activity
NAS
PMID:28386764
Roles of tau protein in health and disease.
ACCEPT
Summary: tau-protein kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
MAPT/TAU, MAP2, MAP1B
file:human/CDK5/CDK5-uniprot.txt
microtubule-binding proteins (e.g. MAPT/TAU, MAP2, MAP1B)
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0016020 membrane
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: membrane is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0030426 growth cone
ISS
GO_REF:0000024
ACCEPT
Summary: growth cone is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0043005 neuron projection
ISS
GO_REF:0000024
ACCEPT
Summary: neuron projection is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0004674 protein serine/threonine kinase activity
NAS
PMID:28386764
Roles of tau protein in health and disease.
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0051966 regulation of synaptic transmission, glutamatergic
ISS
GO_REF:0000024
ACCEPT
Summary: regulation of synaptic transmission, glutamatergic is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0005737 cytoplasm
ISS
GO_REF:0000024
ACCEPT
Summary: cytoplasm is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0005874 microtubule
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: microtubule is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
PMID:17491008
p35 binds directly to alpha/beta-tubulin and microtubules
PMID:17491008
Microtubule polymers but not the alpha/beta-tubulin heterodimer block p35 interaction with Cdk5
GO:0008017 microtubule binding
TAS NOT
PMID:17491008
Microtubule association of the neuronal p35 activator of Cdk...
MARK AS OVER ANNOTATED
Summary: Microtubule binding is over-attributed to CDK5 itself.
Reason: The cited evidence supports microtubule binding by the p35/CDK5R1 activator and regulation of CDK5-p35 activity by microtubules, not direct CDK5 microtubule-binding as its molecular function.
Supporting Evidence:
PMID:17491008
p35 binds directly to alpha/beta-tubulin and microtubules
PMID:17491008
Microtubule polymers but not the alpha/beta-tubulin heterodimer block p35 interaction with Cdk5
GO:0000226 microtubule cytoskeleton organization
TAS
PMID:17491008
Microtubule association of the neuronal p35 activator of Cdk...
ACCEPT
Summary: microtubule cytoskeleton organization is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0031175 neuron projection development
TAS
PMID:17491008
Microtubule association of the neuronal p35 activator of Cdk...
ACCEPT
Summary: neuron projection development is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0048167 regulation of synaptic plasticity
TAS
PMID:24607229
Memory enhancement by targeting Cdk5 regulation of NR2B.
ACCEPT
Summary: regulation of synaptic plasticity is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:1903076 regulation of protein localization to plasma membrane
ISS
GO_REF:0000024
ACCEPT
Summary: regulation of protein localization to plasma membrane is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:1904646 cellular response to amyloid-beta
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: cellular response to amyloid-beta is a secondary or broad CDK5 process annotation.
Reason: The term reflects a true downstream or disease/stress context, but it is broader or less central than CDK5 kinase activity and neuronal/synaptic substrate regulation.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0005654 nucleoplasm
TAS
Reactome:R-HSA-8863014
KEEP AS NON CORE
Summary: nucleoplasm is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005654 nucleoplasm
TAS
Reactome:R-HSA-8863587
KEEP AS NON CORE
Summary: nucleoplasm is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005654 nucleoplasm
TAS
Reactome:R-HSA-6805276
KEEP AS NON CORE
Summary: nucleoplasm is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0016241 regulation of macroautophagy
TAS
PMID:21499257
Cdk5-mediated phosphorylation of endophilin B1 is required f...
ACCEPT
Summary: Regulation of macroautophagy is a supported PN-relevant CDK5 substrate-specific process.
Reason: Human/neuron evidence shows CDK5 phosphorylates SH3GLB1/endophilin B1 and is required for induced autophagy in starved neurons and Parkinson disease models.
Supporting Evidence:
PMID:21499257
unexpected role for Cdk5 in the regulation of induced autophagy in neurons
PMID:21499257
autophagy induction in starved neurons
file:human/CDK5/CDK5-uniprot.txt
Phosphorylation of SH3GLB1 is required for autophagy induction in starved neurons
GO:1903421 regulation of synaptic vesicle recycling
NAS
PMID:22745285
Synaptic vesicle pools and dynamics.
ACCEPT
Summary: regulation of synaptic vesicle recycling is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0045861 negative regulation of proteolysis
IMP
PMID:24548080
CDK5 protects from caspase-induced Ataxin-3 cleavage and neu...
KEEP AS NON CORE
Summary: negative regulation of proteolysis is a secondary or broad CDK5 process annotation.
Reason: The term reflects a true downstream or disease/stress context, but it is broader or less central than CDK5 kinase activity and neuronal/synaptic substrate regulation.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0005829 cytosol
TAS
Reactome:R-HSA-399944
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005829 cytosol
TAS
Reactome:R-HSA-399951
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005829 cytosol
TAS
Reactome:R-NUL-9032945
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005829 cytosol
TAS
Reactome:R-HSA-180047
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005829 cytosol
TAS
Reactome:R-HSA-8863007
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005829 cytosol
TAS
Reactome:R-HSA-8863011
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005829 cytosol
TAS
Reactome:R-HSA-8863013
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0005829 cytosol
TAS
Reactome:R-HSA-8863587
KEEP AS NON CORE
Summary: cytosol is a broad or complex-context CDK5 localization.
Reason: This location is compatible with CDK5 biology but is less informative than CDK5 kinase-complex, synaptic, neuronal projection, and growth-cone contexts.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
GO:0048167 regulation of synaptic plasticity
ISS
GO_REF:0000024
ACCEPT
Summary: regulation of synaptic plasticity is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0001764 neuron migration
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: neuron migration is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0007268 chemical synaptic transmission
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: chemical synaptic transmission is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0007416 synapse assembly
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: synapse assembly is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0016079 synaptic vesicle exocytosis
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: synaptic vesicle exocytosis is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0030182 neuron differentiation
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: neuron differentiation is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0042981 regulation of apoptotic process
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: regulation of apoptotic process is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0048167 regulation of synaptic plasticity
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: regulation of synaptic plasticity is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0048488 synaptic vesicle endocytosis
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: synaptic vesicle endocytosis is a core CDK5 synaptic process.
Reason: CDK5 phosphorylates synaptic release, endocytosis, and NMDAR-associated substrates and regulates synaptic plasticity/neurotransmission.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
PMID:24607229
controls the receptor's cell surface expression
PMID:24607229
serine 1116 of NR2B is phosphorylated by cyclin-dependent kinase 5 (Cdk5)
PMID:24607229
increases NR2B surface levels, facilitates synaptic transmission, and improves memory formation
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0048675 axon extension
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: axon extension is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0048709 oligodendrocyte differentiation
IDA
PMID:18042622
Cdk5 regulates differentiation of oligodendrocyte precursor ...
ACCEPT
Summary: oligodendrocyte differentiation is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0051402 neuron apoptotic process
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
KEEP AS NON CORE
Summary: Keep neuron apoptotic process as a non-core p25-linked neurotoxicity/stress annotation rather than canonical core CDK5 neuronal kinase biology.
Reason: The strongest apoptosis evidence is pathological calpain cleavage of CDK5R1/p35 to p25, causing constitutive and mislocalized CDK5 activity in neurodegenerative stress models; this is not the core developmental/synaptic CDK5 function.
Supporting Evidence:
PMID:10604467
p25, a truncated form of p35, accumulates in neurons in the brains of patients with Alzheimer's disease
PMID:10604467
p25/Cdk5 complex in cultured primary neurons induces cytoskeletal disruption, morphological degeneration and apoptosis
PMID:10604467
cleavage of p35, followed by accumulation of p25, may be involved in the pathogenesis of cytoskeletal abnormalities and neuronal death in neurodegenerative diseases
GO:0051726 regulation of cell cycle
TAS
PMID:21473899
Cdk5: multitasking between physiological and pathological co...
ACCEPT
Summary: regulation of cell cycle is a core CDK5 process. Historically CDK5 was thought to lack a direct cell-cycle role; Zheng et al. 2024 (Nature) showed CDK5 is active during mitosis and, with cyclin B1, is required for mitotic fidelity, establishing this as a genuine direct function.
Reason: Experimentally established by the demonstration that CDK5 forms a functional CDK-cyclin complex with cyclin B1 and ensures mitotic fidelity (Zheng et al. 2024, PMID:39232161). Treated as a core CDK5 kinase function in proliferating cells, complementary to its p35/p39-activated neuronal/synaptic signaling.
Supporting Evidence:
PMID:39232161
CDK5 is active throughout mitosis
PMID:39232161
cyclin B1 is a mitotic co-factor of CDK5
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
GO:0061001 regulation of dendritic spine morphogenesis
ISS
GO_REF:0000024
ACCEPT
Summary: regulation of dendritic spine morphogenesis is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0004674 protein serine/threonine kinase activity
IDA
PMID:20357208
Cyclin-dependent kinase 5 modulates the transcriptional acti...
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0045892 negative regulation of DNA-templated transcription
IMP
PMID:20357208
Cyclin-dependent kinase 5 modulates the transcriptional acti...
KEEP AS NON CORE
Summary: negative regulation of DNA-templated transcription is a secondary or broad CDK5 process annotation.
Reason: The term reflects a true downstream or disease/stress context, but it is broader or less central than CDK5 kinase activity and neuronal/synaptic substrate regulation.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0004674 protein serine/threonine kinase activity
IDA
PMID:21145489
The proapoptotic function of Noxa in human leukemia cells is...
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004674 protein serine/threonine kinase activity
ISS
GO_REF:0000024
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0005176 ErbB-2 class receptor binding
ISS
GO_REF:0000024
MARK AS OVER ANNOTATED
Summary: ErbB-2 class receptor binding overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0005515 protein binding
IPI
PMID:12223541
The cyclin-dependent kinase 5 activators p35 and p39 interac...
MARK AS OVER ANNOTATED
Summary: Generic protein binding does not describe CDK5 function.
Reason: The specific function is CDK5-regulated phosphorylation in CDK5R/p35-p25-p39 complexes and substrate-specific neuronal/autophagy signaling. Generic protein binding rows should not be treated as informative GO molecular-function annotations.
GO:0005634 nucleus
ISS
GO_REF:0000024
ACCEPT
Summary: nucleus is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0016301 kinase activity
ISS
GO_REF:0000024
MODIFY
Summary: kinase activity is correct but too broad for CDK5.
Reason: Replace the broad kinase parent with the more informative cyclin-dependent protein serine/threonine kinase activity term.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0030182 neuron differentiation
ISS
GO_REF:0000024
ACCEPT
Summary: neuron differentiation is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
ISS
GO_REF:0000024
ACCEPT
Summary: axon is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0030425 dendrite
ISS
GO_REF:0000024
ACCEPT
Summary: dendrite is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0030549 acetylcholine receptor activator activity
ISS
GO_REF:0000024
MARK AS OVER ANNOTATED
Summary: acetylcholine receptor activator activity overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0031175 neuron projection development
ISS
GO_REF:0000024
ACCEPT
Summary: neuron projection development is part of core CDK5 neuronal kinase biology.
Reason: CDK5 regulates neuronal development, neurite/axon growth, cytoskeletal dynamics, synaptogenesis, oligodendrocyte differentiation, and neuronal survival/death.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0031594 neuromuscular junction
ISS
GO_REF:0000024
ACCEPT
Summary: neuromuscular junction is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0043025 neuronal cell body
ISS
GO_REF:0000024
ACCEPT
Summary: neuronal cell body is a supported CDK5 localization/context.
Reason: The localization is consistent with CDK5 neuronal kinase function across cytoplasm, nucleus, membranes, synapses, growth cones, and neuronal projections.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
SUBCELLULAR LOCATION: [Isoform 1]: Cytoplasm
file:human/CDK5/CDK5-uniprot.txt
Nucleus {ECO:0000269|PubMed:12691662}
file:human/CDK5/CDK5-uniprot.txt
Cell membrane {ECO:0000269|PubMed:17009320}
file:human/CDK5/CDK5-uniprot.txt
Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
PMID:21473899
normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
GO:0043125 ErbB-3 class receptor binding
ISS
GO_REF:0000024
MARK AS OVER ANNOTATED
Summary: ErbB-3 class receptor binding overstates a downstream/regulatory interaction as a CDK5 molecular function.
Reason: These transferred receptor/regulator-binding terms do not capture CDK5's catalytic function and are less defensible than kinase activity plus substrate-specific process annotations.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0043525 positive regulation of neuron apoptotic process
ISS
GO_REF:0000024
KEEP AS NON CORE
Summary: Keep positive regulation of neuron apoptotic process as a non-core p25-linked neurotoxicity/stress annotation rather than canonical core CDK5 neuronal kinase biology.
Reason: The strongest apoptosis evidence is pathological calpain cleavage of CDK5R1/p35 to p25, causing constitutive and mislocalized CDK5 activity in neurodegenerative stress models; this is not the core developmental/synaptic CDK5 function.
Supporting Evidence:
PMID:10604467
p25, a truncated form of p35, accumulates in neurons in the brains of patients with Alzheimer's disease
PMID:10604467
p25/Cdk5 complex in cultured primary neurons induces cytoskeletal disruption, morphological degeneration and apoptosis
PMID:10604467
cleavage of p35, followed by accumulation of p25, may be involved in the pathogenesis of cytoskeletal abnormalities and neuronal death in neurodegenerative diseases
GO:0050321 tau-protein kinase activity
ISS
GO_REF:0000024
ACCEPT
Summary: tau-protein kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
MAPT/TAU, MAP2, MAP1B
file:human/CDK5/CDK5-uniprot.txt
microtubule-binding proteins (e.g. MAPT/TAU, MAP2, MAP1B)
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
GO:0004672 protein kinase activity
TAS
PMID:1639063
A family of human cdc2-related protein kinases.
MODIFY
Summary: protein kinase activity is correct but too broad for CDK5.
Reason: Replace the broad kinase parent with the more informative cyclin-dependent protein serine/threonine kinase activity term.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004672 protein kinase activity
TAS
PMID:7834371
Expression of CDK5 (PSSALRE kinase), a neural cdc2-related p...
MODIFY
Summary: protein kinase activity is correct but too broad for CDK5.
Reason: Replace the broad kinase parent with the more informative cyclin-dependent protein serine/threonine kinase activity term.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
GO:0004674 protein serine/threonine kinase activity
TAS
PMID:1639063
A family of human cdc2-related protein kinases.
ACCEPT
Summary: protein serine/threonine kinase activity is a core CDK5 molecular function.
Reason: CDK5 is a CDK-family proline-directed serine/threonine protein kinase that uses ATP and is activated in CDK5R-containing kinase complexes; tau/MAPT and other neuronal proteins are established substrates.
Supporting Evidence:
file:human/CDK5/CDK5-uniprot.txt
Proline-directed serine/threonine-protein kinase
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
file:human/CDK5/CDK5-uniprot.txt
Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
file:human/CDK5/CDK5-uniprot.txt
Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
file:human/CDK5/CDK5-uniprot.txt
Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1

Core Functions

CDK5 is a CDK5R-activated proline-directed serine/threonine kinase that phosphorylates neuronal, synaptic, cytoskeletal, stress-response, and autophagy-associated substrates.

Supporting Evidence:
  • file:human/CDK5/CDK5-uniprot.txt
    Proline-directed serine/threonine-protein kinase
  • file:human/CDK5/CDK5-uniprot.txt
    Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
  • file:human/CDK5/CDK5-uniprot.txt
    Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
  • file:human/CDK5/CDK5-uniprot.txt
    Activated by interaction with CDK5R1 (p35) and CDK5R2 (p39)
  • file:human/CDK5/CDK5-uniprot.txt
    Heterodimer composed of a catalytic subunit CDK5 and a regulatory subunit CDK5R1
  • file:human/CDK5/CDK5-uniprot.txt
    Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
  • PMID:21473899
    normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity
  • file:human/CDK5/CDK5-uniprot.txt
    regulates neurotransmitter movements by phosphorylating substrates associated with neurotransmitter release and synapse plasticity
  • PMID:24607229
    controls the receptor's cell surface expression
  • PMID:21499257
    unexpected role for Cdk5 in the regulation of induced autophagy in neurons
  • PMID:21499257
    autophagy induction in starved neurons
  • file:human/CDK5/CDK5-uniprot.txt
    Phosphorylation of SH3GLB1 is required for autophagy induction in starved neurons

In proliferating (non-neuronal) cells CDK5 partners with cyclin B1, rather than its neuronal p35/p39 activators, and is active during mitosis; this CDK5-cyclin B1 complex behaves as a canonical CDK-cyclin kinase that phosphorylates mitotic substrates to safeguard mitotic fidelity and genome stability.

Supporting Evidence:
  • PMID:39232161
    CDK5 is active throughout mitosis
  • PMID:39232161
    cyclin B1 is a mitotic co-factor of CDK5
  • file:human/CDK5/CDK5-deep-research-falcon.md
    CDK5 can form a complex with cyclin B1 and regulate mitotic fidelity, challenging the traditional view that CDK5 has no cell cycle function

CDK5 phosphorylates MAPT/tau and other microtubule-associated neuronal substrates, contributing to cytoskeletal regulation and neurodegeneration-relevant tau biology.

Supporting Evidence:
  • file:human/CDK5/CDK5-uniprot.txt
    MAPT/TAU, MAP2, MAP1B
  • file:human/CDK5/CDK5-uniprot.txt
    microtubule-binding proteins (e.g. MAPT/TAU, MAP2, MAP1B)
  • file:human/CDK5/CDK5-uniprot.txt
    Proline-directed serine/threonine-protein kinase
  • file:human/CDK5/CDK5-uniprot.txt
    Reaction=L-seryl-[protein] + ATP = O-phospho-L-seryl-[protein] + ADP
  • file:human/CDK5/CDK5-uniprot.txt
    Reaction=L-threonyl-[protein] + ATP = O-phospho-L-threonyl-[protein]
  • file:human/CDK5/CDK5-uniprot.txt
    Regulates several neuronal development and physiological processes including neuronal survival, migration and differentiation, axonal and neurite growth, synaptogenesis, oligodendrocyte differentiation, synaptic plasticity and neurotransmission
  • PMID:21473899
    normally associated with neuronal processes such as migration, cortical layering and synaptic plasticity

References

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Suggested Questions for Experts

Q: Should human CDK5 be curated directly to basal autophagy/autophagosome maturation based on conserved Acinus regulation, or only to SH3GLB1-dependent regulation of induced macroautophagy?

Suggested experts: GO autophagy editors, CDK5 neuronal signaling experts, Drosophila autophagy experts

Q: Which CDK5 substrate-binding annotations should be retained as specific MF annotations versus represented as phosphorylation/regulatory process annotations?

Suggested experts: GO molecular-function editors, neurobiology curators

Suggested Experiments

Experiment: Test whether human CDK5 phosphorylates ACIN1 at sites corresponding to Drosophila Acinus S437 and whether this affects basal autophagy flux or autophagosome maturation in neuronal cells.

Hypothesis: The Drosophila Cdk5-Acinus basal-autophagy module is conserved only if human CDK5 directly phosphorylates ACIN1 and changes basal autophagic flux.

Type: kinase assay/autophagy flux assay

Experiment: Dissect CDK5-dependent SH3GLB1/endophilin B1 phosphorylation from other CDK5 neuronal substrates using phosphosite-specific rescue mutants in starved neurons.

Hypothesis: CDK5 regulation of macroautophagy is mediated through SH3GLB1 phosphorylation rather than a general CDK5 role in all autophagy steps.

Type: phosphosite rescue/autophagy imaging

Experiment: Using the analog-sensitive CDK5 chemical-genetic system from Zheng et al. 2024, map the mitotic CDK5-cyclin B1 phosphoproteome in non-neuronal proliferating cells and compare it to the CDK1-cyclin B1 substrate set, to determine whether CDK5 cell-cycle annotations should be refined to specific mitotic substrates/processes.

Hypothesis: CDK5-cyclin B1 phosphorylates a distinct subset of mitotic substrates that ensures chromosome segregation fidelity, separable from CDK1-cyclin B1 activity.

Type: analog-sensitive kinase phosphoproteomics

Deep Research

Falcon

(CDK5-deep-research-falcon.md)

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πŸ“š Additional Documentation

Notes

(CDK5-notes.md)

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Pn Notes

(CDK5-pn-notes.md)

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πŸ“„ View Raw YAML

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